BRPI0516754A - usos e derivados de benzoxazina e quinoxalina - Google Patents
usos e derivados de benzoxazina e quinoxalinaInfo
- Publication number
- BRPI0516754A BRPI0516754A BRPI0516754-0A BRPI0516754A BRPI0516754A BR PI0516754 A BRPI0516754 A BR PI0516754A BR PI0516754 A BRPI0516754 A BR PI0516754A BR PI0516754 A BRPI0516754 A BR PI0516754A
- Authority
- BR
- Brazil
- Prior art keywords
- benzoxazine
- quinoxaline
- derivatives
- preparation
- medicament
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Abstract
USOS E DERIVADOS DE BENZOXAZINA E QUINOXALINA. Compostos da fórmula 1: ou um sal farmaceuticamente aceitável, destes, em que k, m, n, p, q, X, Y, Z, Ar, R¹, R², R³ e R¬ 4¬ são como definidos aqui bem como métodos para a preparação destes, composições farmacêuticas contendo-os e o uso destes para a preparação de um medicamento.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US61470504P | 2004-09-30 | 2004-09-30 | |
US63060804P | 2004-11-24 | 2004-11-24 | |
PCT/EP2005/010238 WO2006037481A1 (en) | 2004-09-30 | 2005-09-22 | Benzoxazine and quinoxaline derivatives and uses |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0516754A true BRPI0516754A (pt) | 2008-09-16 |
Family
ID=35385358
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0516754-0A BRPI0516754A (pt) | 2004-09-30 | 2005-09-22 | usos e derivados de benzoxazina e quinoxalina |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP1797051B1 (pt) |
JP (1) | JP2008514662A (pt) |
KR (1) | KR100875041B1 (pt) |
AR (1) | AR051115A1 (pt) |
AT (1) | ATE477248T1 (pt) |
AU (1) | AU2005291541B2 (pt) |
BR (1) | BRPI0516754A (pt) |
CA (1) | CA2581921A1 (pt) |
DE (1) | DE602005022896D1 (pt) |
IL (1) | IL182304A0 (pt) |
MX (1) | MX2007003911A (pt) |
MY (1) | MY139409A (pt) |
NO (1) | NO20071616L (pt) |
NZ (1) | NZ553848A (pt) |
RU (1) | RU2382036C2 (pt) |
TW (1) | TW200626567A (pt) |
WO (1) | WO2006037481A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE602005026543D1 (de) * | 2004-09-30 | 2011-04-07 | Hoffmann La Roche | Zusammensetzungen und verfahren zur behandlung kognitiver störungen |
CL2007003044A1 (es) * | 2006-10-24 | 2008-07-04 | Wyeth Corp | Compuestos derivados de benzoxazina; composicion farmaceutica que los comprende; y uso para el tratamiento de un trastorno psicotico, bipolar, depresivo y abuso o dependencia de sustancias entre otros. |
BRPI0920520A2 (pt) * | 2008-09-08 | 2015-12-22 | Hoffmann La Roche | benzoxazinas 5-subistituídas |
AU2015286049B2 (en) * | 2014-07-08 | 2018-03-01 | Sunshine Lake Pharma Co., Ltd. | Aromatic heterocyclic derivatives and pharmaceutical applications thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW224941B (pt) * | 1989-11-08 | 1994-06-11 | Yamanouchi Pharma Co Ltd | |
NZ512765A (en) * | 1998-12-17 | 2003-10-31 | Wyeth Corp | 2,3,4,4A-tetrahydro-1H-pyrazino(1,2-A)quinoxalin- 5(6H)one derivatives being 5HT2C agonists |
CN1561338A (zh) * | 2001-10-04 | 2005-01-05 | 惠氏公司 | 作为5-羟基色胺-6配体的苯并二氢吡喃衍生物 |
CN100429206C (zh) * | 2002-05-13 | 2008-10-29 | 弗·哈夫曼-拉罗切有限公司 | 作为5-ht6调节剂的苯并嗪衍生物及其用途 |
DE602005026543D1 (de) * | 2004-09-30 | 2011-04-07 | Hoffmann La Roche | Zusammensetzungen und verfahren zur behandlung kognitiver störungen |
-
2005
- 2005-09-22 CA CA002581921A patent/CA2581921A1/en not_active Abandoned
- 2005-09-22 WO PCT/EP2005/010238 patent/WO2006037481A1/en active Application Filing
- 2005-09-22 EP EP05796666A patent/EP1797051B1/en active Active
- 2005-09-22 DE DE602005022896T patent/DE602005022896D1/de active Active
- 2005-09-22 RU RU2007110479/04A patent/RU2382036C2/ru not_active IP Right Cessation
- 2005-09-22 BR BRPI0516754-0A patent/BRPI0516754A/pt not_active IP Right Cessation
- 2005-09-22 AU AU2005291541A patent/AU2005291541B2/en not_active Expired - Fee Related
- 2005-09-22 MX MX2007003911A patent/MX2007003911A/es active IP Right Grant
- 2005-09-22 JP JP2007533918A patent/JP2008514662A/ja active Pending
- 2005-09-22 AT AT05796666T patent/ATE477248T1/de active
- 2005-09-22 KR KR1020077007227A patent/KR100875041B1/ko not_active IP Right Cessation
