AU2003262262A1 - Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereof - Google Patents
Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereofInfo
- Publication number
- AU2003262262A1 AU2003262262A1 AU2003262262A AU2003262262A AU2003262262A1 AU 2003262262 A1 AU2003262262 A1 AU 2003262262A1 AU 2003262262 A AU2003262262 A AU 2003262262A AU 2003262262 A AU2003262262 A AU 2003262262A AU 2003262262 A1 AU2003262262 A1 AU 2003262262A1
- Authority
- AU
- Australia
- Prior art keywords
- medicinal
- same
- composition containing
- pyrazole derivatives
- medicinal composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/7056—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing five-membered rings with nitrogen as a ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/095—Sulfur, selenium, or tellurium compounds, e.g. thiols
- A61K31/10—Sulfides; Sulfoxides; Sulfones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/205—Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A61K31/366—Lactones having six-membered rings, e.g. delta-lactones
- A61K31/37—Coumarins, e.g. psoralen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
- A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
- A61K31/737—Sulfated polysaccharides, e.g. chondroitin sulfate, dermatan sulfate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2002-247864 | 2002-08-27 | ||
JP2002247864 | 2002-08-27 | ||
PCT/JP2003/010550 WO2004019958A1 (en) | 2002-08-27 | 2003-08-21 | Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2003262262A1 true AU2003262262A1 (en) | 2004-03-19 |
Family
ID=31972489
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2003262262A Abandoned AU2003262262A1 (en) | 2002-08-27 | 2003-08-21 | Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereof |
Country Status (3)
Country | Link |
---|---|
JP (1) | JP4606876B2 (en) |
AU (1) | AU2003262262A1 (en) |
WO (1) | WO2004019958A1 (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7524822B2 (en) | 2006-01-11 | 2009-04-28 | Boehringer Ingelheim International Gmbh | Crystalline form of 1′-(1-methylethyl)-4′-[(2-fluoro-4-methoxyphenyl)methyl]-5′-methyl-1H-pyrazol-3′-O-β-D-glucopyranoside, a method for its preparation and the use thereof for preparing medicaments |
Families Citing this family (45)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20050089156A (en) * | 2002-12-04 | 2005-09-07 | 깃세이 야쿠힌 고교 가부시키가이샤 | Preventive or remedy for diseases caused by hyperglycemia |
JP4679155B2 (en) * | 2002-12-25 | 2011-04-27 | キッセイ薬品工業株式会社 | Nitrogen-containing heterocyclic derivative, pharmaceutical composition containing the same, and pharmaceutical use thereof |
EP2397462A3 (en) | 2003-01-14 | 2012-04-04 | Cytokinetics, Inc. | Compounds, compositions and methods of treatment for heart failure |
US8785403B2 (en) | 2003-08-01 | 2014-07-22 | Mitsubishi Tanabe Pharma Corporation | Glucopyranoside compound |
ES2844401T3 (en) | 2003-08-01 | 2021-07-22 | Mitsubishi Tanabe Pharma Corp | Novel compounds that have inhibitory activity against the sodium-dependent glucose transporter |
US7375090B2 (en) | 2003-08-26 | 2008-05-20 | Boehringer Ingelheim International Gmbh | Glucopyranosyloxy-pyrazoles, pharmaceutical compositions containing these compounds, the use thereof and processed for the preparation thereof |
DE102004028241B4 (en) * | 2004-06-11 | 2007-09-13 | Sanofi-Aventis Deutschland Gmbh | New fluoroglycoside derivatives of pyrazoles, medicines containing these compounds and manufacture of these medicines |
