CY1122712T1 - ΧΡΗΣΗ ΠΑΡΑΓΩΓΩΝ ΠΥΡΑΖΟΛΟΠΥΡΙΜΙΔΙΝΗΣ ΓΙΑ ΤΗ ΘΕΡΑΠΕΙΑ ΣΧΕΤΙΚΩΝ ΜΕ PI3Kδ ΔΙΑΤΑΡΑΧΩΝ - Google Patents
ΧΡΗΣΗ ΠΑΡΑΓΩΓΩΝ ΠΥΡΑΖΟΛΟΠΥΡΙΜΙΔΙΝΗΣ ΓΙΑ ΤΗ ΘΕΡΑΠΕΙΑ ΣΧΕΤΙΚΩΝ ΜΕ PI3Kδ ΔΙΑΤΑΡΑΧΩΝInfo
- Publication number
- CY1122712T1 CY1122712T1 CY20201100177T CY201100177T CY1122712T1 CY 1122712 T1 CY1122712 T1 CY 1122712T1 CY 20201100177 T CY20201100177 T CY 20201100177T CY 201100177 T CY201100177 T CY 201100177T CY 1122712 T1 CY1122712 T1 CY 1122712T1
- Authority
- CY
- Cyprus
- Prior art keywords
- related disorders
- treatment
- pyrazolopyrimidine derivatives
- pi3kδ
- pi3kδ related
- Prior art date
Links
- OGEBRHQLRGFBNV-RZDIXWSQSA-N chembl2036808 Chemical class C12=NC(NCCCC)=NC=C2C(C=2C=CC(F)=CC=2)=NN1C[C@H]1CC[C@H](N)CC1 OGEBRHQLRGFBNV-RZDIXWSQSA-N 0.000 title 1
- 102000038030 PI3Ks Human genes 0.000 abstract 1
- 108091007960 PI3Ks Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
Η παρούσα δήλωση παρέχει μεθόδους θεραπείας σχετικών με ΡΙ3Κδ διαταραχών χρησιμοποιώντας ενώσεις του Τύπου (Ι): ή φαρμακευτικώς αποδεκτά άλατα αυτών.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361771480P | 2013-03-01 | 2013-03-01 | |
PCT/US2014/019372 WO2014134426A1 (en) | 2013-03-01 | 2014-02-28 | USE OF PYRAZOLOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PI3Kδ RELATED DISORDERS |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1122712T1 true CY1122712T1 (el) | 2021-03-12 |
Family
ID=50288319
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20201100177T CY1122712T1 (el) | 2013-03-01 | 2020-02-26 | ΧΡΗΣΗ ΠΑΡΑΓΩΓΩΝ ΠΥΡΑΖΟΛΟΠΥΡΙΜΙΔΙΝΗΣ ΓΙΑ ΤΗ ΘΕΡΑΠΕΙΑ ΣΧΕΤΙΚΩΝ ΜΕ PI3Kδ ΔΙΑΤΑΡΑΧΩΝ |
Country Status (32)
Country | Link |
---|---|
US (5) | US9932341B2 (el) |
EP (3) | EP4233869A3 (el) |
JP (4) | JP6545106B2 (el) |
KR (4) | KR20230145517A (el) |
CN (2) | CN105120871B (el) |
AR (1) | AR094964A1 (el) |
AU (4) | AU2014223257B2 (el) |
BR (1) | BR112015020941A2 (el) |
CA (1) | CA2901993C (el) |
CL (1) | CL2015002442A1 (el) |
CR (1) | CR20150472A (el) |
CY (1) | CY1122712T1 (el) |
DK (1) | DK2961410T3 (el) |
EA (2) | EA202192151A1 (el) |
ES (2) | ES2774436T3 (el) |
HK (1) | HK1221398A1 (el) |
HR (1) | HRP20200263T1 (el) |
HU (1) | HUE047719T2 (el) |
IL (5) | IL301180A (el) |
LT (1) | LT2961410T (el) |
MX (2) | MX367713B (el) |
MY (1) | MY177875A (el) |
PE (1) | PE20151996A1 (el) |
PH (2) | PH12015501920A1 (el) |
PL (1) | PL2961410T3 (el) |
PT (1) | PT2961410T (el) |
RS (1) | RS59958B1 (el) |
SG (3) | SG10201912275YA (el) |
SI (1) | SI2961410T1 (el) |
TW (4) | TWI657090B (el) |
UA (1) | UA119641C2 (el) |
WO (1) | WO2014134426A1 (el) |
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KR20220066179A (ko) | 2014-04-08 | 2022-05-23 | 인사이트 코포레이션 | Jak 및 pi3k 억제제 조합에 의한 b-세포 악성종양의 치료 |
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2014
- 2014-02-27 TW TW103106906A patent/TWI657090B/zh active
- 2014-02-27 TW TW108100664A patent/TWI687220B/zh active
- 2014-02-27 TW TW110124946A patent/TW202214254A/zh unknown
- 2014-02-27 TW TW109104878A patent/TWI736135B/zh active
- 2014-02-28 PE PE2015001833A patent/PE20151996A1/es not_active Application Discontinuation
- 2014-02-28 AR ARP140100679A patent/AR094964A1/es unknown
- 2014-02-28 MX MX2015011273A patent/MX367713B/es active IP Right Grant
