CN1839131A - 吡咯烷甲腈类化合物及其作为dpp－iv抑制剂的应用 - Google Patents

吡咯烷甲腈类化合物及其作为dpp－iv抑制剂的应用 Download PDF

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Publication number
CN1839131A
CN1839131A CNA2003801104652A CN200380110465A CN1839131A CN 1839131 A CN1839131 A CN 1839131A CN A2003801104652 A CNA2003801104652 A CN A2003801104652A CN 200380110465 A CN200380110465 A CN 200380110465A CN 1839131 A CN1839131 A CN 1839131A
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ethyl
oxo
piperidin
diazanyl
cyano
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Chinese (zh)
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A·杉卡拉那拉亚南
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Torrent Pharmaceuticals Ltd
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Torrent Pharmaceuticals Ltd
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
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  • Health & Medical Sciences (AREA)
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  • General Chemical & Material Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pulmonology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Psychiatry (AREA)
CNA2003801104652A 2003-10-06 2003-10-06 吡咯烷甲腈类化合物及其作为dpp－iv抑制剂的应用 Pending CN1839131A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/IB2003/004377 WO2005033106A1 (en) 2003-10-06 2003-10-06 Azolidinecarbonitriles and their use as dpp-iv inhibitors

Publications (1)

Publication Number Publication Date
CN1839131A true CN1839131A (zh) 2006-09-27

Family

ID=34401253

Family Applications (1)

Application Number Title Priority Date Filing Date
CNA2003801104652A Pending CN1839131A (zh) 2003-10-06 2003-10-06 吡咯烷甲腈类化合物及其作为dpp－iv抑制剂的应用

Country Status (8)

Country Link
EP (1) EP1682540A1 (de)
JP (1) JP2007516154A (de)
CN (1) CN1839131A (de)
AU (1) AU2003269307A1 (de)
BR (1) BR0318533A (de)
CA (1) CA2534634A1 (de)
PL (1) PL380189A3 (de)
WO (1) WO2005033106A1 (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008055945A1 (en) 2006-11-09 2008-05-15 Probiodrug Ag 3-hydr0xy-1,5-dihydr0-pyrr0l-2-one derivatives as inhibitors of glutaminyl cyclase for the treatment of ulcer, cancer and other diseases
SI2091948T1 (sl) 2006-11-30 2012-07-31 Probiodrug Ag Novi inhibitorji glutaminil ciklaze
EP2142514B1 (de) 2007-04-18 2014-12-24 Probiodrug AG Thioharnstoffderivate als glutaminylcyclaseinhibitoren
ES2548913T3 (es) 2009-09-11 2015-10-21 Probiodrug Ag Derivados heterocíclicos como inhibidores de glutaminil ciclasa
JP6026284B2 (ja) 2010-03-03 2016-11-16 プロビオドルグ エージー グルタミニルシクラーゼの阻害剤
JP5688745B2 (ja) 2010-03-10 2015-03-25 プロビオドルグ エージー グルタミニルシクラーゼ（ｑｃ、ｅｃ２．３．２．５）の複素環阻害剤
WO2011131748A2 (en) 2010-04-21 2011-10-27 Probiodrug Ag Novel inhibitors
WO2012123563A1 (en) 2011-03-16 2012-09-20 Probiodrug Ag Benz imidazole derivatives as inhibitors of glutaminyl cyclase
WO2012170702A1 (en) 2011-06-08 2012-12-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
EP3461819B1 (de) 2017-09-29 2020-05-27 Probiodrug AG Hemmer der glutaminylcyclase

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL111785A0 (en) * 1993-12-03 1995-01-24 Ferring Bv Dp-iv inhibitors and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
BR0318533A (pt) 2006-09-12
JP2007516154A (ja) 2007-06-21
AU2003269307A1 (en) 2005-04-21
WO2005033106A1 (en) 2005-04-14
PL380189A3 (pl) 2007-01-08
CA2534634A1 (en) 2005-04-14
EP1682540A1 (de) 2006-07-26

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