CN101679210B - 旋光性α氨基乙缩醛外消旋化的方法 - Google Patents
旋光性α氨基乙缩醛外消旋化的方法 Download PDFInfo
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- CN101679210B CN101679210B CN2008800166936A CN200880016693A CN101679210B CN 101679210 B CN101679210 B CN 101679210B CN 2008800166936 A CN2008800166936 A CN 2008800166936A CN 200880016693 A CN200880016693 A CN 200880016693A CN 101679210 B CN101679210 B CN 101679210B
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/04—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C217/28—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines
- C07C217/40—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having one amino group and at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the carbon skeleton, e.g. ethers of polyhydroxy amines having at least two singly-bound oxygen atoms, with at least one being part of an etherified hydroxy group, bound to the same carbon atom of the carbon skeleton, e.g. amino-ketals, ortho esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/02—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C217/48—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C249/04—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/582—Recycling of unreacted starting or intermediate materials
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Description
Claims (16)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0755190A FR2916441B1 (fr) | 2007-05-22 | 2007-05-22 | Procede de racemisation d'alpha-aminoacetals optiquement actifs. |
FR0755190 | 2007-05-22 | ||
PCT/EP2008/056219 WO2008142088A1 (en) | 2007-05-22 | 2008-05-21 | Process of racemisation of optically active alpha aminoacetals |
Publications (2)
Publication Number | Publication Date |
---|---|
CN101679210A CN101679210A (zh) | 2010-03-24 |
CN101679210B true CN101679210B (zh) | 2013-08-14 |
Family
ID=38925562
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN2008800166936A Expired - Fee Related CN101679210B (zh) | 2007-05-22 | 2008-05-21 | 旋光性α氨基乙缩醛外消旋化的方法 |
Country Status (10)
Country | Link |
---|---|
US (1) | US8350092B2 (zh) |
EP (1) | EP2162426B1 (zh) |
JP (1) | JP5529726B2 (zh) |
CN (1) | CN101679210B (zh) |
CA (1) | CA2687823C (zh) |
DK (1) | DK2162426T3 (zh) |
ES (1) | ES2402174T3 (zh) |
FR (1) | FR2916441B1 (zh) |
RU (1) | RU2470912C2 (zh) |
WO (1) | WO2008142088A1 (zh) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20100016464A (ko) * | 2007-04-12 | 2010-02-12 | 다우 글로벌 테크놀로지스 인크. | 다중하이드록실화된-지방족 탄화수소 또는 이의 에스터의 클로로하이드린으로의 전환 |
FR2927900B1 (fr) * | 2008-02-27 | 2010-09-17 | Clariant Specialty Fine Chem | Procede de preparation d'alpha-aminoacetals optiquement actifs. |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4769486A (en) * | 1986-08-26 | 1988-09-06 | Toyo Soda Manufacturing Co., Ltd. | Method for racemizing an optically active amino acid |
EP0779261A1 (en) * | 1995-12-13 | 1997-06-18 | Uop | Continuous process for racemization of benzylic alcohols, ethers, and esters by solid acid catalyst |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE388849B (sv) * | 1974-02-14 | 1976-10-18 | Haessle Ab | Forfarande for framstellning av nya aminer med beta-receptorstimulerande verkan |
JPS59170058A (ja) | 1983-03-16 | 1984-09-26 | Tanabe Seiyaku Co Ltd | アミノ酸の光学分割方法 |
DE3782191T2 (de) | 1986-06-05 | 1993-02-25 | Ici America Inc | Difluorketoverbindungen. |
GB8809316D0 (en) | 1987-05-11 | 1988-05-25 | Ici America Inc | Heterocyclic ketones |
IL91997A0 (en) | 1988-11-03 | 1990-07-12 | American Cyanamid Co | Aryloxy benzotriazole herbicidal agents and methods for the preparation thereof |
DE3843390A1 (de) * | 1988-12-23 | 1990-07-05 | Basf Ag | Verfahren zur herstellung von optisch aktiven (alpha)-aminoacetalen |
US5614649A (en) | 1994-11-14 | 1997-03-25 | Cephalon, Inc. | Multicatalytic protease inhibitors |
US5476964A (en) * | 1994-11-21 | 1995-12-19 | Uop | Continuous racemization of benzylic alcohols, ethers, and esters by solid acid catalyst |
DE19505992C2 (de) * | 1995-02-21 | 1997-04-10 | Degussa | Verfahren zur Herstellung von racemischen Aminoalkoholen |
DE19643126A1 (de) * | 1996-10-18 | 1998-04-23 | Basf Ag | Metall-Festbettkatalysator nach Raney, Verfahren zu seiner Herstellung sowie ein Verfahren zur Hydrierung von Polymeren unter Verwendung dieses Katalysators |
