DD133150A5 - METHOD FOR THE PRODUCTION OF MULTIPLE HALOGENATED STEROIDS - Google Patents

METHOD FOR THE PRODUCTION OF MULTIPLE HALOGENATED STEROIDS

Info

Publication number: DD133150A5
Authority: DD; German Democratic Republic
Prior art keywords: production; multiple halogenated; halogenated steroids; steroids; halogenated
Prior art date: 1976-09-29

Application number

DD7700201226A

Other languages

German (de)

Inventor

Jaroslav Kalvoda

Georg Anner

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-09-29

Filing date

1977-09-27

Publication date

1978-12-13

1977-09-27 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1978-12-13 Publication of DD133150A5 publication Critical patent/DD133150A5/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/008—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
- C07J7/0085—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by an halogen atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0061—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
- C07J5/0069—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
- C07J5/0076—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkyl group
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
- C07J71/0015—Oxiranes at position 9(11)

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Rheumatology (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DD7700201226A 1976-09-29 1977-09-27 METHOD FOR THE PRODUCTION OF MULTIPLE HALOGENATED STEROIDS DD133150A5 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
LU75903A LU75903A1 (en)	1976-09-29	1976-09-29

Publications (1)

Publication Number	Publication Date
DD133150A5 true DD133150A5 (en)	1978-12-13

Family

ID=19728370

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DD7700201226A DD133150A5 (en)	1976-09-29	1977-09-27	METHOD FOR THE PRODUCTION OF MULTIPLE HALOGENATED STEROIDS

Country Status (24)

Country	Link
JP (1)	JPS5356652A (en)
AT (3)	AT363197B (en)
AU (1)	AU514200B2 (en)
BE (1)	BE859120A (en)
CA (1)	CA1101410A (en)
CH (9)	CH624967A5 (en)
CY (1)	CY1178A (en)
DD (1)	DD133150A5 (en)
DE (1)	DE2743069A1 (en)
DK (1)	DK146017C (en)
ES (1)	ES462763A1 (en)
FR (1)	FR2366311A1 (en)
GB (1)	GB1563638A (en)
HK (1)	HK16683A (en)
HU (1)	HU175218B (en)
IE (1)	IE46047B1 (en)
IL (1)	IL53012A (en)
KE (1)	KE3258A (en)
LU (1)	LU75903A1 (en)
MY (1)	MY8400092A (en)
NL (1)	NL7710089A (en)
SE (1)	SE436751B (en)
SG (1)	SG3383G (en)
ZA (1)	ZA775800B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL187577C (en) *	1978-04-05	1991-11-18	Sibla Srl	3-ACETOXY-9BETA, 11BETA-EPOXY-PREGNA-1,3,5-TRIEN, PROCESS FOR THE PREPARATION THEREOF, AND PROCESS FOR THE PREPARATION OF 6-alpha-halogen-1,4-diene-3-ones.
DE3227312A1 (en) *	1982-07-19	1984-01-19	Schering AG, 1000 Berlin und 4709 Bergkamen	NEW 6.16 DIMETHYL CORTICOIDS, THEIR PRODUCTION AND USE
EP0523132A1 (en) *	1990-03-27	1993-01-20	Schering Corporation	PROCESS FOR 9$g(a)-HYDROXY STEROID DEHYDRATION
US5972922A (en) *	1990-06-11	1999-10-26	Alcon Laboratories, Inc.	Steroids which inhibit angiogenesis
MXPA04005188A (en)	2001-11-29	2004-08-11	Taro Pharma Ind	Method for the production of 6-alpha-fluoro corticosteroids.
US8809307B2 (en)	2010-11-22	2014-08-19	Dow Pharmaceutical Sciences, Inc.	Pharmaceutical formulations containing corticosteroids for topical administration
US11957753B2 (en)	2010-11-22	2024-04-16	Bausch Health Ireland Limited	Pharmaceutical formulations containing corticosteroids for topical administration
ES2812451T3 (en)	2015-06-18	2021-03-17	Bausch Health Ireland Ltd	Topical compositions comprising a corticosteroid and a retinoid to treat psoriasis

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB898292A (en) *	1959-03-18	1962-06-06	Upjohn Co	Improvements in or relating to steroids and the manufacture thereof
US3644340A (en) *	1970-03-19	1972-02-22	Syntex Corp	Preparation of 21-chloro steroids
US3992422A (en) *	1975-08-14	1976-11-16	Schering Corporation	Process for the preparation of 21-halogeno-21-desoxy-17α-acyloxy-20-keto-pregnenes

