CA2291665A1 - Process for preparing 3-(7-amidino-2-naphthyl)-2-phenylpropionic acid derivatives - Google Patents

Process for preparing 3-(7-amidino-2-naphthyl)-2-phenylpropionic acid derivatives Download PDF

Info

Publication number
CA2291665A1
CA2291665A1 CA002291665A CA2291665A CA2291665A1 CA 2291665 A1 CA2291665 A1 CA 2291665A1 CA 002291665 A CA002291665 A CA 002291665A CA 2291665 A CA2291665 A CA 2291665A CA 2291665 A1 CA2291665 A1 CA 2291665A1
Authority
CA
Canada
Prior art keywords
group
salt
alkyl
pyrrolidinyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002291665A
Other languages
English (en)
French (fr)
Inventor
Toru Makino
Yukio Yokoyama
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Pharmaceutical Co Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2291665A1 publication Critical patent/CA2291665A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/12—Oxygen or sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
CA002291665A 1997-05-30 1998-05-29 Process for preparing 3-(7-amidino-2-naphthyl)-2-phenylpropionic acid derivatives Abandoned CA2291665A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP14204297 1997-05-30
JP9-142042 1997-05-30
PCT/JP1998/002379 WO1998054132A1 (fr) 1997-05-30 1998-05-29 Procede de preparation de derives d'acide 3-(7-amidino-2-naphthyl)-2-phenylpropionique

Publications (1)

Publication Number Publication Date
CA2291665A1 true CA2291665A1 (en) 1998-12-03

Family

ID=15306044

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002291665A Abandoned CA2291665A1 (en) 1997-05-30 1998-05-29 Process for preparing 3-(7-amidino-2-naphthyl)-2-phenylpropionic acid derivatives

Country Status (14)

Country Link
US (1) US6342609B2 (de)
EP (1) EP0990646B1 (de)
JP (1) JP3241741B2 (de)
KR (1) KR100527833B1 (de)
CN (1) CN1181053C (de)
AU (1) AU7454998A (de)
CA (1) CA2291665A1 (de)
DE (1) DE69823506T2 (de)
ES (1) ES2221984T3 (de)
HK (1) HK1027109A1 (de)
NO (1) NO313876B1 (de)
PT (1) PT990646E (de)
TW (1) TW513402B (de)
WO (1) WO1998054132A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6949567B2 (en) 2001-02-26 2005-09-27 4Sc Ag Compounds for the treatment of protozoal diseases
CH695999A5 (de) 2002-02-28 2006-11-15 Wilex Ag Verfahren zur Herstellung von 3- Amidinophenylalanin-Derivaten.
CN100513398C (zh) 2002-12-03 2009-07-15 Axys药物公司 作为因子viia抑制剂的2-(2-羟基联苯-3-基)-1h-苯并咪唑-5-甲脒衍生物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA928276B (en) * 1991-10-31 1993-05-06 Daiichi Seiyaku Co Aromatic amidine derivates and salts thereof.
JP3457694B2 (ja) * 1993-02-04 2003-10-20 第一製薬株式会社 インフルエンザ感染予防・治療薬
DE4424713A1 (de) * 1994-07-13 1996-01-18 Boehringer Ingelheim Kg Substituierte Benzamidine, ihre Herstellung und Verwendung als Arnzneistoffe

Also Published As

Publication number Publication date
EP0990646B1 (de) 2004-04-28
NO995841D0 (no) 1999-11-29
NO995841L (no) 2000-01-20
WO1998054132A1 (fr) 1998-12-03
ES2221984T3 (es) 2005-01-16
NO313876B1 (no) 2002-12-16
TW513402B (en) 2002-12-11
CN1181053C (zh) 2004-12-22
JP3241741B2 (ja) 2001-12-25
DE69823506D1 (de) 2004-06-03
US20010001802A1 (en) 2001-05-24
CN1258275A (zh) 2000-06-28
US6342609B2 (en) 2002-01-29
DE69823506T2 (de) 2004-09-23
EP0990646A4 (de) 2001-01-17
PT990646E (pt) 2004-09-30
KR20010012780A (ko) 2001-02-26
KR100527833B1 (ko) 2005-11-09
EP0990646A1 (de) 2000-04-05
AU7454998A (en) 1998-12-30
HK1027109A1 (en) 2001-01-05

Similar Documents

Publication Publication Date Title
US20050107614A1 (en) Process for the preparation of repaglinide
US5977381A (en) Process for making 3-amino-pyrolidine derivatives
EP0990646B1 (de) Verfahren zur herstellung von 3-(7-amidino-2-naphthyl)-2-phenylpropionsäure-derivaten
US5179212A (en) Process for the preparation of 3-pyrrolidinols and intermediates therefor
JP4688292B2 (ja) 純粋な鏡像体であるｎ−メチル−ｎ−［（１ｓ）−１−フェニル−２−（（３ｓ）−３−ヒドロキシピロリジン−１−イル）エチル］−２，２−ジフェニルアセトアミドの製造方法
JP3266603B2 (ja) ３−（７−アミジノ−２−ナフチル）−２−フェニルプロピオン酸誘導体の製造方法
JP3266603B6 (ja) ３−（７−アミジノ−２−ナフチル）−２−フェニルプロピオン酸誘導体の製造方法
US5981794A (en) γ-oxo-homophenylalanine derivatives and process for producing homophenylalanine derivatives by reducing the same
US10723691B2 (en) Process for preparing salicyloyl-L-carnitine hydrochloride
EP0844242B1 (de) Verfahren zur Herstellung von 4-Hydroxy-2-Pyrrolidinon und Verfahren zu deren Reinigung
US5929242A (en) Manufacture of levobupivacaine and analogues thereof from L-lysine
WO2000029369A1 (fr) Derives d'acide aminoacrylique et procede de production correspondant
US6252089B1 (en) Method of producing 4-hydroxy-2-pyrrolidinone and method of purifying the same
AU5479700A (en) Process for preparing (-)-(1s,4r) n-protected 4-amino-2-cyclopentene-1-carboxylate esters
JP2000044539A (ja) 光学活性環式アミノ酸エステル誘導体およびその製造方法
JP2005306782A (ja) Ｌ−カルノシンの新規合成方法
JP2001031647A (ja) ４−ヒドロキシ−２−ピロリジノンの精製方法
JP2001328993A (ja) 光学活性ホスフィン化合物
JPS63183548A (ja) Ｎ−ヒドロキシアミノ酸類の製造法
WO1994002487A1 (en) Novel pyridonecarboxylic acid derivatives and processes for preparing the same
JPH0331287A (ja) セファロスポリン化合物の合成法
WO2002008184A1 (en) Process for preparing distamycin derivatives

Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued