BRPI0716240B8 - composto de n-piridilpiperidina, método para a sua produção, e agente de controle de pestes - Google Patents

composto de n-piridilpiperidina, método para a sua produção, e agente de controle de pestes Download PDF

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Publication number
BRPI0716240B8
BRPI0716240B8 BRPI0716240A BRPI0716240A BRPI0716240B8 BR PI0716240 B8 BRPI0716240 B8 BR PI0716240B8 BR PI0716240 A BRPI0716240 A BR PI0716240A BR PI0716240 A BRPI0716240 A BR PI0716240A BR PI0716240 B8 BRPI0716240 B8 BR PI0716240B8
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BR
Brazil
Prior art keywords
pyridylpiperidine compound
production
control agent
pest control
group
Prior art date
Application number
BRPI0716240A
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English (en)
Inventor
Uenaka Go
Endo Yasuhiro
Shirai Yuichi
Original Assignee
Oat Agrio Co Ltd
Otsuka Agritechno Co Ltd
Otsuka Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oat Agrio Co Ltd, Otsuka Agritechno Co Ltd, Otsuka Chemical Co Ltd filed Critical Oat Agrio Co Ltd
Publication of BRPI0716240A2 publication Critical patent/BRPI0716240A2/pt
Publication of BRPI0716240B1 publication Critical patent/BRPI0716240B1/pt
Publication of BRPI0716240B8 publication Critical patent/BRPI0716240B8/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms

Abstract

composto de n-piridilpiperidina, método para a sua produção, e agente de controle de pestes. a presente invenção refere-se a um composto de n- piridilpiperidina da invenção é representado pela fórmula (1), em que r¹ é um átomo de halogêneo, um grupo de c1-4 haloalquila, um grupo de ciano, um grupo de nitro, ou grupo de c1-4 alcoxicarbonila; r², r³ r4, r5, r6, r7, r8, e r9 são cada um independentemente um átomo de hidrogênio ou um grupo de c1- alquila; r¹° é um átomo de hidrogênio, etc.; r¹¹ é um átomo de halogêneo, etc.; x é um átomo de oxigênio ou um átomo de enxofre, m é um número inteiro de 1 a 4; e n é um número inteiro de 1 ou 2. o composo de n-piridilpiperidina da invenção possui uma excelente atividade miticida contra ácaros aranha e ácaros da ferrugem.
BRPI0716240A 2006-09-01 2007-08-29 composto de n-piridilpiperidina, método para a sua produção, e agente de controle de pestes BRPI0716240B8 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2006-237557 2006-09-01
JP2006237557 2006-09-01
JP2007-100825 2007-04-06
JP2007100825 2007-04-06
PCT/JP2007/066807 WO2008026658A1 (ja) 2006-09-01 2007-08-29 Ｎ－ピリジルピペリジン化合物、その製造方法及び有害生物防除剤

Publications (3)

Publication Number Publication Date
BRPI0716240A2 BRPI0716240A2 (pt) 2013-08-13
BRPI0716240B1 BRPI0716240B1 (pt) 2016-05-10
BRPI0716240B8 true BRPI0716240B8 (pt) 2019-09-17

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0716240A BRPI0716240B8 (pt) 2006-09-01 2007-08-29 composto de n-piridilpiperidina, método para a sua produção, e agente de controle de pestes

Country Status (13)

Country Link
US (1) US7994094B2 (pt)
EP (1) EP2050745B1 (pt)
JP (1) JP5121717B2 (pt)
KR (1) KR101428681B1 (pt)
CN (1) CN101511818B (pt)
AT (1) ATE550334T1 (pt)
AU (1) AU2007289681B2 (pt)
BR (1) BRPI0716240B8 (pt)
CA (1) CA2661741C (pt)
ES (1) ES2382481T3 (pt)
HK (1) HK1137744A1 (pt)
TW (1) TWI401027B (pt)
WO (1) WO2008026658A1 (pt)

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NZ622505A (en) 2009-06-29 2015-12-24 Agios Pharmaceuticals Inc Therapeutic compounds and compositions
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KR101280160B1 (ko) 2009-09-02 2013-06-28 이화여자대학교 산학협력단 피라졸 유도체, 이의 제조방법 및 이를 포함하는 골다공증 예방 및 치료용 조성물
AR079493A1 (es) 2009-12-21 2012-02-01 Nippon Soda Co Compuesto de amina ciclica y acaricida
AR081721A1 (es) 2010-02-25 2012-10-17 Nippon Soda Co Compuesto de amina ciclica y acaricida
JP5837091B2 (ja) 2010-12-17 2015-12-24 アジオス ファーマシューティカルズ， インコーポレイテッド ピルビン酸キナーゼｍ２（ｐｋｍ２）調節剤としての新規ｎ−（４−（アゼチジン−１−カルボニル）フェニル）−（ヘテロ−）アリールスルホンアミド誘導体
JP6092118B2 (ja) 2010-12-21 2017-03-08 アジオス ファーマシューティカルズ， インコーポレイテッド ニ環式ｐｋｍ２活性化剤
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KR101633957B1 (ko) * 2012-08-27 2016-06-27 이화여자대학교 산학협력단 피라졸 유도체를 포함하는 신장질환 예방 또는 치료용 조성물
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Also Published As

Publication number Publication date
TW200826844A (en) 2008-07-01
TWI401027B (zh) 2013-07-11
WO2008026658A8 (ja) 2008-10-30
AU2007289681B2 (en) 2012-10-04
JPWO2008026658A1 (ja) 2010-01-21
CN101511818B (zh) 2013-05-08
CA2661741A1 (en) 2008-03-06
WO2008026658A1 (ja) 2008-03-06
EP2050745B1 (en) 2012-03-21
CN101511818A (zh) 2009-08-19
EP2050745A4 (en) 2011-04-27
CA2661741C (en) 2014-04-29
US7994094B2 (en) 2011-08-09
ATE550334T1 (de) 2012-04-15
US20100137582A1 (en) 2010-06-03
EP2050745A1 (en) 2009-04-22
BRPI0716240A2 (pt) 2013-08-13
ES2382481T9 (es) 2012-07-20
JP5121717B2 (ja) 2013-01-16
AU2007289681A1 (en) 2008-03-06
HK1137744A1 (en) 2010-08-06
BRPI0716240B1 (pt) 2016-05-10
ES2382481T3 (es) 2012-06-08
KR20090043563A (ko) 2009-05-06
KR101428681B1 (ko) 2014-08-11

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Owner name: OTSUKA AGRITECHNO CO., LTD. (JP)

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
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Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 29/08/2007, OBSERVADAS AS CONDICOES LEGAIS.

B25D Requested change of name of applicant approved
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Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 29/08/2007, OBSERVADAS AS CONDICOES LEGAIS. (CO) REFERENTE A RPI 2366 DE 10/05/2016, QUANTO AO ITEM (72) NOME DO INVENTOR.