CY1107500T1 - Η χρηση του φλουμαζενιλ στην αναπτυξη ενος φαρμακου για τη θepαπευτικη αντιμετωπιση της εξαρτησης απο το αλκοολ - Google Patents
Η χρηση του φλουμαζενιλ στην αναπτυξη ενος φαρμακου για τη θepαπευτικη αντιμετωπιση της εξαρτησης απο το αλκοολInfo
- Publication number
- CY1107500T1 CY1107500T1 CY20061101651T CY061101651T CY1107500T1 CY 1107500 T1 CY1107500 T1 CY 1107500T1 CY 20061101651 T CY20061101651 T CY 20061101651T CY 061101651 T CY061101651 T CY 061101651T CY 1107500 T1 CY1107500 T1 CY 1107500T1
- Authority
- CY
- Cyprus
- Prior art keywords
- flumazenil
- drug
- development
- alternative treatment
- alcohol addiction
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
- A61K31/5517—1,4-Benzodiazepines, e.g. diazepam or clozapine condensed with five-membered rings having nitrogen as a ring hetero atom, e.g. imidazobenzodiazepines, triazolam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Addiction (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Silver Salt Photography Or Processing Solution Therefor (AREA)
Abstract
Η εφεύρεση αφορά στη χρήση του φλουμαζενίλ στην ανάπτυξη ενός φαρμάκου που χρησιμοποιείται για τη διαδοχική χορήγηση μικρών ποσοτήτων φλουμαζενίλ κατά πυκνά διαστήματα, μέχρις ότου χορηγηθεί μια θεραπευτικά αποτελεσματική ποσότητα για να αντιμετωπισθεί η εξάρτηση από το αλκοόλ.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES200100106 | 2001-01-17 | ||
EP02716090A EP1374952B1 (en) | 2001-01-17 | 2002-01-10 | Use of flumazenil in developing a drug for the treatment of alcohol dependence |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1107500T1 true CY1107500T1 (el) | 2013-03-13 |
Family
ID=8496426
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20061101651T CY1107500T1 (el) | 2001-01-17 | 2006-11-14 | Η χρηση του φλουμαζενιλ στην αναπτυξη ενος φαρμακου για τη θepαπευτικη αντιμετωπιση της εξαρτησης απο το αλκοολ |
Country Status (23)
Country | Link |
---|---|
US (2) | US7348321B2 (el) |
EP (1) | EP1374952B1 (el) |
JP (2) | JP2004519461A (el) |
KR (1) | KR100712570B1 (el) |
CN (1) | CN1486205A (el) |
AT (1) | ATE338575T1 (el) |
AU (1) | AU2002226427B2 (el) |
BR (1) | BR0206549A (el) |
CA (1) | CA2433833C (el) |
CR (1) | CR7049A (el) |
CY (1) | CY1107500T1 (el) |
DE (1) | DE60214527T2 (el) |
DK (1) | DK1374952T3 (el) |
ES (1) | ES2269661T3 (el) |
HK (1) | HK1061661A1 (el) |
IL (1) | IL156798A0 (el) |
MX (1) | MXPA03006411A (el) |
NZ (2) | NZ527583A (el) |
PT (1) | PT1374952E (el) |
RU (1) | RU2300378C2 (el) |
UA (1) | UA78199C2 (el) |
WO (1) | WO2002056964A1 (el) |
ZA (1) | ZA200305922B (el) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20050192271A1 (en) | 2003-07-15 | 2005-09-01 | Hythiam, Inc. | Use of selective chloride channel modulators to treat alcohol and/or stimulant substance abuse |
US20060172998A1 (en) * | 2005-02-03 | 2006-08-03 | Halikas James A | Method of preventing relapse in the abstinent substance dependent individual |
US20060172996A1 (en) * | 2005-02-03 | 2006-08-03 | Halikas James A | Method of preventing relapse in the abstinent substance dependent individual |
EP1868593A2 (en) * | 2005-04-07 | 2007-12-26 | Hythiam, Inc. | Improved methods of and compositions for the prevention of anxiety, substance abuse, and dependence |
US20060263304A1 (en) * | 2005-05-23 | 2006-11-23 | Halikas James A | Method of controlling alcohol intake and reversing alcohol effects |
SG183696A1 (en) * | 2007-08-06 | 2012-09-27 | Biotie Therapies Inc | Medicaments comprising nepicastat for use in treating dependence on a substance |
EP2186517A4 (en) * | 2007-08-08 | 2010-08-18 | Ibanez Juan Jose Legarda | USE AND METHODS OF USING A SEROTONIN3 (5-HT3) RECEPTOR ANTAGONIST AND CHLORIDE CHANNEL MODULATOR FOR THE TREATMENT OF DRUG OR DRUG ADDICTION OR DEPENDENCE OR CENTER NERVOUS DISORDERS |
