DE69518323D1 - Oxaborole und deren salze, und deren verwendung als biozide - Google Patents
Oxaborole und deren salze, und deren verwendung als biozideInfo
- Publication number
- DE69518323D1 DE69518323D1 DE69518323T DE69518323T DE69518323D1 DE 69518323 D1 DE69518323 D1 DE 69518323D1 DE 69518323 T DE69518323 T DE 69518323T DE 69518323 T DE69518323 T DE 69518323T DE 69518323 D1 DE69518323 D1 DE 69518323D1
- Authority
- DE
- Germany
- Prior art keywords
- pct
- oxaborole
- biocides
- salts
- date dec
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 239000003139 biocide Substances 0.000 title 1
- OHENQANLQNOMAO-UHFFFAOYSA-N oxaborole Chemical compound O1B=CC=C1 OHENQANLQNOMAO-UHFFFAOYSA-N 0.000 title 1
- 230000000813 microbial effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
- C08K5/00—Use of organic ingredients
- C08K5/0008—Organic ingredients according to more than one of the "one dot" groups of C08K5/01 - C08K5/59
- C08K5/0058—Biocides
-
- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09D—COATING COMPOSITIONS, e.g. PAINTS, VARNISHES OR LACQUERS; FILLING PASTES; CHEMICAL PAINT OR INK REMOVERS; INKS; CORRECTING FLUIDS; WOODSTAINS; PASTES OR SOLIDS FOR COLOURING OR PRINTING; USE OF MATERIALS THEREFOR
- C09D5/00—Coating compositions, e.g. paints, varnishes or lacquers, characterised by their physical nature or the effects produced; Filling pastes
- C09D5/14—Paints containing biocides, e.g. fungicides, insecticides or pesticides
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- Polymers & Plastics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Biodiversity & Conservation Biology (AREA)
- Materials Engineering (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Micro-Organisms Or Cultivation Processes Thereof (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB9411587A GB9411587D0 (en) | 1994-06-09 | 1994-06-09 | Compound, composition and use |
PCT/GB1995/001206 WO1995033754A1 (en) | 1994-06-09 | 1995-05-26 | Oxaboroles and salts thereof, and their use as biocides |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69518323D1 true DE69518323D1 (de) | 2000-09-14 |
DE69518323T2 DE69518323T2 (de) | 2001-02-01 |
Family
ID=10756481
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69518323T Expired - Fee Related DE69518323T2 (de) | 1994-06-09 | 1995-05-26 | Oxaborole und deren salze, und deren verwendung als biozide |
Country Status (14)
Country | Link |
---|---|
US (1) | US5880188A (de) |
EP (1) | EP0765331B1 (de) |
JP (1) | JPH10500983A (de) |
KR (1) | KR970703349A (de) |
CN (1) | CN1068005C (de) |
AT (1) | ATE195316T1 (de) |
AU (1) | AU681291B2 (de) |
BR (1) | BR9507966A (de) |
CA (1) | CA2190155A1 (de) |
DE (1) | DE69518323T2 (de) |
GB (1) | GB9411587D0 (de) |
NO (1) | NO965235L (de) |
TW (1) | TW368397B (de) |
WO (1) | WO1995033754A1 (de) |
Families Citing this family (62)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1009415A4 (de) * | 1997-06-13 | 2000-10-25 | Univ Northwestern | g(B)-LAKTAMASE HEMMER UND VERWENDUNGEN DAVON |
US6184363B1 (en) | 1997-06-13 | 2001-02-06 | Northwestern University | Inhibitors of β-lactamases and uses therefor |