KR101276136B1 (en) | 2004-06-17 | 2013-06-18 | 싸이토키네틱스, 인코포레이티드 | Compounds, compositions and methods |
US7176222B2 (en) | 2004-07-27 | 2007-02-13 | Cytokinetics, Inc. | Syntheses of ureas |
MY147375A (en) | 2005-01-31 | 2012-11-30 | Mitsubishi Tanabe Pharma Corp | Indole derivatives |
JP4888840B2 (en) * | 2005-07-22 | 2012-02-29 | 味の素株式会社 | Process for the preparation of pyrazole-O-glycoside derivatives and novel intermediates of said process |
US7538223B2 (en) | 2005-08-04 | 2009-05-26 | Cytokinetics, Inc. | Compounds, compositions and methods |
US7825120B2 (en) | 2005-12-15 | 2010-11-02 | Cytokinetics, Inc. | Certain substituted ((piperazin-1-ylmethyl)benzyl)ureas |
US20070161617A1 (en) | 2005-12-15 | 2007-07-12 | Morgan Bradley P | Certain chemical entities, compositions and methods |
WO2007078815A2 (en) | 2005-12-16 | 2007-07-12 | Cytokinetics, Inc. | Certain chemical entities, compositions, and methods |
JP5178526B2 (en) | 2005-12-19 | 2013-04-10 | サイトキネティクス・インコーポレーテッド | Compounds, compositions and methods |
JP2009167103A (en) * | 2006-05-02 | 2009-07-30 | Taisho Pharmaceutical Co Ltd | Pyrazolyl 5-thioglycoside compound |
PE20110235A1 (en) | 2006-05-04 | 2011-04-14 | Boehringer Ingelheim Int | PHARMACEUTICAL COMBINATIONS INCLUDING LINAGLIPTIN AND METMORPHINE |
US7973012B2 (en) | 2006-05-19 | 2011-07-05 | Taisho Pharmaceutical Co., Ltd | C-phenyl glycitol compound |
BRPI0713058A2 (en) | 2006-06-29 | 2012-04-10 | Taisho Pharmaceutical Co., Ltd. | c-phenyl 1-thioglycitol compound |
TWI418556B (en) | 2006-07-27 | 2013-12-11 | Mitsubishi Tanabe Pharma Corp | Indole derivatives |
ES2397664T3 (en) | 2006-12-04 | 2013-03-08 | Janssen Pharmaceutica, N.V. | Glucopyranosyl derivatives containing thienyl as antidiabetics |
UY30730A1 (en) | 2006-12-04 | 2008-07-03 | Mitsubishi Tanabe Pharma Corp | CRYSTAL FORM OF HEMIHYDRATE 1- (B (BETA) -D-GLUCOPYRANOSIL) -4-METHYL-3- [5- (4-FLUOROPHENYL) -2-TIENYLMETHYL] BENZENE |
CA2672176A1 (en) | 2006-12-14 | 2008-06-19 | Taisho Pharmaceutical Co., Ltd. | 1-phenyl 1-thio-d-glucitol derivative |
CA2699285C (en) | 2007-09-10 | 2016-12-13 | Ahmed F. Abdel-Magid | Process for the preparation of compounds useful as inhibitors of sodium-dependent glucose transporter (sglt) |
NZ586336A (en) * | 2007-12-27 | 2011-06-30 | Kissei Pharmaceutical | Monosebacate of pyrazole derivative |
CL2008003653A1 (en) | 2008-01-17 | 2010-03-05 | Mitsubishi Tanabe Pharma Corp | Use of a glucopyranosyl-derived sglt inhibitor and a selected dppiv inhibitor to treat diabetes; and pharmaceutical composition. |
US9056850B2 (en) | 2008-10-17 | 2015-06-16 | Janssen Pharmaceutica N.V. | Process for the preparation of compounds useful as inhibitors of SGLT |
PE20120648A1 (en) | 2009-02-23 | 2012-05-31 | Taisho Pharmaceutical Co Ltd | 4-ISOPROPYLPHENYLGLUCITOL COMPOUNDS AS SGLT1 INHIBITORS |
US20110009347A1 (en) | 2009-07-08 | 2011-01-13 | Yin Liang | Combination therapy for the treatment of diabetes |
AU2010270202B2 (en) | 2009-07-10 | 2014-04-24 | Janssen Pharmaceutica Nv | Crystallisation process for 1-(beta-D-glucopyranosyl)-4-methyl-3- [5-(4-fluorophenyl)-2-thienylmethyl] benzene |
CN102648196B (en) | 2009-10-14 | 2016-04-27 | 詹森药业有限公司 | Can be used as the preparation method of the compound of the inhibitor of SGLT2 |
CA2777857C (en) | 2009-11-02 | 2014-12-02 | Pfizer Inc. | Dioxa-bicyclo[3.2.1]octane-2,3,4-triol derivatives |
WO2011107494A1 (en) | 2010-03-03 | 2011-09-09 | Sanofi | Novel aromatic glycoside derivatives, medicaments containing said compounds, and the use thereof |