AU2010215075B2 (en) * | 2009-02-20 | 2015-08-20 | Palmaya Pty Ltd | Pharmaceutical preparation and delivery system |
US8930050B2 (en) * | 2009-04-29 | 2015-01-06 | Marine Canada Acquisition Inc. | Method and system for increasing or decreasing engine throttle in a marine vessel |
US20100280684A1 (en) * | 2009-04-29 | 2010-11-04 | Pierre Garon | Synchronization of shift and throttle controls in a marine vessel |
US8347859B2 (en) * | 2009-04-29 | 2013-01-08 | Marine Canada Acquisition Inc. | Automatic throttle calibration in a marine vessel |
US8387589B2 (en) * | 2009-04-29 | 2013-03-05 | Marine Canada Acqusition Inc. | Position sensor for an output shaft used in a shift and throttle system |
US8406944B2 (en) * | 2010-02-10 | 2013-03-26 | Pierre Garon | Control system and method for starting and stopping marine engines |
US8845490B2 (en) | 2010-02-10 | 2014-09-30 | Marine Canada Acquisition Inc. | Method and system for delaying shift and throttle commands based on engine speed in a marine vessel |
US8182396B2 (en) * | 2010-02-10 | 2012-05-22 | Marine Canada Acquisition In.c | Method and system for delaying shift and throttle commands based on engine speed in a marine vessel |
AU2012221704B2 (en) | 2011-02-23 | 2013-12-05 | Coeruleus Ltd. | Flumazenil complexes, compositions comprising same and uses thereof |
RU2468799C1 (ru) * | 2011-08-03 | 2012-12-10 | Общество с ограниченной ответственностью "Урал Крафт" | Способ купирования алкогольного абстинентного синдрома посредством блокады бензодиазепиновых рецепторов |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5519017A (en) * | 1990-03-29 | 1996-05-21 | Lts Lohmann Therapie-Systeme Gmbh + Co. Kg | Pharmaceutic formulation for the treatment of alcoholism |
SE9100860D0 (sv) * | 1991-03-22 | 1991-03-22 | Kabi Pharmacia Ab | New use |
GB9420010D0 (en) | 1994-10-01 | 1994-11-16 | Marck Sharp & Dohme Limited | Nucleic acids |
US20030176456A1 (en) * | 2001-12-21 | 2003-09-18 | June Harry L. | Methods for reducing alcohol cravings in chronic alcoholics |
US6740677B2 (en) | 2002-08-19 | 2004-05-25 | Hong Xue | Methods of treating benzodiazepine site (BZD-S) associated syndromes using 2′ hydroxyflavonoids |
-
2002
- 2002-01-10 JP JP2002557469A patent/JP2004519461A/ja active Pending
- 2002-01-10 KR KR1020037009461A patent/KR100712570B1/ko not_active IP Right Cessation
- 2002-01-10 CN CNA028038029A patent/CN1486205A/zh active Pending
- 2002-01-10 CA CA002433833A patent/CA2433833C/en not_active Expired - Fee Related
- 2002-01-10 NZ NZ527583A patent/NZ527583A/xx not_active IP Right Cessation
- 2002-01-10 RU RU2003125274/15A patent/RU2300378C2/ru not_active IP Right Cessation
- 2002-01-10 DK DK02716090T patent/DK1374952T3/da active
- 2002-01-10 MX MXPA03006411A patent/MXPA03006411A/es active IP Right Grant
- 2002-01-10 EP EP02716090A patent/EP1374952B1/en not_active Expired - Lifetime
- 2002-01-10 ZA ZA200305922A patent/ZA200305922B/en unknown
- 2002-01-10 AT AT02716090T patent/ATE338575T1/de active
- 2002-01-10 BR BR0206549-5A patent/BR0206549A/pt not_active Application Discontinuation
- 2002-01-10 AU AU2002226427A patent/AU2002226427B2/en not_active Ceased
- 2002-01-10 NZ NZ539400A patent/NZ539400A/en not_active IP Right Cessation
- 2002-01-10 ES ES02716090T patent/ES2269661T3/es not_active Expired - Lifetime
- 2002-01-10 WO PCT/ES2002/000008 patent/WO2002056964A1/es active IP Right Grant
- 2002-01-10 PT PT02716090T patent/PT1374952E/pt unknown
- 2002-01-10 DE DE60214527T patent/DE60214527T2/de not_active Expired - Lifetime
- 2002-01-10 IL IL15679802A patent/IL156798A0/xx unknown
- 2002-10-01 UA UA2003087768A patent/UA78199C2/uk unknown
-
2003
- 2003-07-15 US US10/621,229 patent/US7348321B2/en active Active
- 2003-08-06 CR CR7049A patent/CR7049A/es unknown
-
2004
