DK0447891T3 - Thieno(2,3-d)pyrimidinderivater - Google Patents

Thieno(2,3-d)pyrimidinderivater

Info

Publication number
DK0447891T3
DK0447891T3 DK91103547T DK91103547T DK0447891T3 DK 0447891 T3 DK0447891 T3 DK 0447891T3 DK 91103547 T DK91103547 T DK 91103547T DK 91103547 T DK91103547 T DK 91103547T DK 0447891 T3 DK0447891 T3 DK 0447891T3
Authority
DK
Denmark
Prior art keywords
thieno
pyrimidine derivatives
pyrimidine
derivatives
Prior art date
Application number
DK91103547T
Other languages
Danish (da)
English (en)
Inventor
Karl-Heinz Dr Etzbach
Matthias Dr Wiesenfeldt
Peter Dr Hofmeister
Christoph Dr Kuenast
Karl-Otto Dr Westphalen
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Application granted granted Critical
Publication of DK0447891T3 publication Critical patent/DK0447891T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
DK91103547T 1990-03-19 1991-03-08 Thieno(2,3-d)pyrimidinderivater DK0447891T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19904008726 DE4008726A1 (de) 1990-03-19 1990-03-19 Thieno(2,3-d)pyrimidinderivate

Publications (1)

Publication Number Publication Date
DK0447891T3 true DK0447891T3 (da) 1994-05-30

Family

ID=6402524

Family Applications (1)

Application Number Title Priority Date Filing Date
DK91103547T DK0447891T3 (da) 1990-03-19 1991-03-08 Thieno(2,3-d)pyrimidinderivater

Country Status (6)

Country Link
EP (1) EP0447891B1 (fr)
JP (1) JPH04217685A (fr)
CA (1) CA2038521A1 (fr)
DE (2) DE4008726A1 (fr)
DK (1) DK0447891T3 (fr)
ES (1) ES2052296T3 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110177795A (zh) * 2016-12-26 2019-08-27 韩美药品株式会社 制备噻吩并嘧啶化合物的新方法和中间体