BRPI0411582A (pt) * | 2003-06-16 | 2006-08-08 | Anacor Pharmaceuticals Inc | substáncias terapêuticas contendo boro hidroliticamente resistentes e método de uso |
KR20050047699A (ko) * | 2003-11-18 | 2005-05-23 | 주식회사 엘지생명과학 | 살균성 수성 액상수화제 |
US7767657B2 (en) | 2005-02-16 | 2010-08-03 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
CA2597982C (en) * | 2005-02-16 | 2014-07-08 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
MX335993B (es) * | 2005-12-30 | 2016-01-07 | Anacor Pharmaceuticals Inc | Moleculas pequeñas que contienen boro. |
SI2719388T1 (sl) * | 2006-02-16 | 2019-06-28 | Anacor Pharmaceuticals, Inc. | Majhne molekule, polnjene z borom, kot učinkovine proti vnetjem |
US20070197388A1 (en) * | 2006-02-22 | 2007-08-23 | Buckman Laboratories International, Inc. | Haloperoxidase treatment to control algae |
RU2486914C2 (ru) * | 2006-03-16 | 2013-07-10 | Молеак Пте Лтд | Комбинированная терапия для лечения пациентов с неврологическими нарушениями и церебральным инфарктом |
US8106031B2 (en) * | 2006-05-02 | 2012-01-31 | Anacor Pharmaceuticals, Inc. | Hydrolytically-resistant boron-containing therapeutics and methods of use |
EP1900378A1 (de) * | 2006-08-31 | 2008-03-19 | Novartis AG | Pharmazeutische Zusammensetzungen zur Behandlung von Pilzinfektionen |
JO3396B1 (ar) * | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
JP5504454B2 (ja) * | 2007-12-06 | 2014-05-28 | 国立大学法人京都大学 | 新規なホウ素化合物、それらの製造方法およびそれらを用いた機能性電子素子 |
JP5745279B2 (ja) * | 2008-01-09 | 2015-07-08 | アナコール ファーマシューティカルズ,インコーポレイテッド | 抗炎症剤としてのホウ素含有小分子 |
MX2010009765A (es) | 2008-03-06 | 2013-07-12 | Anacor Pharmaceuticals Inc | Moleculas pequeñas que contienen boro como agentes anti-inflamatorios. |
EP2285384A4 (de) * | 2008-05-12 | 2012-04-25 | Anacor Pharmaceuticals Inc | Borhaltige kleine moleküle |
EP2348863A4 (de) * | 2008-09-04 | 2012-03-07 | Anacor Pharmaceuticals Inc | Borhaltige kleine moleküle |
WO2010028005A1 (en) | 2008-09-04 | 2010-03-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
EP2343279B1 (de) | 2008-10-15 | 2018-02-28 | Kissei Pharmaceutical Co., Ltd. | Ringkondensiertes derivat und medizinische anwendung davon |
US9493489B2 (en) * | 2008-10-15 | 2016-11-15 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as anti-protozoal agents |
EP2378886A4 (de) * | 2008-12-17 | 2012-08-29 | Anacor Pharmaceuticals Inc | (s)-3-aminomethyl-7-(3-hydroxypropoxy)-3h-benzo[c][1,2]oxaborol-1-ol-polymorphe |
BR112012001987A2 (pt) * | 2009-07-28 | 2015-09-01 | Anacor Pharmaceuticals Inc | Composto, combinação, formulação farmacêutica, uso de um composto, uma combinação ou um sal farmaceuticamente aceitável dos mesmos, e, métodos para tratar uma infecção bacteriana, para matar ou inibir o crescimento de uma bactéria, e para inibir uma beta-lactamase. |
AP4039A (en) | 2009-08-14 | 2017-02-28 | Daitao Chen | Boron-containing small molecules as antiprotozoal agents |
WO2011022337A1 (en) * | 2009-08-19 | 2011-02-24 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
WO2011049971A1 (en) | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
US20110212918A1 (en) * | 2009-11-11 | 2011-09-01 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
WO2011094450A1 (en) | 2010-01-27 | 2011-08-04 | Anacor Pharmaceuticals, Inc | Boron-containing small molecules |