JP6227406B2 (en) | 2010-05-11 | 2017-11-08 | ヤンセン ファーマシューティカ エヌ.ベー. | Pharmaceutical formulations containing 1- (β-D-glucopyranosyl) -2-thienyl-methylbenzene derivatives as inhibitors of SGLT |
WO2012023600A1 (en) | 2010-08-20 | 2012-02-23 | 大正製薬株式会社 | 4-isopropyl-6-methoxyphenyl glucitol compound |
KR20130097711A (en) | 2010-08-20 | 2013-09-03 | 다이쇼 세이야꾸 가부시끼가이샤 | Crystal form of 4-isopropylphenyl glucitol compound and process for production thereof |
WO2012140120A1 (en) | 2011-04-13 | 2012-10-18 | Janssen Pharmaceutica Nv | Process for the preparation of compounds useful as inhibitors of sglt2 |
US9035044B2 (en) | 2011-05-09 | 2015-05-19 | Janssen Pharmaceutica Nv | L-proline and citric acid co-crystals of (2S, 3R, 4R, 5S,6R)-2-(3-((5-(4-fluorophenyl)thiopen-2-yl)methyl)4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol |
WO2012176804A1 (en) * | 2011-06-20 | 2012-12-27 | キッセイ薬品工業株式会社 | Glucopyranosyloxypyrazole derivative |
TW201425326A (en) | 2012-10-05 | 2014-07-01 | Lilly Co Eli | Novel urea compounds |
KR102078433B1 (en) | 2013-02-04 | 2020-02-17 | 다이쇼 세이야꾸 가부시끼가이샤 | Prophylactic or therapeutic drug for constipation |
EP2774619B1 (en) | 2013-03-04 | 2016-05-18 | BioActive Food GmbH | Composition for the treatment of hyperglycaemic diseases |
EP2944311A1 (en) | 2014-05-16 | 2015-11-18 | BioActive Food GmbH | Combination of biologically active substances for treating hyperglycemic diseases |
US20170071970A1 (en) | 2015-09-15 | 2017-03-16 | Janssen Pharmaceutica Nv | Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3989730B2 (en) * | 1999-08-31 | 2007-10-10 | キッセイ薬品工業株式会社 | Glucopyranosyloxypyrazole derivative, pharmaceutical composition containing the same, and production intermediate thereof |
WO2002036602A1 (en) * | 2000-11-02 | 2002-05-10 | Ajinomoto Co., Inc. | Novel pyrazole derivatives and diabetes remedies containing the same |
CN1238363C (en) * | 2000-12-28 | 2006-01-25 | 橘生药品工业株式会社 | Glucopyranosyloxypyrazole derivatives and use thereof in medicines |
TW593329B (en) * | 2001-02-26 | 2004-06-21 | Kissei Pharmaceutical | Glucopyranosyloxypyrazole derivatives and pharmaceutical uses thereof |
DE60237580D1 (en) * | 2001-02-27 | 2010-10-21 | Kissei Pharmaceutical | GLYCOPYRANOSYLOXYPYRAZOLE DERIVATIVES AND THEIR MEDICAL USE |
WO2002088157A1 (en) * | 2001-04-27 | 2002-11-07 | Ajinomoto Co., Inc. | N-substituted pyrazolyl-o-glycoside derivatives and remedial agent for diabetes containing the same |
CA2448741C (en) * | 2001-05-30 | 2010-06-22 | Kissei Pharmaceutical Co., Ltd. | Glucopyranosyloxypyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate therefor |
JP4115105B2 (en) * | 2001-07-02 | 2008-07-09 | 協和醗酵工業株式会社 | Pyrazole derivative |
CA2484306A1 (en) * | 2002-04-26 | 2003-11-06 | Katsumi Maezono | Prophylactic and therapeutic agent of diabetes mellitus |
CA2494179C (en) * | 2002-08-08 | 2012-04-24 | Kissei Pharmaceutical Co., Ltd. | Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof |
JP2004137245A (en) * | 2002-08-23 | 2004-05-13 | Kissei Pharmaceut Co Ltd | Pyrazole derivative, pharmaceutical composition containing the same, its pharmaceutical use and production intermediate |
-
2003
- 2003-08-21 WO PCT/JP2003/010550 patent/WO2004019958A1/en active Application Filing
- 2003-08-21 AU AU2003262262A patent/AU2003262262A1/en not_active Abandoned
- 2003-08-21 JP JP2004532694A patent/JP4606876B2/en not_active Expired - Fee Related
