CR7812A - Compuestos de purina y usos de los mismos como ligandos de receptor de cannabinoides - Google Patents

Compuestos de purina y usos de los mismos como ligandos de receptor de cannabinoides

Info

Publication number
CR7812A
CR7812A CR7812A CR7812A CR7812A CR 7812 A CR7812 A CR 7812A CR 7812 A CR7812 A CR 7812A CR 7812 A CR7812 A CR 7812A CR 7812 A CR7812 A CR 7812A
Authority
CR
Costa Rica
Prior art keywords
cannabinoid
compounds
purina
same
receiver links
Prior art date
Application number
CR7812A
Other languages
English (en)
Inventor
Andrew Griffith David
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of CR7812A publication Critical patent/CR7812A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/28—Oxygen atom
    • C07D473/30—Oxygen atom attached in position 6, e.g. hypoxanthine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Toxicology (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nutrition Science (AREA)
  • Immunology (AREA)

Abstract

Se describen en la memoria descriptiva compuestos de formula I que actuan como ligandos de receptor de cannabinoides y sus usos en el tratamiento de enfermedades ligadas a la medicion de los receptores de cannabinoide en animales.
CR7812A 2002-10-28 2005-04-28 Compuestos de purina y usos de los mismos como ligandos de receptor de cannabinoides CR7812A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42187402P 2002-10-28 2002-10-28

Publications (1)

Publication Number Publication Date
CR7812A true CR7812A (es) 2005-06-08

Family

ID=32176739

Family Applications (1)

Application Number Title Priority Date Filing Date
CR7812A CR7812A (es) 2002-10-28 2005-04-28 Compuestos de purina y usos de los mismos como ligandos de receptor de cannabinoides

Country Status (45)

Country Link
US (2) US7129239B2 (es)
EP (1) EP1558615B8 (es)
JP (2) JP3954618B2 (es)
KR (1) KR100674560B1 (es)
CN (3) CN100478343C (es)
AP (1) AP1916A (es)
AR (1) AR041835A1 (es)
AT (1) ATE371658T1 (es)
AU (1) AU2003269368B2 (es)
BR (1) BR0314918A (es)
CA (1) CA2503900C (es)
CO (1) CO5560546A2 (es)
CR (1) CR7812A (es)
CU (1) CU23535A3 (es)
CY (1) CY1107505T1 (es)
DE (1) DE60316012T2 (es)
DK (1) DK1558615T3 (es)
DO (1) DOP2003000742A (es)
EA (1) EA008176B1 (es)
EC (1) ECSP055767A (es)
EG (1) EG24662A (es)
ES (1) ES2291669T3 (es)
GE (1) GEP20084325B (es)
GT (1) GT200300232A (es)
HK (2) HK1081189A1 (es)
HR (1) HRP20050378A2 (es)
IS (1) IS2602B (es)
MA (1) MA27479A1 (es)
MX (1) MXPA05003882A (es)
MY (1) MY140010A (es)
NL (1) NL1024643C2 (es)
NO (1) NO332195B1 (es)
NZ (1) NZ539589A (es)
OA (1) OA13080A (es)
PE (1) PE20040781A1 (es)
PL (1) PL376311A1 (es)
PT (1) PT1558615E (es)
RS (2) RS20050306A (es)
SG (1) SG148071A1 (es)
TN (1) TNSN05121A1 (es)
TW (1) TWI327567B (es)
UA (1) UA79507C2 (es)
UY (1) UY28044A1 (es)
WO (1) WO2004037823A1 (es)
ZA (1) ZA200503378B (es)

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