CY1114767T1 - Ν,ν-υποκατεστημενες ενωσεις 3-αμινοπυρρολιδινης χρησιμες ως αναστολεις επαναπροσληψης μονοαμινων - Google Patents

Ν,ν-υποκατεστημενες ενωσεις 3-αμινοπυρρολιδινης χρησιμες ως αναστολεις επαναπροσληψης μονοαμινων

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Publication number
CY1114767T1
CY1114767T1 CY20141100049T CY141100049T CY1114767T1 CY 1114767 T1 CY1114767 T1 CY 1114767T1 CY 20141100049 T CY20141100049 T CY 20141100049T CY 141100049 T CY141100049 T CY 141100049T CY 1114767 T1 CY1114767 T1 CY 1114767T1
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CY
Cyprus
Prior art keywords
monoamines
substituted
compounds useful
salt
halogen atoms
Prior art date
Application number
CY20141100049T
Other languages
English (en)
Inventor
Muneaki Kurimura
Shinichi Taira
Takahiro Tomoyasu
Nobuaki Ito
Kuninori Tai
Noriaki Takemura
Takayuki Matsuzaki
Yasuhiro Menjo
Shin Miyamura
Yohji Sakurai
Akihito Watanabe
Yasuyo Sakata
Takumi Masumoto
Kohei Akazawa
Haruhiko Sugino
Naoki Amada
Satoshi Ohashi
Tomoichi Shinohara
Hirofumi Sasaki
Chisako Morita
Junko Yamashita
Satoko Nakajima
Original Assignee
Otsuka Pharmaceutical Co., Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36693623&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1114767(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharmaceutical Co., Ltd filed Critical Otsuka Pharmaceutical Co., Ltd
Publication of CY1114767T1 publication Critical patent/CY1114767T1/el

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Abstract

Η παρούσα εφεύρεση παρέχει μια ένωση πυρρολιδίνης του Γενικού Χημικού Τύπου (1) ή ένα άλας εξ αυτής, όπου τα R101 και R102 είναι το κάθε ένα ανεξαρτήτως μια ομάδα φαινυλίου, οι οποίες μπορεί να έχουν ένα ή περισσότερα υποκατάστατα που επιλέγονται από άτομα αλογόνου και ομάδες κατώτερου αλκυλίου προαιρετικώς υποκατεστημένες με ένα ή περισσότερα άτομα αλογόνου, κλπ. Η ένωση πυρρολιδίνης ή ένα άλας εξ αυτής της παρούσας εφεύρεσης είναι χρησιμοποιήσιμη για την παραγωγή ενός φαρμακευτικού παρασκευάσματος έχοντας ένα ευρύτερο θεραπευτικό φάσμα και όντας δυνάμενη εκδήλωσης επαρκών θεραπευτικών επιδράσεων μετά από βραχυχρόνια χορήγηση.
CY20141100049T 2005-05-13 2014-01-20 Ν,ν-υποκατεστημενες ενωσεις 3-αμινοπυρρολιδινης χρησιμες ως αναστολεις επαναπροσληψης μονοαμινων CY1114767T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2005141230 2005-05-13
EP11185205.9A EP2407451B1 (en) 2005-05-13 2006-05-12 N,N-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors

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CY1114767T1 true CY1114767T1 (el) 2016-12-14

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WO2004050024A2 (en) 2002-11-27 2004-06-17 Incyte Corporation 3-aminopyrrolidine derivatives as modulators of chemokine receptors
TWI449692B (zh) * 2005-05-13 2014-08-21 Otsuka Pharma Co Ltd 吡咯烷化合物（三）
BRPI0619263A2 (pt) * 2005-11-30 2011-09-27 Hoffmann La Roche indóis de 3-amino-1-arilpropila e indóis aza-substituìdos, métodos para prepará-los, composição farmacêutica e uso dos referidos indóis
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