1976
- 1976-09-29 LU LU75903A patent/LU75903A1/xx unknown
- 1976-12-09 CH CH1549976A patent/CH624967A5/en not_active IP Right Cessation
1977
- 1977-06-08 SE SE7706673A patent/SE436751B/en not_active IP Right Cessation
- 1977-06-09 DK DK256977A patent/DK146017C/en not_active IP Right Cessation
- 1977-09-14 NL NL7710089A patent/NL7710089A/en not_active Application Discontinuation
- 1977-09-24 DE DE19772743069 patent/DE2743069A1/en active Granted
- 1977-09-26 CH CH1172177A patent/CH632279A5/en not_active IP Right Cessation
- 1977-09-27 FR FR7729043A patent/FR2366311A1/en active Granted
- 1977-09-27 CA CA287,560A patent/CA1101410A/en not_active Expired
- 1977-09-27 GB GB40131/77A patent/GB1563638A/en not_active Expired
- 1977-09-27 AU AU29148/77A patent/AU514200B2/en not_active Expired
- 1977-09-27 CY CY1178A patent/CY1178A/en unknown
- 1977-09-27 DD DD7700201226A patent/DD133150A5/en unknown
- 1977-09-28 IL IL53012A patent/IL53012A/en unknown
- 1977-09-28 ZA ZA00775800A patent/ZA775800B/en unknown
- 1977-09-28 IE IE1979/77A patent/IE46047B1/en not_active IP Right Cessation
- 1977-09-28 HU HU77CI1774A patent/HU175218B/en unknown
- 1977-09-28 BE BE181243A patent/BE859120A/en not_active IP Right Cessation
- 1977-09-28 AT AT0691077A patent/AT363197B/en not_active IP Right Cessation
- 1977-09-29 JP JP11619377A patent/JPS5356652A/en active Granted
- 1977-09-29 ES ES462763A patent/ES462763A1/en not_active Expired
1979
- 1979-02-28 AT AT0151279A patent/AT363202B/en not_active IP Right Cessation
- 1979-02-28 AT AT0151379A patent/AT363203B/en not_active IP Right Cessation
1980
- 1980-11-18 CH CH853780A patent/CH625808A5/en not_active IP Right Cessation
- 1980-11-18 CH CH853980A patent/CH625810A5/en not_active IP Right Cessation
- 1980-11-18 CH CH853880A patent/CH625809A5/en not_active IP Right Cessation
1981
- 1981-10-26 CH CH683281A patent/CH632000A5/en not_active IP Right Cessation
- 1981-10-26 CH CH683181A patent/CH631999A5/en not_active IP Right Cessation
- 1981-10-26 CH CH683081A patent/CH631998A5/en not_active IP Right Cessation
1982
- 1982-01-06 CH CH4682A patent/CH632521A5/en not_active IP Right Cessation
1983
- 1983-01-20 SG SG33/83A patent/SG3383G/en unknown
- 1983-01-21 KE KE3258A patent/KE3258A/en unknown
- 1983-05-19 HK HK166/83A patent/HK16683A/en not_active IP Right Cessation
1984
- 1984-12-30 MY MY92/84A patent/MY8400092A/en unknown

Also Published As

Publication number	Publication date
CH631999A5 (en)	1982-09-15
CH624967A5 (en)	1981-08-31
CH632000A5 (en)	1982-09-15
FR2366311B1 (en)	1982-12-03
AU2914877A (en)	1979-04-05
HU175218B (en)	1980-06-28
AT363202B (en)	1981-07-27
CA1101410A (en)	1981-05-19
IE46047L (en)	1978-03-29
DE2743069A1 (en)	1978-03-30
CH632279A5 (en)	1982-09-30
ZA775800B (en)	1978-08-30
JPS5356652A (en)	1978-05-23
IL53012A0 (en)	1977-11-30
ATA151379A (en)	1980-12-15
AT363203B (en)	1981-07-27
HK16683A (en)	1983-05-27
CH631998A5 (en)	1982-09-15
JPS6214557B2 (en)	1987-04-02
DE2743069C2 (en)	1987-03-05
SE436751B (en)	1985-01-21
DK146017B (en)	1983-05-24
MY8400092A (en)	1984-12-31
SG3383G (en)	1983-09-09
ES462763A1 (en)	1978-05-16
NL7710089A (en)	1978-03-31
IL53012A (en)	1982-05-31
FR2366311A1 (en)	1978-04-28
CH625810A5 (en)	1981-10-15
KE3258A (en)	1983-03-04
ATA151279A (en)	1980-12-15
CH625808A5 (en)	1981-10-15
ATA691077A (en)	1980-12-15
IE46047B1 (en)	1983-02-09
AU514200B2 (en)	1981-01-29
CY1178A (en)	1983-06-10
CH625809A5 (en)	1981-10-15
SE7706673L (en)	1978-03-30
BE859120A (en)	1978-03-28
GB1563638A (en)	1980-03-26
DK146017C (en)	1983-10-24
AT363197B (en)	1981-07-10
CH632521A5 (en)	1982-10-15
DK256977A (en)	1978-03-30
LU75903A1 (en)	1978-05-16