- 2004-07-02 HK HK04104732A patent/HK1061661A1/xx not_active IP Right Cessation
-
2006
- 2006-11-14 CY CY20061101651T patent/CY1107500T1/el unknown
-
2008
- 2008-02-06 US US12/026,643 patent/US20080132492A1/en not_active Abandoned
- 2008-04-28 JP JP2008116697A patent/JP2008201796A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
HK1061661A1 (en) | 2004-09-30 |
NZ539400A (en) | 2006-04-28 |
DE60214527D1 (de) | 2006-10-19 |
RU2300378C2 (ru) | 2007-06-10 |
AU2002226427B2 (en) | 2006-11-16 |
PT1374952E (pt) | 2006-12-29 |
NZ527583A (en) | 2006-03-31 |
MXPA03006411A (es) | 2004-12-02 |
CR7049A (es) | 2008-02-20 |
BR0206549A (pt) | 2004-02-25 |
IL156798A0 (en) | 2004-02-08 |
ATE338575T1 (de) | 2006-09-15 |
KR100712570B1 (ko) | 2007-05-02 |
DK1374952T3 (da) | 2007-01-02 |
EP1374952A1 (en) | 2004-01-02 |
US20040092509A1 (en) | 2004-05-13 |
ES2269661T3 (es) | 2007-04-01 |
JP2004519461A (ja) | 2004-07-02 |
EP1374952B1 (en) | 2006-09-06 |
ZA200305922B (en) | 2004-08-02 |
JP2008201796A (ja) | 2008-09-04 |
CN1486205A (zh) | 2004-03-31 |
KR20040020046A (ko) | 2004-03-06 |
UA78199C2 (en) | 2007-03-15 |
RU2003125274A (ru) | 2005-01-20 |
US20080132492A1 (en) | 2008-06-05 |
DE60214527T2 (de) | 2007-04-05 |
US7348321B2 (en) | 2008-03-25 |
CA2433833A1 (en) | 2002-07-25 |
CA2433833C (en) | 2009-06-02 |
WO2002056964A1 (es) | 2002-07-25 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1107500T1 (el) | Η χρηση του φλουμαζενιλ στην αναπτυξη ενος φαρμακου για τη θepαπευτικη αντιμετωπιση της εξαρτησης απο το αλκοολ | |
CY1118651T1 (el) | Αζακυκλικες ενωσεις για χρηση στην θεραπευτικη αντιμετωπιση ασθενειων που σχετιζονται με τη σεροτονινη | |
CY1119369T1 (el) | Ιατρικα παρασκευασματα για τη θεραπευτικη αγωγη της ανεπαρκειας της αλφα-γαλακτοσιδασης α | |
CY1120977T1 (el) | Θεραπεια των ασθενειων αποθηκευσης γλυκογονου τυπου ιι | |
EA200101156A1 (ru) | ЛЕКАРСТВЕННЫЕ КОМПОЗИЦИИ НОВОГО ТИПА НА ОСНОВЕ ОБЛАДАЮЩИХ ХОЛИНЕРГИЧЕСКИМ ДЕЙСТВИЕМ СОЕДИНЕНИЙ И β-МИМЕТИКОВ | |
CY1106845T1 (el) | Χρηση της φλουμαζενιλης για την παρασκευη ενος φαρμακου για την αγωγη της εξαρτησεως απο την κοκαϊνη | |
JP2006501240A5 (el) | ||
TR200002786T2 (tr) | Meloksikam için yeni galenik bir formülasyon. | |
DE602004027936D1 (de) | Tocopherolmodifizierte therapeutische arzneimittelverbindung | |
ATE359077T1 (de) | Orale gabe von 6-hydroxy-oxymorphon als analgetikum | |
NO20101190L (no) | Anvendelse av buprenorfin i fremstillingen av et medikament | |
CY2009002I1 (el) | Χρηση αμινοξικων αντισπασμωδικων για τη θεραπευτικη αγωγη του πονου | |
EA200300503A1 (ru) | Новые лекарственные композиции на основе солей тиотропия и солей салметерола | |
CY1106122T1 (el) | Αναστολεις τρανσφepασης φαρνεσυλ πρωτεϊνης για τη θepαπευτικη αντιμετωπιση της νοσου ευepεθιστου εντερου | |
CY1111396T1 (el) | Ρινικη χορηγηση μετοκλοπραμιδης για την αγωγη της γαστροπαρεσης | |
EE200200107A (et) | Kiire algtoimega selektiivse serotoniini tagasihaaramise inhibiitori kasutamine ravimi valmistamiseks, mis on ette nähtud seksuaalse funktsioonihäireravimiseks | |
CY1109361T1 (el) | Υποκατεστημενες 4-αμινοκυκλοεξανολες | |
IS6558A (is) | Blandaðar sjúkdómsmeðferðir með æðaskaðandi virkni | |
IS2259B (is) | Aðferð til meðferðar á netjuhersli með notkun mótlyfs við integríninu alfa-4 undireiningunni | |
CY1105317T1 (el) | Χρηση υποκατεστημενων ενωσεων 6-διμεθυλαμινομεθυλο-1-φαινυλο-κυκλοεξανιου για τη θepαπεια της ακρατειας ουρων | |
CY1105142T1 (el) | Χρηση υποκατεστημενων ενωσεων 6-διμεθυλαμινομεθυλο-1-φαινυλο-κυκλοεξανιου για τη θepαπεια της ακρατειας ουρων | |
DE60134735D1 (de) | Neue neurokinin-antagonisten zum gebrauch als arzneimittel | |
EA200401303A1 (ru) | Лекарственные средства, содержащие стероиды и новое антихолинергическое средство | |
ATE302008T1 (de) | Behandlung von entzündlichen erkrankungen | |
SE0004827D0 (sv) | Therapeutic compounds |