AP2012006482A0 (en) | 2010-03-19 | 2012-10-31 | Anacor Pharmacueticals Inc | Boron-containing small molecules as anti-protozoalagent |
JP5952280B2 (ja) | 2010-09-07 | 2016-07-13 | アナコール ファーマシューティカルズ,インコーポレーテッド | 細菌感染治療用のベンゾオキサボロール誘導体 |
UY34367A (es) * | 2011-10-07 | 2014-08-29 | Syngenta Participations Ag | ?método para proteger material de propagación vegetal o plantas útiles?. |
WO2013057740A2 (en) | 2011-10-07 | 2013-04-25 | Syngenta Participations Ag | Method for protecting useful plants or plant propagation material |
US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
CN107646865B (zh) * | 2013-01-30 | 2020-07-03 | 美国陶氏益农公司 | 苯硼酸半酯作为挥发性抗微生物剂在肉类、植物或植物部分上的用途 |
US20220125049A1 (en) * | 2013-01-30 | 2022-04-28 | Agrofresh Inc. | Method and system for centralized management, monitoring, and controlled delivery of biological compounds to fruit storage rooms |
US9585396B2 (en) | 2013-01-30 | 2017-03-07 | Agrofresh Inc. | Volatile applications against pathogens |
US8669207B1 (en) | 2013-01-30 | 2014-03-11 | Dow Agrosciences, Llc. | Compounds and compositions |
WO2014147009A1 (en) * | 2013-03-18 | 2014-09-25 | Syngenta Participations Ag | Novel microbiocides |
WO2014173880A1 (en) | 2013-04-22 | 2014-10-30 | Syngenta Participations Ag | Novel microbiocides |
AU2014202928B1 (en) * | 2013-06-05 | 2014-09-11 | Agrofresh Inc. | Compounds and compositions |
US20170000132A1 (en) * | 2013-12-23 | 2017-01-05 | Syngenta Participations Ag | Benzoxaborole fungicides |
EP3086645A1 (de) * | 2013-12-23 | 2016-11-02 | Syngenta Participations AG | Benzoxaborolfungizide |
MA41495A (fr) * | 2015-02-12 | 2017-12-19 | Anacor Pharmaceuticals Inc | Composés benzoxaborole et leurs utilisations |
US9730454B2 (en) * | 2015-02-12 | 2017-08-15 | Agrofresh Inc. | Fungicidal compounds and compositions |
US9737075B2 (en) | 2015-04-09 | 2017-08-22 | The Penn State Research Foundation | Synergistic benzoxaborole-containing anti-fungicidal composition |
WO2017024022A1 (en) * | 2015-08-06 | 2017-02-09 | The Penn State Research Foundation | Benzoxaborole-containing coating resistant to cellulose-supportable fungus |
WO2017031041A1 (en) * | 2015-08-17 | 2017-02-23 | Channel Therapeutics, Inc. | Functionalized aminobenzoboroxoles |
CN113321672A (zh) * | 2016-03-02 | 2021-08-31 | 比尔及梅琳达盖茨基金会 | 含硼小分子 |
TW201733442A (zh) | 2016-03-07 | 2017-10-01 | 農業保鮮股份有限公司 | 殺有害生物劑之汽化給予 |
TW201735792A (zh) | 2016-03-07 | 2017-10-16 | 農業保鮮股份有限公司 | 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法 |
US11447506B2 (en) | 2016-05-09 | 2022-09-20 | Anacor Pharmaceuticals, Inc. | Crystal forms of crisaborole in free form and preparation method and use thereof |
EP3455227A1 (de) | 2016-05-12 | 2019-03-20 | Anacor Pharmaceuticals, Inc | Oxaborolester und verwendungen davon |
EP3704100B1 (de) | 2017-11-02 | 2023-08-30 | Halcyon Labs Private Limited | Neues verfahren zur herstellung von tavaborol und dessen zwischenprodukte |
US11834466B2 (en) | 2017-11-30 | 2023-12-05 | 5Metis, Inc. | Benzoxaborole compounds and formulations thereof |
WO2019173814A1 (en) | 2018-03-09 | 2019-09-12 | University Of The Sciences | Protective groups and methods for protecting benzoxaboroles or oxaboroles |