Families Citing this family (58)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7772432B2 (en) 1991-09-19 2010-08-10 Astrazeneca Ab Amidobenzamide derivatives which are useful as cytokine inhibitors
DE4208254A1 (de) * 1992-03-14 1993-09-16 Hoechst Ag Substituierte pyrimidine, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel und fungizid
US5869486A (en) * 1995-02-24 1999-02-09 Ono Pharmaceutical Co., Ltd. Fused pyrimidines and pyriazines as pharmaceutical compounds
ATE226936T1 (de) * 1995-08-08 2002-11-15 Ono Pharmaceutical Co Hydroxamsäurederivate verwendbar zur hemmung von gelatinase
US6232320B1 (en) * 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
GB9906566D0 (en) * 1999-03-23 1999-05-19 Zeneca Ltd Chemical compounds
DE19924668A1 (de) 1999-05-28 2000-11-30 Bayer Ag Substituierte alpha-Phenyl-beta-Ketosulfone
US6503914B1 (en) 2000-10-23 2003-01-07 Board Of Regents, The University Of Texas System Thienopyrimidine-based inhibitors of the Src family
US7427623B2 (en) 2001-09-11 2008-09-23 Smithkline Beecham Corporation 4-Amino-2,3-disubstituted thieno[2,3-d]pyrimidines and pharmacetical compositions thereof
AU2003246972A1 (en) 2002-08-06 2004-02-23 Astrazeneca Ab Condensed pyridines and pyrimidines with tie2 (tek) activity
JP2004137270A (ja) * 2002-09-26 2004-05-13 Nippon Nohyaku Co Ltd 新規除草剤、その使用方法、新規置換チエノピリミジン誘導体及びその中間体並びにそれらの製造方法
AR044743A1 (es) * 2002-09-26 2005-10-05 Nihon Nohyaku Co Ltd Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,
ES2217956B1 (es) * 2003-01-23 2006-04-01 Almirall Prodesfarma, S.A. Nuevos derivados de 4-aminotieno(2,3-d)pirimidin-6-carbonitrilo.
US7030240B2 (en) * 2003-03-31 2006-04-18 Predix Pharmaceuticals Holdings, Inc. Piperidinylamino-thieno[2,3-d] pyrimidine compounds
US7612078B2 (en) 2003-03-31 2009-11-03 Epix Delaware, Inc. Piperidinylamino-thieno[2,3-D] pyrimidine compounds
US7419978B2 (en) 2003-10-22 2008-09-02 Bristol-Myers Squibb Company Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
TW200538120A (en) * 2004-02-20 2005-12-01 Kirin Brewery Compound having TGF-beta inhibitory activity and pharmaceutical composition containing same
US7488736B2 (en) 2004-05-17 2009-02-10 Epix Delaware, Inc. Thienopyridinone compounds and methods of treatment
US7601725B2 (en) 2004-07-16 2009-10-13 Sunesis Pharmaceuticals, Inc. Thienopyrimidines useful as Aurora kinase inhibitors
US7598265B2 (en) 2004-09-30 2009-10-06 Epix Delaware, Inc. Compositions and methods for treating CNS disorders
US7576211B2 (en) 2004-09-30 2009-08-18 Epix Delaware, Inc. Synthesis of thienopyridinone compounds and related intermediates
KR20140008471A (ko) * 2004-10-21 2014-01-21 다우 아그로사이언시즈 엘엘씨 살진균 활성을 갖는 티에노-피리미딘 화합물
US7674822B2 (en) 2004-11-24 2010-03-09 Wyeth PTP1b inhibitors
EP1899353A1 (fr) * 2005-06-22 2008-03-19 DeveloGen Aktiengesellschaft Thienopyrimidines pour compositions pharmaceutiques
US7531482B2 (en) 2005-10-21 2009-05-12 Dow Agrosciences Llc Thieno-pyrimidine compounds having fungicidal activity
EP2078721B1 (fr) 2005-10-21 2014-01-22 Dow AgroSciences LLC Composés thiéno-pyrimidines ayant une activité fongicide
AR059898A1 (es) 2006-03-15 2008-05-07 Janssen Pharmaceutica Nv Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2
WO2007115822A1 (fr) 2006-04-07 2007-10-18 Develogen Aktiengesellschaft Thiénopyrimidines ayant une activité inhibitrice mnk1/mnk2 utilisées dans des compositions pharmaceutiques
BRPI0711772B8 (pt) 2006-05-22 2017-08-01 Basf Se método para combater ou controlar insetos, aracnídeos ou nematódeos; método para proteger colheitas e plantas em crescimento do ataque ou infestação de insetos, aracnídeos ou nematódeos; e método para proteger sementes dos insetos de solo e raízes e rebentos das mudas dos insetos de solo; composto e composição agricultural ou veterinária
EP1889847A1 (fr) 2006-07-10 2008-02-20 DeveloGen Aktiengesellschaft Dérivés de pyrrolopyrimidine pour applications pharmaceutiques
TW200845978A (en) 2007-03-07 2008-12-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
CN101801951B (zh) 2007-09-14 2013-11-13 杨森制药有限公司 1’,3’-二取代的-4-苯基-3,4,5,6-四氢-2h,1’h-[1,4’]二吡啶-2’-酮
EP2194788A2 (fr) 2007-10-04 2010-06-16 Dow AgroSciences LLC Compositions pesticides
DK2276346T3 (en) * 2008-04-30 2017-02-27 Nat Health Research Institutes FUSED BICYCLIC PYRIMIDINE COMPOUNDS AS AURORAKINASE INHIBITORS
US8486953B2 (en) 2008-08-26 2013-07-16 Boehringer Ingelheim International Gmbh Thienopyrimidines for pharmaceutical compositions
RU2510396C2 (ru) 2008-09-02 2014-03-27 Янссен Фармасьютикалз, Инк. 3-азабицикло[3.1.0]гексильные производные в качестве модуляторов метаботропных глутаматных рецепторов
AU2009319387B2 (en) 2008-11-28 2012-05-10 Addex Pharma S.A. Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
US8114894B2 (en) 2008-12-03 2012-02-14 Nanotherapeutics, Inc. Bicyclic compounds and methods of making and using same
RS53075B (en) 2009-05-12 2014-04-30 Janssen Pharmaceuticals Inc. 1,2,4-TRIAZOLO [4,3-A] PYRIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OR PREVENTION OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS
JP5707390B2 (ja) 2009-05-12 2015-04-30 ジャンセン ファーマシューティカルズ， インコーポレイテッド １，２，４−トリアゾロ［４，３−ａ］ピリジン誘導体およびｍＧｌｕＲ２受容体の正のアロステリック調節因子としてのその使用
MY153913A (en) 2009-05-12 2015-04-15 Janssen Pharmaceuticals Inc 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
BR112012002164B1 (pt) * 2009-07-30 2021-04-20 Merial, Inc compostos inseticidas de 4-amino-tieno[2,3-d]-pirimidina e métodos para seu uso
BR112012021453A2 (pt) 2010-02-26 2017-02-21 Boehringer Ingelheim Int tienopirimidina, sua composição farmacêutica e seu uso
UY33241A (es) 2010-02-26 2011-09-30 Boehringer Ingelheim Int ?Tienopirimidinas que contienen heterocicloalquilo para composiciones farmacéuticas?.
JP5575274B2 (ja) 2010-02-26 2014-08-20 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 医薬組成物のためのｍｎｋｌ／ｍｎｋ２阻害活性を有する４−［シクロアルキルオキシ（ヘテロ）アリールアミノ］チエノ「２，３−ｄ］ピリミジン
TW201219401A (en) 2010-09-14 2012-05-16 Lexicon Pharmaceuticals Inc Bicyclic inhibitors of Notum Pectinacetylesterase and methods of their use
EP2661435B1 (fr) 2010-11-08 2015-08-19 Janssen Pharmaceuticals, Inc. Dérivés 1,2,4-triazolo[4,3-a]pyridine et leur utilisation en tant que modulateurs allostériques positifs des récepteurs mglur2
EP2649069B1 (fr) 2010-11-08 2015-08-26 Janssen Pharmaceuticals, Inc. Dérivés de 1,2,4-triazolo[4,3-a]pyridine et leur utilisation en tant que modulateurs allostériques positifs des récepteurs mglur2
EP2643320B1 (fr) 2010-11-08 2015-03-04 Janssen Pharmaceuticals, Inc. Dérivés de la 1,2,4-triazolo [4,3-a] pyridine et leur utilisation en tant que modulateurs allostériques positifs des récepteurs mglur2
AR090037A1 (es) 2011-11-15 2014-10-15 Xention Ltd Derivados de tieno y/o furo-pirimidinas y piridinas inhibidores de los canales de potasio
CN104902751A (zh) * 2012-11-09 2015-09-09 住友化学株式会社 促进植物生长的方法
JO3368B1 (ar) 2013-06-04 2019-03-13 Janssen Pharmaceutica Nv مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
FR3015483B1 (fr) * 2013-12-23 2016-01-01 Servier Lab Nouveaux derives de thienopyrimidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
DK3431106T3 (da) 2014-01-21 2021-03-15 Janssen Pharmaceutica Nv Kombinationer omfattende positive allosteriske modulatorer eller orthosteriske agonister af metabotrop glutamaterg subtype 2-receptor og anvendelse af disse
ES2860298T3 (es) 2014-01-21 2021-10-04 Janssen Pharmaceutica Nv Combinaciones que comprenden moduladores alostéricos positivos del receptor glutamatérgico metabotrópico de subtipo 2 y su uso
RU2746282C1 (ru) * 2020-07-30 2021-04-12 Федеральное государственное бюджетное образовательное учреждение высшего образования "Кубанский государственный университет" (ФГБОУ ВО "КубГУ") Способ повышения урожайности озимой пшеницы