Publication	Publication Date	Title
DD134224A5 (en)	1979-02-14	METHOD FOR THE PRODUCTION OF SUBSTITUTED AMINOSAURES
DD128672A5 (en)	1977-11-30	PROCESS FOR THE PREPARATION OF M-ARYLOXYBENZALDEHYDE
AT348995B (en)	1979-03-12	PROCESS FOR THE PREPARATION OF ACYLCYANIDES
DD129777A5 (en)	1978-02-08	PROCESS FOR THE PREPARATION OF PHENOXYPROPIONSAEUREDERIVATES
DD128659A5 (en)	1977-11-30	PROCESS FOR THE PREPARATION OF 4-ANDROST-3-ONEN
AT347926B (en)	1979-01-25	PROCESS FOR THE PREPARATION OF ACYLCYANIDES
DD133150A5 (en)	1978-12-13	METHOD FOR THE PRODUCTION OF MULTIPLE HALOGENATED STEROIDS
DD129903A5 (en)	1978-02-15	PROCESS FOR THE PREPARATION OF BENZOYLCYANIDE
AT352753B (en)	1979-10-10	METHOD FOR THE PRODUCTION OF METHYL DICHLORPHOSPHANE
AT348509B (en)	1979-02-26	PROCESS FOR THE PREPARATION OF ACYLCYANIDES
AT349454B (en)	1979-04-10	PROCESS FOR THE PRODUCTION OF ALFA-CYANO-BENZYLESTERS
ATA980876A (en)	1979-07-15	PROCESS FOR THE PRODUCTION OF 2-OXO-PYRROLIDINE-N-ALKYLAMIDES
AT351676B (en)	1979-08-10	METHOD FOR THE PRODUCTION OF 7-ALKOXY-3-CHLORMETHYL-3-CEPHEMES
AT357280B (en)	1980-06-25	METHOD FOR THE PRODUCTION OF 17ALPHA- -ALKINYL-ANDROST-4-ENDERIVATEN
DD129782A5 (en)	1978-02-08	PROCESS FOR THE PREPARATION OF CHOLECYSTOKININ-PANCREOZYMIN OCTAPEPTIDAMIDE SULFATESTER
DD128591A5 (en)	1977-11-30	PROCESS FOR THE PREPARATION OF 2-OXO-1-PYRROLIDINES
DD128953A1 (en)	1977-12-21	PROCESS FOR THE PREPARATION OF ALKALICELLULOSE
DD129792A5 (en)	1978-02-08	PROCESS FOR THE PREPARATION OF 1-OXADETHIACEPHALOSPORINES
DD129980A5 (en)	1978-02-22	PROCESS FOR THE PREPARATION OF TRANS-DIHYDROINDOLSES
AT348506B (en)	1979-02-26	PROCESS FOR THE PRODUCTION OF BIS-POLYBROMPHENOXY-ALKANES
DD128663A1 (en)	1977-11-30	METHOD FOR THE CONTINUOUS PRODUCTION OF PERESTERN
AT345786B (en)	1978-10-10	PROCESS FOR THE PREPARATION OF O-DIALKYLAMINOMETHYLPHENOLS
DD128749A1 (en)	1977-12-07	PROCESS FOR THE PREPARATION OF HEXABROMBENZOL
DD127931A1 (en)	1977-10-19	PROCESS FOR THE PREPARATION OF BENZIMIDAZOLENE
AT347918B (en)	1979-01-25	PROCESS FOR THE PRODUCTION OF HEXACHLOROCYCLOBUTEN