GB9623908D0 (en) | 1996-11-18 | 1997-01-08 | Hoffmann La Roche | Amino acid derivatives |
HU226421B1 (en) * | 1998-11-09 | 2008-12-29 | Sanofi Aventis | Process for racemizing optically active 2-(2-chlorophenyl)-2-(2-(2-thienyl)-ethylamino)-acetamides |
JP4296783B2 (ja) * | 2002-01-15 | 2009-07-15 | 住友化学株式会社 | ニトロ化合物の製造方法とその触媒 |
FR2843112B1 (fr) | 2002-07-30 | 2004-10-22 | Clariant | Procede de preparation d'amines primaires. |
JP4461891B2 (ja) * | 2003-06-02 | 2010-05-12 | 住友化学株式会社 | ラセミアミンの製造方法 |
FR2927900B1 (fr) | 2008-02-27 | 2010-09-17 | Clariant Specialty Fine Chem | Procede de preparation d'alpha-aminoacetals optiquement actifs. |
-
2007
- 2007-05-22 FR FR0755190A patent/FR2916441B1/fr not_active Expired - Fee Related
-
2008
- 2008-05-21 US US12/601,067 patent/US8350092B2/en active Active
- 2008-05-21 ES ES08759824T patent/ES2402174T3/es active Active
- 2008-05-21 DK DK08759824.9T patent/DK2162426T3/da active
- 2008-05-21 EP EP08759824A patent/EP2162426B1/en not_active Not-in-force
- 2008-05-21 CN CN2008800166936A patent/CN101679210B/zh not_active Expired - Fee Related
- 2008-05-21 CA CA 2687823 patent/CA2687823C/en not_active Expired - Fee Related
- 2008-05-21 WO PCT/EP2008/056219 patent/WO2008142088A1/en active Application Filing
- 2008-05-21 JP JP2010508831A patent/JP5529726B2/ja not_active Expired - Fee Related
- 2008-05-21 RU RU2009142986/04A patent/RU2470912C2/ru not_active IP Right Cessation
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4769486A (en) * | 1986-08-26 | 1988-09-06 | Toyo Soda Manufacturing Co., Ltd. | Method for racemizing an optically active amino acid |
EP0779261A1 (en) * | 1995-12-13 | 1997-06-18 | Uop | Continuous process for racemization of benzylic alcohols, ethers, and esters by solid acid catalyst |
Non-Patent Citations (1)
Title |
---|
Fanny Guillaumie et al.,.Solid-phase synthesis of C-terminal peptide aldehydes from aminoacetals anchored to a backbone amide linker(BAL) handle.《Tetrahedron Letters》.2000,第41卷(第32期),6131-6135. * |
Also Published As
Publication number | Publication date |
---|---|
DK2162426T3 (da) | 2013-04-08 |
CA2687823C (en) | 2015-03-31 |
RU2470912C2 (ru) | 2012-12-27 |
EP2162426A1 (en) | 2010-03-17 |
JP5529726B2 (ja) | 2014-06-25 |
ES2402174T3 (es) | 2013-04-29 |
RU2009142986A (ru) | 2011-06-27 |
EP2162426B1 (en) | 2013-01-02 |
JP2010527959A (ja) | 2010-08-19 |
FR2916441B1 (fr) | 2009-08-28 |
FR2916441A1 (fr) | 2008-11-28 |
CA2687823A1 (en) | 2008-11-27 |
CN101679210A (zh) | 2010-03-24 |
WO2008142088A1 (en) | 2008-11-27 |
US20100152490A1 (en) | 2010-06-17 |
US8350092B2 (en) | 2013-01-08 |
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C14 | Grant of patent or utility model | ||
GR01 | Patent grant | ||
C56 | Change in the name or address of the patentee | ||
CP02 | Change in the address of a patent holder |
Address after: French Te Rosli Buller I Patentee after: Clariant Specialty Fine Chemicals (France) Address before: French pitot Patentee before: Clariant Specialty Fine Chemicals (France) Address after: French Te Rosli Buller I Patentee after: Clariant Specialty Fine Chemicals (France) Address before: French pitot Patentee before: Clariant Specialty Fine Chemicals (France) |
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C56 | Change in the name or address of the patentee |
Owner name: CLARIANT CHEMICAL LAMOTTE SIMPLIFIED CORPORATION Free format text: FORMER NAME: CLARIANT SPECIALTY FINE CHEMIC |
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CP03 | Change of name, title or address |
Address after: Union of France Patentee after: Simple chemical Co. Ltd. for Maxwell Address before: French Te Rosli Buller I Patentee before: Clariant Specialty Fine Chemicals (France) Address after: Union of France Patentee after: Simple chemical Co. Ltd. for Maxwell Address before: French Te Rosli Buller I Patentee before: Clariant Specialty Fine Chemicals (France) |
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CF01 | Termination of patent right due to non-payment of annual fee | ||
CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20130814 Termination date: 20190521 |