- 2014-02-28 SG SG10201912275YA patent/SG10201912275YA/en unknown
- 2014-02-28 EP EP23161858.8A patent/EP4233869A3/en active Pending
- 2014-02-28 UA UAA201509435A patent/UA119641C2/uk unknown
- 2014-02-28 CA CA2901993A patent/CA2901993C/en active Active
- 2014-02-28 MY MYPI2015002108A patent/MY177875A/en unknown
- 2014-02-28 KR KR1020237033761A patent/KR20230145517A/ko not_active Application Discontinuation
- 2014-02-28 ES ES14710739T patent/ES2774436T3/es active Active
- 2014-02-28 US US14/193,481 patent/US9932341B2/en active Active
- 2014-02-28 EP EP19208523.1A patent/EP3632442B1/en active Active
- 2014-02-28 EP EP14710739.5A patent/EP2961410B1/en active Active
- 2014-02-28 AU AU2014223257A patent/AU2014223257B2/en active Active
- 2014-02-28 WO PCT/US2014/019372 patent/WO2014134426A1/en active Application Filing
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- 2014-02-28 KR KR1020217027697A patent/KR102454308B1/ko active IP Right Grant
- 2014-02-28 PL PL14710739T patent/PL2961410T3/pl unknown
- 2014-02-28 JP JP2015560346A patent/JP6545106B2/ja active Active
- 2014-02-28 EA EA202192151A patent/EA202192151A1/ru unknown
- 2014-02-28 RS RS20200176A patent/RS59958B1/sr unknown
- 2014-02-28 LT LTEP14710739.5T patent/LT2961410T/lt unknown
- 2014-02-28 EA EA201591612A patent/EA201591612A1/ru unknown
- 2014-02-28 SI SI201431449T patent/SI2961410T1/sl unknown
- 2014-02-28 BR BR112015020941A patent/BR112015020941A2/pt not_active Application Discontinuation
- 2014-02-28 DK DK14710739.5T patent/DK2961410T3/da active
- 2014-02-28 IL IL301180A patent/IL301180A/en unknown
- 2014-02-28 SG SG10201707130UA patent/SG10201707130UA/en unknown
- 2014-02-28 CN CN201480021187.1A patent/CN105120871B/zh active Active
- 2014-02-28 KR KR1020227035039A patent/KR102586858B1/ko active IP Right Grant
- 2014-02-28 CN CN201810796220.8A patent/CN109010343A/zh active Pending
- 2014-02-28 HU HUE14710739A patent/HUE047719T2/hu unknown
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- 2014-02-28 KR KR1020157027010A patent/KR102298150B1/ko active IP Right Grant
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2015
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2016
- 2016-06-07 HK HK16106523.5A patent/HK1221398A1/zh unknown
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2018
- 2018-03-02 US US15/910,708 patent/US20190040067A1/en not_active Abandoned
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2019
- 2019-04-25 JP JP2019084393A patent/JP6776399B2/ja active Active
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2020
- 2020-02-17 HR HRP20200263TT patent/HRP20200263T1/hr unknown
- 2020-02-26 CY CY20201100177T patent/CY1122712T1/el unknown
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2021
- 2021-06-13 IL IL283943A patent/IL283943B2/en unknown
- 2021-06-30 US US17/364,695 patent/US20210332059A1/en active Pending
- 2021-06-30 US US17/364,551 patent/US20220106318A1/en active Pending
- 2021-06-30 US US17/364,585 patent/US20220119393A1/en active Pending
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2022
- 2022-08-16 AU AU2022218495A patent/AU2022218495A1/en active Pending
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