CR10139A - "combinación de un inhibidor de acetilcolinesterasa y un antagonista de 5-ht6 para el tratamiento de la disfusión congnitiva" - Google Patents
"combinación de un inhibidor de acetilcolinesterasa y un antagonista de 5-ht6 para el tratamiento de la disfusión congnitiva"Info
- Publication number
- CR10139A CR10139A CR10139A CR10139A CR10139A CR 10139 A CR10139 A CR 10139A CR 10139 A CR10139 A CR 10139A CR 10139 A CR10139 A CR 10139A CR 10139 A CR10139 A CR 10139A
- Authority
- CR
- Costa Rica
- Prior art keywords
- treatment
- combination
- antagonist
- inhibitor
- disfusion
- Prior art date
Links
- 229940124801 5-HT6 antagonist Drugs 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 239000003751 serotonin 6 antagonist Substances 0.000 title 1
- 229940100578 Acetylcholinesterase inhibitor Drugs 0.000 abstract 1
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 239000003420 antiserotonin agent Substances 0.000 abstract 1
- 239000000544 cholinesterase inhibitor Substances 0.000 abstract 1
- 208000010877 cognitive disease Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención suministra un método para el tratamiento de un trastorno cognitivo tal como la enfermedad de Alzheimer en un paciente que lo necesita que comprende suministrar a dicho paciente una cantidad terapéuticamente afectiva de una combinación de un inhibidor de acetilcolinesterasa y un antagonista 5-hidroxitriptamina-6.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US75884106P | 2006-01-13 | 2006-01-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR10139A true CR10139A (es) | 2008-09-30 |
Family
ID=38109582
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR10139A CR10139A (es) | 2006-01-13 | 2008-07-11 | "combinación de un inhibidor de acetilcolinesterasa y un antagonista de 5-ht6 para el tratamiento de la disfusión congnitiva" |
Country Status (20)
Country | Link |
---|---|
US (1) | US20070167431A1 (es) |
EP (1) | EP1971334A2 (es) |
JP (1) | JP2009523728A (es) |
KR (1) | KR20080096657A (es) |
CN (1) | CN101370499A (es) |
AR (1) | AR060019A1 (es) |
AU (1) | AU2007208516A1 (es) |
BR (1) | BRPI0706515A2 (es) |
CA (1) | CA2635920A1 (es) |
CR (1) | CR10139A (es) |
EC (1) | ECSP088619A (es) |
GT (1) | GT200800138A (es) |
IL (1) | IL192694A0 (es) |
MX (1) | MX2008009021A (es) |
NO (1) | NO20082894L (es) |
PE (1) | PE20071143A1 (es) |
RU (1) | RU2008126245A (es) |
TW (1) | TW200733976A (es) |
WO (1) | WO2007087151A2 (es) |
ZA (1) | ZA200806070B (es) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005012254A1 (en) | 2003-07-22 | 2005-02-10 | Arena Pharmaceuticals, Inc. | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related therto |
CA2658959A1 (en) * | 2006-06-23 | 2007-12-27 | Laboratorios Del Dr. Esteve, S.A. | Combination of a cholinesterase inhibitor and a compound with 5-ht6 receptor affinity |
AR061637A1 (es) * | 2006-06-26 | 2008-09-10 | Epix Delaware Inc | Composiciones y metodos de tratamiento de trastornos del snc |
EP2508177A1 (en) | 2007-12-12 | 2012-10-10 | Glaxo Group Limited | Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
WO2009123714A2 (en) | 2008-04-02 | 2009-10-08 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
US9126946B2 (en) | 2008-10-28 | 2015-09-08 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto |
RU2467749C1 (ru) * | 2011-04-21 | 2012-11-27 | Государственное образовательное учреждение высшего профессионального образования "Воронежская государственная медицинская академия им. Н.Н. Бурденко" Министерства здравоохранения и социального развития Российской Федерации | Способ коррекции уровня сахара крови и лечения пациентов с сахарным диабетом второго типа с когнитивными нарушениями |
JO3459B1 (ar) | 2012-09-09 | 2020-07-05 | H Lundbeck As | تركيبات صيدلانية لعلاج مرض الزهايمر |
CN111943890B (zh) * | 2014-11-03 | 2023-10-31 | 艾欧米制药有限公司 | 药用化合物 |
WO2016179569A1 (en) * | 2015-05-07 | 2016-11-10 | Axovant Sciences Ltd. | Compositions and methods of treating a neurodegenerative disease |
