DE3686387D1 - Verfahren zur herstellung von 3-aminopyrrolidine. - Google Patents

Verfahren zur herstellung von 3-aminopyrrolidine.

Info

Publication number
DE3686387D1
DE3686387D1 DE8686113972T DE3686387T DE3686387D1 DE 3686387 D1 DE3686387 D1 DE 3686387D1 DE 8686113972 T DE8686113972 T DE 8686113972T DE 3686387 T DE3686387 T DE 3686387T DE 3686387 D1 DE3686387 D1 DE 3686387D1
Authority
DE
Germany
Prior art keywords
aminopyrrolidine
producing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE8686113972T
Other languages
English (en)
Other versions
DE3686387T2 (de
Inventor
Kou Hojo
Anji Sakamoto
Masumi Tsutsumi
Tamotsu Yamada
Kazuhiko Nakazono
Kazuya Ishimori
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Tokyo Chemical Industries Co Ltd
Original Assignee
Tokyo Kasei Kogyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP22604185A external-priority patent/JPS62201864A/ja
Priority claimed from JP22604285A external-priority patent/JPS6287565A/ja
Priority claimed from JP18660786A external-priority patent/JPS6341452A/ja
Application filed by Tokyo Kasei Kogyo Co Ltd filed Critical Tokyo Kasei Kogyo Co Ltd
Application granted granted Critical
Publication of DE3686387D1 publication Critical patent/DE3686387D1/de
Publication of DE3686387T2 publication Critical patent/DE3686387T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/14—Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE8686113972T 1985-10-11 1986-10-08 Verfahren zur herstellung von 3-aminopyrrolidine. Expired - Lifetime DE3686387T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP22604185A JPS62201864A (ja) 1985-10-11 1985-10-11 ３―アミノピロリジンの製造法
JP22604285A JPS6287565A (ja) 1985-10-11 1985-10-11 ３−アミノピロリジンおよびその塩の製造法
JP18660786A JPS6341452A (ja) 1986-08-08 1986-08-08 Ｎ，ｎ’，ｎ’−置換−３−アミノピロリジンの製造法

Publications (2)

Publication Number Publication Date
DE3686387D1 true DE3686387D1 (de) 1992-09-17
DE3686387T2 DE3686387T2 (de) 1993-01-14

Family

ID=27325774

Family Applications (1)

Application Number Title Priority Date Filing Date
DE8686113972T Expired - Lifetime DE3686387T2 (de) 1985-10-11 1986-10-08 Verfahren zur herstellung von 3-aminopyrrolidine.

Country Status (3)