- 2005-09-22 NZ NZ553848A patent/NZ553848A/en not_active IP Right Cessation
- 2005-09-27 TW TW094133563A patent/TW200626567A/zh unknown
- 2005-09-27 AR ARP050104050A patent/AR051115A1/es unknown
- 2005-09-28 MY MYPI20054561A patent/MY139409A/en unknown
-
2007
- 2007-03-27 NO NO20071616A patent/NO20071616L/no not_active Application Discontinuation
- 2007-03-29 IL IL182304A patent/IL182304A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
AR051115A1 (es) | 2006-12-20 |
CA2581921A1 (en) | 2006-04-13 |
RU2382036C2 (ru) | 2010-02-20 |
MX2007003911A (es) | 2007-05-21 |
KR20070047844A (ko) | 2007-05-07 |
AU2005291541A1 (en) | 2006-04-13 |
NZ553848A (en) | 2010-01-29 |
EP1797051B1 (en) | 2010-08-11 |
TW200626567A (en) | 2006-08-01 |
IL182304A0 (en) | 2007-07-24 |
ATE477248T1 (de) | 2010-08-15 |
EP1797051A1 (en) | 2007-06-20 |
MY139409A (en) | 2009-09-30 |
NO20071616L (no) | 2007-04-25 |
DE602005022896D1 (de) | 2010-09-23 |
RU2007110479A (ru) | 2008-11-10 |
WO2006037481A1 (en) | 2006-04-13 |
KR100875041B1 (ko) | 2008-12-19 |
JP2008514662A (ja) | 2008-05-08 |
AU2005291541B2 (en) | 2011-03-10 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BRPI0511532A (pt) | composto, uso do mesmo, composição farmacêutica, e, métodos para a terapia de distúrbios gastrointestinais funcionais e de sìndrome do intestino irritável em um animal de sangue quente, e para a preparação de um composto | |
UY30183A1 (es) | Derivados de quinolina | |
BRPI0511504A (pt) | composto ou um sal farmaceuticamente aceitável do mesmo, e, agente preventivo ou terapêutico para uma doença resultante de beta-amilóides | |
ECSP10010197A (es) | Derivados de piridina y pirazina útiles en el tratamiento de trastornos de proliferación celular | |
BRPI0515860B8 (pt) | derivados de tetralin e indano, seus usos, e composição farmacêutica | |
BRPI0607545A2 (pt) | composto, uso de um composto de fórmula i ou um sal farmaceuticamente aceitável do mesmo, e, composição farmacêutica | |
UY29781A1 (es) | Compuestos diazaspiro sustituidos, sales farmacéuticamente aceptables, composiciones farmacéuticas que contienen los compuestos o sales, métodos de preparación y usos | |
BRPI0720551A2 (pt) | composto ou um sal farmaceuticamente aceitável do mesmo, e, uso do mesmo, método para o tratamento de câncer, processos para a preparação de uma composição farmacêutica e de um composto ou de um sal farmaceuticamente aceitável do mesmo | |
MY144655A (en) | Pyrimidine urea derivatives as kinase inhibitors | |
SE0402735D0 (sv) | Novel compounds | |
UY27604A1 (es) | Compuestos químicos. | |
DE60140814D1 (de) | N-phenyl-2-pyrimidine-amine derivatives | |
BRPI0517792A (pt) | macrolonas - quinolonas amino-substituìdas | |
TW200621737A (en) | 2-carbamide-4-phenylthiazole derivatives, preparation thereof and therapeutic use thereof | |
NO20091893L (no) | Nye 1,4-benzotiepin-1,1-dioksidderivater som er substituert med benzylgrupper, fremgangsmater for fremstilling av medisiner inneholdende forbindelsene og anvendelse derav. | |
NO20085087L (no) | Nye heterocykliske forbindelser | |
ATE499372T1 (de) | Azabenzimidalzolderivate, ihre herstellung und ihre verwendung als antikrebsmittel | |
NO20062491L (no) | Benzoksazinderivter og deres anvendelse | |
BRPI0413094A (pt) | derivados de quinolina e seu uso em terapia | |
BRPI0508485A (pt) | compostos de pentafluorsulfanila, sua fabricação e uso como agentes farmacêuticos | |
TW200639156A (en) | New compounds | |
BRPI0416853A (pt) | pirazolila e imidazolila pirimidinas | |
BRPI0720742B8 (pt) | derivados de heteroaril pirrolidinil e piperidinil cetona, seus usos e composição farmacêutica compreendo os mesmos | |
SE0302546D0 (sv) | New compounds | |
BRPI0411246A (pt) | composto, uso do mesmo, composição farmacêutica, e, métodos para terapia contra dor em um animal de sangue quente e para a preparação de um composto |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 7A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2168 DE 24/07/2012. |