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1570494A (en) * 1975-11-28 1980-07-02 Ici Ltd Thienopyrimidine derivatives and their use as pesticides
ZA782648B (en) * 1977-05-23 1979-06-27 Ici Australia Ltd The prevention,control or eradication of infestations of ixodid ticks

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110177795A (zh) * 2016-12-26 2019-08-27 韩美药品株式会社 制备噻吩并嘧啶化合物的新方法和中间体

Also Published As

Publication number Publication date
EP0447891A1 (fr) 1991-09-25
EP0447891B1 (fr) 1994-04-27
CA2038521A1 (fr) 1991-09-20
ES2052296T3 (es) 1994-07-01
DE59101477D1 (de) 1994-06-01
DE4008726A1 (de) 1991-09-26
JPH04217685A (ja) 1992-08-07

Similar Documents

Publication Publication Date Title
DK0447891T3 (da) Thieno(2,3-d)pyrimidinderivater
EP0407342A3 (en) Pyrimidine derivatives
HU9300964D0 (en) Nucleoside derivatives
FI944305A (fi) Pyrido(2,3-d)pyrimidiinijohdannaiset fosfodiesteraasi-inhibiittoreina
OA09677A (en) Nucleoside derivatives
FI930429A (fi) Nya 1,4-dihyropyridinderivat
LV11176A (lv) Uracila atvasinajumi
DE69110093T2 (de) Pyrimidinderivate.
NO912804D0 (no) Purinderivater.
DK232387D0 (da) Diastereoisomere tetrahydropyrido (2,3-d) pyrimi- din derivativer
NO895217L (no) Substituerte pyrido(2,3-d)pyrimidiner.
DE3769721D1 (de) 4(3h)-oxo-5,6,7,8-tetrahydropyrido(2,3-d)pyrimidinderivate.
FI912963A0 (fi) Hjaernverksamheten oekande pyrimidinylderivat.
DE69004844T2 (de) Pyrimidin-Derivate.
EP0457505A3 (en) Pyrimidine derivatives
DE69132738T2 (de) Antivirale tetrahydroimidazo[1,4]benzodiazepin-2-(thio)one
DE3276808D1 (de) Pyrido (2,3-d) pyrimidines
DK0417840T3 (da) Antivirale tetrahydroimidazo(1,4)benzodiazepiner
GB8902688D0 (en) Pyrimidine derivatives
KR930700523A (ko) 뉴클레오티드 유도체
IE901141L (en) Pyrimidine derivatives
IE901756L (en) Pyrimidine derivatives
NO912552D0 (no) Fremgangsmaate for fremstilling av pyrimidinnukleosider.
HU9204124D0 (en) 1,2,3,3a,8,8a-hexahydro-1,3a,8-trimethyl-pyrrholo/2,3-b/-indole-tetrahydro-isoquinoline-urea derivatives
IT8921215A0 (it) Pirido(2,3 d)pirimidine sostituite.