Country Link
US (1) US4785119A (de)
EP (1) EP0218249B1 (de)
DE (1) DE3686387T2 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63295553A (ja) * 1987-05-01 1988-12-01 Fujisawa Pharmaceut Co Ltd ピロリジン誘導体
US4859776A (en) * 1988-03-11 1989-08-22 Abbott Laboratories (S)-7-(3-aminopyrrolidin-1-yl)-1-(ortho, para-difluorophenyl)-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acid and method for its preparation
US5099032A (en) * 1988-03-11 1992-03-24 Abbott Laboratories Process for the preparation of enantiomerically homogeneous aminopyrrolidinyl naphthyridine and quinolone carboxylic acids.
US4956475A (en) * 1988-03-11 1990-09-11 Abbott Laboratories Preparationof enantiomerically pure 3-protected amino-pyrrolidines
US5264453A (en) * 1988-10-31 1993-11-23 Fujisawa Pharmaceutical Co., Ltd. Pyrrolidine derivatives
US5130323A (en) * 1988-10-31 1992-07-14 Fujisawa Pharmaceutical Co., Ltd. Pyrrolidine derivatives
US5332817A (en) * 1990-01-04 1994-07-26 Pfizer Inc. 3-aminopiperidine derivatives and related nitrogen containing heterocycles
US5232929A (en) * 1990-11-28 1993-08-03 Pfizer Inc. 3-aminopiperidine derivatives and related nitrogen containing heterocycles and pharmaceutical compositions and use
CN1054980A (zh) * 1990-02-19 1991-10-02 杏林制药株式会社 具有旋光活性的8-甲氧基喹诺酮羧酸衍生物，它们的制备方法以及它们的中间体
GB9113031D0 (en) * 1991-06-17 1991-08-07 Smithkline Beecham Plc Compounds
US5177217A (en) * 1992-04-27 1993-01-05 Warner-Lambert Company Process for the manufacture of (S)-3-amino-1-substituted-pyrrolidines
EP1138672A1 (de) * 1998-01-12 2001-10-04 Basilea Pharmaceutica AG Verfahren zur Herstellung von 3-Aminopyrrolidinderivaten
US5977381A (en) * 1998-01-12 1999-11-02 Hoffmann-La Roche Inc. Process for making 3-amino-pyrolidine derivatives
US6531594B2 (en) 2000-08-24 2003-03-11 Mitsubishi Chemical Corporation Process for producing 1H-3-aminopyrrolidine and derivatives thereof
RU2355679C2 (ru) * 2002-11-27 2009-05-20 Инсайт Корпорейшн Производные 3-аминопирролидина в качестве модуляторов рецепторов хемокинов
US7507760B2 (en) * 2004-01-22 2009-03-24 Neuromed Pharmaceuticals Ltd. N-type calcium channel blockers
EP1757582B1 (de) 2004-05-28 2015-12-30 Mitsubishi Tanabe Pharma Corporation Arylalkylamine und verfahren zu deren herstellung
BRPI0516602A (pt) * 2004-10-18 2008-09-16 Lilly Co Eli composto, e, composição farmacêutica
CN1331852C (zh) * 2005-08-25 2007-08-15 浙江大学 N－取代基－3－氨基吡咯烷及其二盐酸盐的合成方法
WO2007143600A2 (en) * 2006-06-05 2007-12-13 Incyte Corporation Sheddase inhibitors combined with cd30-binding immunotherapeutics for the treatment of cd30 positive diseases
EP2050735A4 (de) * 2006-07-28 2011-12-21 Kaneka Corp Verfahren zur herstellung einer optisch aktiven 3-amino-nitrogenierte verbindung

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3424762A (en) * 1966-03-07 1969-01-28 Robins Co Inc A H Certain 3-ureidopyrrolidines
US3424761A (en) * 1966-03-07 1969-01-28 Robins Co Inc A H 3-ureidopyrrolidines
US3424760A (en) * 1966-03-07 1969-01-28 Robins Co Inc A H 3-ureidopyrrolidines
US3433801A (en) * 1966-03-22 1969-03-18 Robins Co Inc A H 1-aryl-3-(n-lower alkyl amino) pyrrolidines
AU417810B2 (en) * 1967-03-20 1971-10-12 1-aryl-3-lower alkylamino-pyrrolidine compound and production thereof
US3509171A (en) * 1967-09-14 1970-04-28 Robins Co Inc A H 3-amino-1-carbamyl and thiocarbamyl pyrrolidines
US3433802A (en) * 1968-06-25 1969-03-18 Robins Co Inc A H 3-(n-lower-alkylanilino)pyrrolidines
US3549658A (en) * 1968-08-12 1970-12-22 Robins Co Inc A H 1-(1-substituted-3-pyrrolidinyl)-3-arylsulfonylureas
US3577440A (en) * 1968-12-23 1971-05-04 Robins Co Inc A H 1-substituted-3-amido-pyrrolidines
US4056535A (en) * 1975-07-09 1977-11-01 Stanford Research Institute N-substituted 3-aminopyrrolidines
US4382937A (en) * 1981-02-27 1983-05-10 Dainippon Pharmaceutical Co., Ltd. Naphthyridine derivatives and their use as anti-bacterials

Also Published As

Publication number Publication date
DE3686387T2 (de) 1993-01-14
EP0218249B1 (de) 1992-08-12
EP0218249A2 (de) 1987-04-15
EP0218249A3 (en) 1989-03-15
US4785119A (en) 1988-11-15

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition