DK117635B - Analogifremgangsmåde til fremstilling af terapeutisk virksomme 3-(piperazinoalkyl)-pyrazoler. - Google Patents

Analogifremgangsmåde til fremstilling af terapeutisk virksomme 3-(piperazinoalkyl)-pyrazoler.

Info

Publication number
DK117635B
DK117635B DK329967AA DK329967A DK117635B DK 117635 B DK117635 B DK 117635B DK 329967A A DK329967A A DK 329967AA DK 329967 A DK329967 A DK 329967A DK 117635 B DK117635 B DK 117635B
Authority
DK
Denmark
Prior art keywords
piperazinoalkyl
pyrazoles
preparation
therapeutically active
analogous process
Prior art date
Application number
DK329967AA
Other languages
English (en)
Inventor
E Ag Merck
Original Assignee
E Ag Merck
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E Ag Merck filed Critical E Ag Merck
Publication of DK117635B publication Critical patent/DK117635B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Catalysts (AREA)
DK329967AA 1966-07-02 1967-06-26 Analogifremgangsmåde til fremstilling af terapeutisk virksomme 3-(piperazinoalkyl)-pyrazoler. DK117635B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE1620016A DE1620016C3 (de) 1966-07-02 1966-07-02 3-{Piperazinoalkyl)-pyrazole und Verfahren zu ihrer Herstellung

Publications (1)

Publication Number Publication Date
DK117635B true DK117635B (da) 1970-05-19

Family

ID=7313285

Family Applications (1)

Application Number Title Priority Date Filing Date
DK329967AA DK117635B (da) 1966-07-02 1967-06-26 Analogifremgangsmåde til fremstilling af terapeutisk virksomme 3-(piperazinoalkyl)-pyrazoler.

Country Status (14)

Country Link
US (1) US3491097A (da)
BE (1) BE700732A (da)
CH (1) CH485751A (da)
CY (1) CY622A (da)
DE (1) DE1620016C3 (da)
DK (1) DK117635B (da)
ES (1) ES342556A1 (da)
FR (1) FR6682M (da)
GB (1) GB1124710A (da)
IL (1) IL28144A (da)
MY (1) MY7200042A (da)
NL (1) NL154739B (da)
SE (1) SE345456B (da)
YU (2) YU32679B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2110568A1 (de) * 1971-03-05 1972-09-07 Merck Patent Gmbh Neue N-Acyl-(piperazinoalkyl)-pyrazole
US3960863A (en) * 1974-06-25 1976-06-01 Sankyo Company Limited Pyrido[1,2-a]pyrimidinone derivatives
US3941881A (en) * 1975-03-14 1976-03-02 American Cyanamid Company Novel 3 or 5-aminopyrazolium salts and fungicidal use thereof
DE2835158A1 (de) * 1978-08-10 1980-02-21 Bayer Ag Substituierte pyrazol-derivate sowie verfahren zu ihrer herstellung
DE4425146A1 (de) * 1994-07-15 1996-01-18 Basf Ag Verwendung heterocyclischer Verbindungen
DE19728996A1 (de) 1997-07-07 1999-01-14 Basf Ag Triazolverbindungen und deren Verwendung
MXPA04012959A (es) * 2002-06-29 2005-05-16 Zentaris Gmbh Arilcarbonilpiperacinas y heteroarilcarbonilpiperacinas y su uso para tratamiento de enfermedades de tumor benigno y maligno.
KR100868353B1 (ko) * 2007-03-08 2008-11-12 한국화학연구원 도파민 d4 수용체 길항제인 신규 피페라지닐프로필피라졸유도체, 이의 제조방법 및 이를 포함하는 약학적 조성물

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2329680A (en) * 1943-01-30 1943-09-14 American Cyanamid Co Defoliation
BE485737A (da) * 1947-11-12
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
CH485751A (de) 1970-02-15
YU261972A (en) 1974-10-31
NL154739B (nl) 1977-10-17
YU32679B (en) 1975-04-30
NL6709008A (da) 1968-01-03
MY7200042A (en) 1972-12-31
CY622A (en) 1971-11-27
FR6682M (da) 1969-02-03
US3491097A (en) 1970-01-20
BE700732A (da) 1968-01-02
DE1620016B2 (de) 1979-01-04
DE1620016A1 (de) 1970-02-12
IL28144A (en) 1972-04-27
SE345456B (da) 1972-05-29
GB1124710A (en) 1968-08-21
DE1620016C3 (de) 1979-08-30
YU261772A (en) 1974-10-31
YU32681B (en) 1975-04-30
ES342556A1 (es) 1968-10-16

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