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7524822B2 (en) | 2006-01-11 | 2009-04-28 | Boehringer Ingelheim International Gmbh | Crystalline form of 1′-(1-methylethyl)-4′-[(2-fluoro-4-methoxyphenyl)methyl]-5′-methyl-1H-pyrazol-3′-O-β-D-glucopyranoside, a method for its preparation and the use thereof for preparing medicaments |
US7838500B2 (en) | 2006-01-11 | 2010-11-23 | Ajinomoto Co., Inc. | Crystalline form of 1′-(1-methylethyl)-4′-[(2-fluoro-4-methoxyphenyl)methyl]-5′-methyl-1H-pyrazol-3′-O-β-D-glucopyranoside, a method for its preparation and the use thereof for preparing medicaments |
Also Published As
Publication number | Publication date |
---|---|
JP4606876B2 (en) | 2011-01-05 |
WO2004019958A1 (en) | 2004-03-11 |
JPWO2004019958A1 (en) | 2005-12-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU2003262262A1 (en) | Pyrazole derivatives, medicinal composition containing the same, and medicinal use thereof | |
HK1082744A1 (en) | Pyrazole derivatives, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof | |
AU2003289440A1 (en) | Nitrogen-containing heterocycic derivatives, medicinal compositions containing the same and medicinal use thereof | |
IL164209A0 (en) | Pyrazole derivatives and pharmaceutical compositions containing the same | |
IL166620A0 (en) | Pyrazole derivatives and pharmaceutical compositions containing the same | |
AU2002306269A1 (en) | N-arylphenylacetamide derivatives and pharmaceutical composition containing the same | |
AU2003289641A1 (en) | The novel coumarin-amide derivatives and its preparation, said drug composition and its use | |
EP1405859A4 (en) | Nitrogenous heterocyclic derivative, medicinal composition containing the same, medicinal use thereof and intermediate therefor | |
IL176005A0 (en) | 2,6-bisheteroaryl-4-aminopyrimidine derivatives and pharmaceutical compositions containing the same | |
AU2001290257A2 (en) | Glucopyranosyloxybenzylbenzene derivatives and medicinal compositions containing the same | |
AU2001290257A1 (en) | Glucopyranosyloxybenzylbenzene derivatives and medicinal compositions containing the same | |
AU2003246810A1 (en) | Diphenylpyridine derivatives, the preparation thereof, and pharmaceutical compositions containing said derivatives | |
AU2001256184A1 (en) | 6-aminoalkyl-dihydropyrimidines and the use thereof as medicaments against viraldiseases | |
IL162548A0 (en) | 4-Oxoquinoline derivatives and pharmaceutical compositions containing the same | |
IL166482A0 (en) | Dihydropyrazolopyridine derivatives and pharmaceutical compositions containing the same | |
HUP0400467A3 (en) | 2-iminopyrrolidine derivatives, pharmaceutical compositions containing them and their use | |
IL163117A (en) | Indazole derivatives and pharmaceutical compositions containing the same | |
AU2003216934A1 (en) | Benzoxazinone derivatives, the preparation and use thereof as medicaments | |
HUP0500024A3 (en) | 6-aminomorphinane derivatives, their use and pharmaceutical compositions containing them | |
AU2003255645A1 (en) | Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof | |
AU2003269018A1 (en) | Acylaminothiazole derivatives, preparation and therapeutic use thereof | |
HUP0303155A3 (en) | 2-thio-substituted imidazole derivatives, the use thereof and pharmaceutical compositions containing them | |
AU2003272903A1 (en) | Pyrazole derivative, medicinal composition containing the same, medicinal use thereof and intermediate in producing the same | |
AU2003271734A1 (en) | 7h-dibenzo(b,g)(1,5)dioxocin-5-one derivatives and use thereof | |
AU4884701A (en) | Malonanilic acid derivatives, medicinal compositions containing the same and usethereof |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |