CH629500A5 - Processes for preparing novel cephalosporins. - Google Patents

Processes for preparing novel cephalosporins. Download PDF

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Publication number
CH629500A5
CH629500A5 CH1259376A CH1259376A CH629500A5 CH 629500 A5 CH629500 A5 CH 629500A5 CH 1259376 A CH1259376 A CH 1259376A CH 1259376 A CH1259376 A CH 1259376A CH 629500 A5 CH629500 A5 CH 629500A5
Authority
CH
Switzerland
Prior art keywords
sodium
formula
potassium
acid
solution
Prior art date
Application number
CH1259376A
Other languages
German (de)
English (en)
Inventor
Murray Arthur Kaplan
William J Gottstein
Alphonse Peter Granatek
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/653,999 external-priority patent/US4026888A/en
Priority claimed from US05/654,314 external-priority patent/US4061862A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH629500A5 publication Critical patent/CH629500A5/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/58Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with a nitrogen atom, which is a member of a hetero ring, attached in position 7

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH1259376A 1975-10-06 1976-10-05 Processes for preparing novel cephalosporins. CH629500A5 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US62000575A 1975-10-06 1975-10-06
US62230675A 1975-10-10 1975-10-10
US64031775A 1975-12-12 1975-12-12
US05/653,999 US4026888A (en) 1975-10-10 1976-01-30 Certain derivatives of particular 3-thiolated cephalosporins
US05/654,314 US4061862A (en) 1975-10-06 1976-02-02 Derivatives of 7-(cyclized)phenylglycyl-3-triazolo-thio methyl cephalosporin

Publications (1)

Publication Number Publication Date
CH629500A5 true CH629500A5 (en) 1982-04-30

Family

ID=27542000

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1259376A CH629500A5 (en) 1975-10-06 1976-10-05 Processes for preparing novel cephalosporins.

Country Status (17)

Country Link
JP (1) JPS6052718B2 (da)
AU (1) AU511344B2 (da)
BE (1) BE846890A (da)
CA (1) CA1113927A (da)
CH (1) CH629500A5 (da)
CY (1) CY1121A (da)
DE (1) DE2645144C2 (da)
DK (2) DK158673C (da)
FR (1) FR2326926A1 (da)
GB (1) GB1521419A (da)
HK (1) HK41281A (da)
IE (1) IE43666B1 (da)
KE (1) KE3154A (da)
LU (1) LU75935A1 (da)
NL (1) NL189670C (da)
SE (1) SE434952B (da)
YU (1) YU40287B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54112892A (en) * 1978-02-23 1979-09-04 Shionogi & Co Ltd Substituted imidazolidinyl-3-chloro-3-cephem-4-carboxylic acid
JPS54115354A (en) * 1978-02-27 1979-09-07 Chugai Pharmaceut Co Ltd Biphenylylglycine derivative
JP7013048B2 (ja) * 2018-03-02 2022-01-31 国立大学法人大阪大学 タンパク質及び/又はペプチド修飾用分子

Also Published As

Publication number Publication date
FR2326926A1 (fr) 1977-05-06
YU40287B (en) 1985-12-31
CA1113927A (en) 1981-12-08
KE3154A (en) 1981-09-18
IE43666B1 (en) 1981-04-22
DE2645144C2 (de) 1986-11-27
GB1521419A (en) 1978-08-16
BE846890A (fr) 1977-04-01
DE2645144A1 (de) 1977-04-14
AU511344B2 (en) 1980-08-14
DK158673C (da) 1991-01-14
DK200488A (da) 1988-04-12
SE434952B (sv) 1984-08-27
DK158673B (da) 1990-07-02
NL189670C (nl) 1993-06-16
JPS6052718B2 (ja) 1985-11-20
DK164225C (da) 1992-10-19
FR2326926B1 (da) 1980-07-11
DK446576A (da) 1977-04-07
NL189670B (nl) 1993-01-18
HK41281A (en) 1981-08-28
IE43666L (en) 1977-04-06
DK200488D0 (da) 1988-04-12
JPS5246094A (en) 1977-04-12
SE7610989L (sv) 1977-04-07
YU243176A (en) 1982-06-30
DK164225B (da) 1992-05-25
LU75935A1 (da) 1977-05-25
NL7611026A (nl) 1977-04-12
CY1121A (en) 1981-12-04
AU1824576A (en) 1978-04-06

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PL Patent ceased