DE3362396D1 - Derivatives of ampicillin and amoxicillin with beta-lactamase inhibitors - Google Patents
Derivatives of ampicillin and amoxicillin with beta-lactamase inhibitorsInfo
- Publication number
- DE3362396D1 DE3362396D1 DE8383302585T DE3362396T DE3362396D1 DE 3362396 D1 DE3362396 D1 DE 3362396D1 DE 8383302585 T DE8383302585 T DE 8383302585T DE 3362396 T DE3362396 T DE 3362396T DE 3362396 D1 DE3362396 D1 DE 3362396D1
- Authority
- DE
- Germany
- Prior art keywords
- amoxicillin
- ampicillin
- beta
- derivatives
- lactamase inhibitors
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/376,487 US4377590A (en) | 1982-05-10 | 1982-05-10 | Derivatives of ampicillin and amoxicillin with beta-lactamase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
DE3362396D1 true DE3362396D1 (en) | 1986-04-10 |
Family
ID=23485209
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE8383302585T Expired DE3362396D1 (en) | 1982-05-10 | 1983-05-09 | Derivatives of ampicillin and amoxicillin with beta-lactamase inhibitors |
Country Status (7)
Country | Link |
---|---|
US (1) | US4377590A (de) |
EP (1) | EP0094227B1 (de) |
JP (1) | JPS58213788A (de) |
DE (1) | DE3362396D1 (de) |
DK (1) | DK206183A (de) |
GR (1) | GR78248B (de) |
IE (1) | IE54771B1 (de) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4462934A (en) | 1983-03-31 | 1984-07-31 | Pfizer Inc. | Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides |
US4916230A (en) * | 1984-07-02 | 1990-04-10 | Merck & Co., Inc. | Process for preparing novel N-(acyloxy-alkoxy)carbonyl derivatives useful as bioreversible prodrug moieties for primary and secondary amine functions in drugs |
KR910009271B1 (ko) * | 1989-06-20 | 1991-11-08 | 김영설 | 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염 |
GB8928373D0 (en) * | 1989-12-15 | 1990-02-21 | Erba Carlo Spa | Beta-lactam derivatives |
US6818787B2 (en) * | 2001-06-11 | 2004-11-16 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
US7232924B2 (en) * | 2001-06-11 | 2007-06-19 | Xenoport, Inc. | Methods for synthesis of acyloxyalkyl derivatives of GABA analogs |
US8048917B2 (en) * | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
US7186855B2 (en) | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
WO2004108733A1 (en) * | 2003-06-05 | 2004-12-16 | Pfizer Products Inc. | Beta-lactamase inhibitor prodrug |
JP5013795B2 (ja) * | 2006-09-25 | 2012-08-29 | Meiji Seikaファルマ株式会社 | 経口投与用カルバペネム |
WO2018030840A1 (ko) * | 2016-08-12 | 2018-02-15 | 가톨릭대학교 산학협력단 | 연조직 경화용 조성물 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2205310A1 (en) * | 1972-11-08 | 1974-05-31 | Aries Robert | Alpha penicillanamido penicillanic acids - long acting antibacterials prepd. by amidation of a mixed anhydride with an alpha amino penicillin |
GB1493197A (en) * | 1975-07-04 | 1977-11-23 | Beecham Group Ltd | Amides of clavulanic acid |
US4234579A (en) * | 1977-06-07 | 1980-11-18 | Pfizer Inc. | Penicillanic acid 1,1-dioxides as β-lactamase inhibitors |
US4244951A (en) * | 1979-05-16 | 1981-01-13 | Pfizer Inc. | Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide |
US4287181A (en) * | 1979-10-22 | 1981-09-01 | Pfizer Inc. | Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors |
US4323499A (en) * | 1981-01-05 | 1982-04-06 | Pfizer Inc. | 6-(2-Aryl-2-(1,1-dioxopenicillanoyloxy-methoxycarbonyl)acetamido penicillanic acids |
-
1982
- 1982-05-10 US US06/376,487 patent/US4377590A/en not_active Expired - Lifetime
-
1983
- 1983-05-03 GR GR71278A patent/GR78248B/el unknown
- 1983-05-09 EP EP83302585A patent/EP0094227B1/de not_active Expired
- 1983-05-09 DK DK206183A patent/DK206183A/da not_active Application Discontinuation
- 1983-05-09 DE DE8383302585T patent/DE3362396D1/de not_active Expired
- 1983-05-09 IE IE1060/83A patent/IE54771B1/en unknown
- 1983-05-10 JP JP58081602A patent/JPS58213788A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP0094227A1 (de) | 1983-11-16 |
DK206183D0 (da) | 1983-05-09 |
GR78248B (de) | 1984-09-26 |
IE831060L (en) | 1983-11-10 |
JPS58213788A (ja) | 1983-12-12 |
IE54771B1 (en) | 1990-01-31 |
DK206183A (da) | 1983-12-22 |
EP0094227B1 (de) | 1986-03-05 |
US4377590A (en) | 1983-03-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8328 | Change in the person/name/address of the agent |
Free format text: LEDERER, F., DIPL.-CHEM. DR., PAT.-ANW., 8000 MUENCHEN |
|
8339 | Ceased/non-payment of the annual fee |