CY1117026T1 - Ετεροκυκλικες ενωσεις για αντιμετωπιση ή προληψη διαταραχων που προκαλουνται απο μειωμενη νευροδιαβιβαση σεροτονινης, νορεπινεφρινης ή ντοπαμινης - Google Patents

Ετεροκυκλικες ενωσεις για αντιμετωπιση ή προληψη διαταραχων που προκαλουνται απο μειωμενη νευροδιαβιβαση σεροτονινης, νορεπινεφρινης ή ντοπαμινης

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Publication number
CY1117026T1
CY1117026T1 CY20151101119T CY151101119T CY1117026T1 CY 1117026 T1 CY1117026 T1 CY 1117026T1 CY 20151101119 T CY20151101119 T CY 20151101119T CY 151101119 T CY151101119 T CY 151101119T CY 1117026 T1 CY1117026 T1 CY 1117026T1
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CY
Cyprus
Prior art keywords
group
nerpin
prevention
treatment
heterocyclic compounds
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Application number
CY20151101119T
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English (en)
Inventor
Nobuaki Ito
Hirofumi Sasaki
Kuninori Tai
Tomoichi Shinohara
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Otsuka Pharmaceutical Co., Ltd
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Publication date
Application filed by Otsuka Pharmaceutical Co., Ltd filed Critical Otsuka Pharmaceutical Co., Ltd
Publication of CY1117026T1 publication Critical patent/CY1117026T1/el

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Abstract

Μία ετεροκυκλική ένωση που παριστάνεται με τον γενικό τύπο (1) ή ένα άλας αυτής: όπου τα m, 1, και n αντίστοιχα παριστάνουν έναν ακέραιο 1 ή 2 · το Χ παριστάνει -Ο- ή -CH2- · το R1 παριστάνει υδρογόνο, μία ομάδα κατώτερου αλκυλίου, μία υδροξυ - ομάδα κατώτερου αλκυλίου, μία προστατευτική ομάδα, ή μία ομάδα τρι-κατώτερου αλκυλοσιλυλοξειδίου - κατώτερου αλκυλίου · τα R2 και R3, που είναι τα ίδια ή διαφορετικά, το κάθε ένα ανεξάρτητα παριστάνει υδρογόνο ή μία ομάδα κατώτερου αλκυλίου · ή τα R2 και R3 είναι συνδεδεμένα ώστε να σχηματίζουν μία ομάδα κυκλο-C3-C8 αλκυλίου · και το R4 παριστάνει μία αρωματική ομάδα ή μία ετεροκυκλική ομάδα, όπου η αρωματική ή ετεροκυκλική ομάδα μπορεί να έχει έναν ή περισσότερους αυθαίρετους υποκατάστατες.
CY20151101119T 2010-09-13 2015-12-08 Ετεροκυκλικες ενωσεις για αντιμετωπιση ή προληψη διαταραχων που προκαλουνται απο μειωμενη νευροδιαβιβαση σεροτονινης, νορεπινεφρινης ή ντοπαμινης CY1117026T1 (el)

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EP11764005.2A EP2616460B1 (en) 2010-09-13 2011-09-12 Heterocyclic compounds for treating or preventing disorders caused by reduced neurotransmission of serotonin, norephnephrine or dopamine.

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