MX2017016413A (es) | 2015-06-12 | 2018-08-01 | Axovant Sciences Gmbh | Derivados de diaril y arilheteroaril urea como moduladores del receptor 5ht2a de serotonina útiles para la profilaxis y el tratamineto de un trastorno conductual del sueño rem. |
MX2018000465A (es) | 2015-07-15 | 2018-09-17 | Axovant Sciences Gmbh | Derivados de diaril y arilheteroaril urea como moduladores del receptor de serotonina 5-ht2a útiles para la profilaxis y el tratamiento de alucinaciones asociadas con una enfermedad neurodegenerativa. |
WO2017147601A1 (en) * | 2016-02-25 | 2017-08-31 | Axovant Sciences Gmbh | Methods of improving balance, gait or both in patients with neurological disease |
TW201806621A (zh) * | 2016-04-26 | 2018-03-01 | H 朗德貝克公司 | 乙醯膽鹼酯酶抑制劑和艾達魯吡啶用於在帕金森氏病患者中減少跌倒之用途 |
US10864191B2 (en) * | 2016-05-11 | 2020-12-15 | H. Lundbeck A/S | 5-HT6 receptor antagonists for use in the treatment of Alzheimer's disease with apathy as comorbidity |
EP3484467B1 (en) * | 2016-05-18 | 2020-04-29 | Suven Life Sciences Limited | Combination of pure 5-ht6 receptor antagonists with acetylcholinesterase inhibitors |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1222511C (zh) * | 2000-11-02 | 2005-10-12 | 惠氏公司 | 作为5-羟色胺-6配体的1-芳基-或1-烷基磺酰基-杂环基吲哚 |
PL377777A1 (pl) * | 2002-12-11 | 2006-02-20 | Pharmacia & Upjohn Company Llc | Leczenie chorób połączeniami agonistów receptora alfa 7-nikotynowego i innych związków |
AU2004213374A1 (en) * | 2003-02-14 | 2004-09-02 | Wyeth | Heterocyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands |
CA2619010C (en) * | 2005-08-15 | 2013-10-01 | Wyeth | Substituted-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands |
-
2006
- 2006-12-28 PE PE2006001716A patent/PE20071143A1/es not_active Application Discontinuation
-
2007
- 2007-01-05 TW TW096100409A patent/TW200733976A/zh unknown
- 2007-01-09 EP EP07716405A patent/EP1971334A2/en not_active Withdrawn
- 2007-01-09 WO PCT/US2007/000354 patent/WO2007087151A2/en active Application Filing
- 2007-01-09 BR BRPI0706515-9A patent/BRPI0706515A2/pt not_active IP Right Cessation
- 2007-01-09 JP JP2008550355A patent/JP2009523728A/ja not_active Withdrawn
- 2007-01-09 AU AU2007208516A patent/AU2007208516A1/en not_active Abandoned
- 2007-01-09 CN CNA200780003019XA patent/CN101370499A/zh active Pending
- 2007-01-09 MX MX2008009021A patent/MX2008009021A/es not_active Application Discontinuation
- 2007-01-09 CA CA002635920A patent/CA2635920A1/en not_active Abandoned
- 2007-01-09 RU RU2008126245/14A patent/RU2008126245A/ru not_active Application Discontinuation
- 2007-01-09 KR KR1020087019279A patent/KR20080096657A/ko not_active Application Discontinuation
- 2007-01-12 AR ARP070100160A patent/AR060019A1/es unknown
- 2007-01-12 US US11/652,725 patent/US20070167431A1/en not_active Abandoned
-
2008
- 2008-06-30 NO NO20082894A patent/NO20082894L/no not_active Application Discontinuation
- 2008-07-08 IL IL192694A patent/IL192694A0/en unknown
- 2008-07-10 GT GT200800138A patent/GT200800138A/es unknown
- 2008-07-11 ZA ZA200806070A patent/ZA200806070B/xx unknown
- 2008-07-11 CR CR10139A patent/CR10139A/es not_active Application Discontinuation
- 2008-07-11 EC EC2008008619A patent/ECSP088619A/es unknown
Also Published As
Publication number | Publication date |
---|---|
AR060019A1 (es) | 2008-05-21 |
TW200733976A (en) | 2007-09-16 |
PE20071143A1 (es) | 2008-01-20 |
EP1971334A2 (en) | 2008-09-24 |
ECSP088619A (es) | 2008-08-29 |
IL192694A0 (en) | 2009-02-11 |
KR20080096657A (ko) | 2008-10-31 |
AU2007208516A8 (en) | 2008-08-07 |
RU2008126245A (ru) | 2010-02-20 |
MX2008009021A (es) | 2008-09-24 |
US20070167431A1 (en) | 2007-07-19 |
CA2635920A1 (en) | 2007-08-02 |
AU2007208516A1 (en) | 2007-08-02 |
CN101370499A (zh) | 2009-02-18 |
NO20082894L (no) | 2008-09-30 |
WO2007087151A2 (en) | 2007-08-02 |
BRPI0706515A2 (pt) | 2011-03-29 |
WO2007087151A3 (en) | 2007-11-15 |
ZA200806070B (en) | 2009-04-29 |
GT200800138A (es) | 2008-10-06 |
JP2009523728A (ja) | 2009-06-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal (granting procedure) |