BRPI0507671A - taxanos substituìdos com éster de ciclopentila em c10 - Google Patents

taxanos substituìdos com éster de ciclopentila em c10

Info

Publication number
BRPI0507671A
BRPI0507671A BRPI0507671-4A BRPI0507671A BRPI0507671A BR PI0507671 A BRPI0507671 A BR PI0507671A BR PI0507671 A BRPI0507671 A BR PI0507671A BR PI0507671 A BRPI0507671 A BR PI0507671A
Authority
BR
Brazil
Prior art keywords
substituent
cyclopentyl ester
ester substituted
substituted taxanes
taxanes
Prior art date
Application number
BRPI0507671-4A
Other languages
English (en)
Inventor
Robert A Holton
Phong Vu
Original Assignee
Univ Florida State Res Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Florida State Res Found filed Critical Univ Florida State Res Found
Publication of BRPI0507671A publication Critical patent/BRPI0507671A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Epoxy Compounds (AREA)

Abstract

TAXANOS SUBSTITUìDOS COM éSTER DE CICLOPENTILA EM C10. A presente invenção se refere-se a um taxano tendo um substituinte de éster de ciclopentila em C10, um substituinte e ceto em C9, um substituinte de hidróxi em C2, um substituinte de 2- tienila em C3' e um substituinte de isopropoxicarbamento em C3.
BRPI0507671-4A 2004-02-13 2005-02-14 taxanos substituìdos com éster de ciclopentila em c10 BRPI0507671A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US54475504P 2004-02-13 2004-02-13
US61350304P 2004-09-27 2004-09-27
PCT/US2005/004442 WO2005079319A2 (en) 2004-02-13 2005-02-14 C10 cyclopentyl ester substituted taxanes

Publications (1)

Publication Number Publication Date
BRPI0507671A true BRPI0507671A (pt) 2007-07-17

Family

ID=34890477

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0507671-4A BRPI0507671A (pt) 2004-02-13 2005-02-14 taxanos substituìdos com éster de ciclopentila em c10

Country Status (22)

Country Link
US (2) US7589111B2 (pt)
EP (1) EP1713798B1 (pt)
JP (1) JP4879757B2 (pt)
KR (1) KR101169818B1 (pt)
AR (1) AR047704A1 (pt)
AT (1) ATE486596T1 (pt)
AU (1) AU2005214065B2 (pt)
BR (1) BRPI0507671A (pt)
CA (1) CA2556200C (pt)
CR (1) CR8554A (pt)
DE (1) DE602005024518D1 (pt)
EC (1) ECSP066765A (pt)
HK (1) HK1097534A1 (pt)
HN (1) HN2005000054A (pt)
IL (1) IL177372A (pt)
NO (1) NO20064090L (pt)
NZ (1) NZ548769A (pt)
PE (1) PE20050693A1 (pt)
RU (1) RU2006132741A (pt)
SV (1) SV2006002010A (pt)
TW (1) TWI353354B (pt)
WO (1) WO2005079319A2 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1303077C (zh) * 2004-01-16 2007-03-07 桂林晖昂生化药业有限责任公司 合成紫杉烷的制备工艺
JP4833126B2 (ja) * 2007-03-26 2011-12-07 Ｎｔｎ株式会社 潤滑剤劣化検出装置および検出装置付き軸受
CN113209287B (zh) * 2021-02-04 2022-07-08 中国农业科学院农业环境与可持续发展研究所 油包水型纳米疫苗佐剂、制备方法及其应用

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Also Published As

Publication number Publication date
ECSP066765A (es) 2006-12-29
CA2556200C (en) 2012-06-26
ATE486596T1 (de) 2010-11-15
JP4879757B2 (ja) 2012-02-22
SV2006002010A (es) 2006-08-23
US7589111B2 (en) 2009-09-15
HK1097534A1 (en) 2007-06-29
WO2005079319A2 (en) 2005-09-01
TW200530209A (en) 2005-09-16
CA2556200A1 (en) 2005-09-01
CR8554A (es) 2008-04-25
AR047704A1 (es) 2006-02-08
AU2005214065A1 (en) 2005-09-01
KR101169818B1 (ko) 2012-07-30
AU2005214065B2 (en) 2009-11-12
IL177372A0 (en) 2006-12-10
JP2007522236A (ja) 2007-08-09
NO20064090L (no) 2006-11-10
PE20050693A1 (es) 2005-09-27
DE602005024518D1 (en) 2010-12-16
EP1713798A4 (en) 2007-12-05
EP1713798B1 (en) 2010-11-03
HN2005000054A (es) 2009-02-18
US20100056614A1 (en) 2010-03-04
EP1713798A2 (en) 2006-10-25
IL177372A (en) 2011-09-27
WO2005079319A3 (en) 2005-11-17
TWI353354B (en) 2011-12-01
KR20060129018A (ko) 2006-12-14
RU2006132741A (ru) 2008-03-20
US20050228037A1 (en) 2005-10-13
NZ548769A (en) 2009-10-30
AU2005214065A2 (en) 2005-09-01
US8003812B2 (en) 2011-08-23

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2308 DE 31/03/2015.