DK1005859T3 - Fremgangsmåde til fremstilling af dispergerbare sterol- og stanolforbindelser - Google Patents

Fremgangsmåde til fremstilling af dispergerbare sterol- og stanolforbindelser

Info

Publication number
DK1005859T3
DK1005859T3 DK99309492T DK99309492T DK1005859T3 DK 1005859 T3 DK1005859 T3 DK 1005859T3 DK 99309492 T DK99309492 T DK 99309492T DK 99309492 T DK99309492 T DK 99309492T DK 1005859 T3 DK1005859 T3 DK 1005859T3
Authority
DK
Denmark
Prior art keywords
sterol
stanol
preparation
compounds
preparing
Prior art date
Application number
DK99309492T
Other languages
English (en)
Inventor
Richard D Bruce
Brid Burruano
Michael R Hoy
Nicholas R Paquette
Original Assignee
Mcneil Ppc Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mcneil Ppc Inc filed Critical Mcneil Ppc Inc
Application granted granted Critical
Publication of DK1005859T3 publication Critical patent/DK1005859T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
DK99309492T 1998-11-30 1999-11-29 Fremgangsmåde til fremstilling af dispergerbare sterol- og stanolforbindelser DK1005859T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US09/200,623 US6242001B1 (en) 1998-11-30 1998-11-30 Method for producing dispersible sterol and stanol compounds

Publications (1)

Publication Number Publication Date
DK1005859T3 true DK1005859T3 (da) 2006-04-03

Family

ID=22742487

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99309492T DK1005859T3 (da) 1998-11-30 1999-11-29 Fremgangsmåde til fremstilling af dispergerbare sterol- og stanolforbindelser

Country Status (9)

Country Link
US (2) US6242001B1 (da)
EP (1) EP1005859B1 (da)
JP (1) JP2000191684A (da)
AT (1) ATE315381T1 (da)
CA (1) CA2290315C (da)
DE (1) DE69929411T2 (da)
DK (1) DK1005859T3 (da)
ES (1) ES2257011T3 (da)
NO (1) NO995687L (da)

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Also Published As

Publication number Publication date
US6242001B1 (en) 2001-06-05
ATE315381T1 (de) 2006-02-15
DE69929411T2 (de) 2006-08-24
NO995687D0 (no) 1999-11-19
DE69929411D1 (de) 2006-04-06
EP1005859B1 (en) 2006-01-11
CA2290315C (en) 2008-11-18
US6387411B2 (en) 2002-05-14
CA2290315A1 (en) 2000-05-30
JP2000191684A (ja) 2000-07-11
NO995687L (no) 2000-05-31
US20010012521A1 (en) 2001-08-09
ES2257011T3 (es) 2006-07-16
EP1005859A1 (en) 2000-06-07

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