AU2019325436B2 (en) * | 2018-08-18 | 2023-10-26 | 5Metis, Inc. | Solid forms of substituted benzoxaborole and compositions thereof |
CU20210023A7 (es) | 2018-10-05 | 2021-10-12 | Pfizer | Inhibidores fenil sustituidos de la piridinil 1,2-oxaborolan-2-ol fosfodiesterasa 4 |
US20210024548A1 (en) * | 2019-07-25 | 2021-01-28 | Massachusetts Institute Of Technology | Boron-containing pharmacophore |
AR120504A1 (es) | 2019-11-22 | 2022-02-16 | Agrofresh Inc | Composición y método para tratar a plantas y partes de plantas con activos volátiles para el control de organismos de descomposición |
CR20220369A (es) | 2020-02-05 | 2022-10-27 | Agrofresh Inc | Compuestos y composiciones antimicrobianos |
CN114644645B (zh) * | 2022-03-08 | 2023-05-26 | 南京农业大学 | 3-吲哚取代苯硼唑类化合物及其制备方法和应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3104255A (en) * | 1960-06-16 | 1963-09-17 | Standard Oil Co | Telomerization of unsaturated hydrocarbons with alkylene glycol borates and telomeric products obtained thereby |
US3361672A (en) * | 1965-10-23 | 1968-01-02 | Mobil Oil Corp | Stabilized organic compositions |
GB1140399A (en) * | 1966-09-16 | 1969-01-15 | Koninklijke Pharma Fab Nv | New diphenylmethoxy derivatives |
US3686398A (en) * | 1970-07-20 | 1972-08-22 | Chevron Res | 10,9-boroxarophenanthrene as fungicides |
GB1396904A (en) * | 1972-08-11 | 1975-06-11 | Ici Ltd | Method for the control of micro-organisms |
-
1994
- 1994-06-09 GB GB9411587A patent/GB9411587D0/en active Pending
-
1995
- 1995-05-26 AU AU25348/95A patent/AU681291B2/en not_active Ceased
- 1995-05-26 DE DE69518323T patent/DE69518323T2/de not_active Expired - Fee Related
- 1995-05-26 US US08/750,081 patent/US5880188A/en not_active Expired - Fee Related
- 1995-05-26 EP EP95919572A patent/EP0765331B1/de not_active Expired - Lifetime
- 1995-05-26 WO PCT/GB1995/001206 patent/WO1995033754A1/en active IP Right Grant
- 1995-05-26 BR BR9507966A patent/BR9507966A/pt not_active Application Discontinuation
- 1995-05-26 CN CN95194519A patent/CN1068005C/zh not_active Expired - Fee Related
- 1995-05-26 CA CA002190155A patent/CA2190155A1/en not_active Abandoned
- 1995-05-26 JP JP8500489A patent/JPH10500983A/ja not_active Withdrawn
- 1995-05-26 AT AT95919572T patent/ATE195316T1/de not_active IP Right Cessation
- 1995-05-30 TW TW084105427A patent/TW368397B/zh active
-
1996
- 1996-12-06 NO NO965235A patent/NO965235L/no unknown
- 1996-12-07 KR KR1019960706993A patent/KR970703349A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
GB9411587D0 (en) | 1994-08-03 |
BR9507966A (pt) | 1997-09-02 |
DE69518323T2 (de) | 2001-02-01 |
TW368397B (en) | 1999-09-01 |
NO965235D0 (no) | 1996-12-06 |
KR970703349A (ko) | 1997-07-03 |
ATE195316T1 (de) | 2000-08-15 |
AU2534895A (en) | 1996-01-04 |
JPH10500983A (ja) | 1998-01-27 |
NO965235L (no) | 1997-01-21 |
CN1068005C (zh) | 2001-07-04 |
CA2190155A1 (en) | 1995-12-14 |
EP0765331A1 (de) | 1997-04-02 |
WO1995033754A1 (en) | 1995-12-14 |
US5880188A (en) | 1999-03-09 |
EP0765331B1 (de) | 2000-08-09 |
AU681291B2 (en) | 1997-08-21 |
CN1155286A (zh) | 1997-07-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8339 | Ceased/non-payment of the annual fee |