BR9911624A - Compostos heterocìclicos substituìdos de cinco membros, composições fungicidas contendo os mesmos e processos para a produção dos mesmos - Google Patents
Compostos heterocìclicos substituìdos de cinco membros, composições fungicidas contendo os mesmos e processos para a produção dos mesmosInfo
- Publication number
- BR9911624A BR9911624A BR9911624-3A BR9911624A BR9911624A BR 9911624 A BR9911624 A BR 9911624A BR 9911624 A BR9911624 A BR 9911624A BR 9911624 A BR9911624 A BR 9911624A
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- lower alkyl
- compound
- substituted
- processes
- Prior art date
Links
- 230000000855 fungicidal effect Effects 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 6
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 125000003118 aryl group Chemical group 0.000 abstract 2
- ABBZJHFBQXYTLU-UHFFFAOYSA-N but-3-enamide Chemical compound NC(=O)CC=C ABBZJHFBQXYTLU-UHFFFAOYSA-N 0.000 abstract 2
- 230000002194 synthesizing effect Effects 0.000 abstract 2
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 abstract 1
- AYFUJEYYHDFXQA-UHFFFAOYSA-N 4-hydroxy-4,5-dimethyl-2-trimethylsilylthiolane-3-carboxylic acid Chemical compound CC1SC([Si](C)(C)C)C(C(O)=O)C1(C)O AYFUJEYYHDFXQA-UHFFFAOYSA-N 0.000 abstract 1
- 241001149475 Gaeumannomyces graminis Species 0.000 abstract 1
- 230000009418 agronomic effect Effects 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- MXMXHPPIGKYTAR-UHFFFAOYSA-N silthiofam Chemical compound CC=1SC([Si](C)(C)C)=C(C(=O)NCC=C)C=1C MXMXHPPIGKYTAR-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/0825—Preparations of compounds not comprising Si-Si or Si-cyano linkages
- C07F7/083—Syntheses without formation of a Si-C bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
- C07F7/0814—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring said ring is substituted at a C ring atom by Si
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Patente de Invenção: "COMPOSTOS HETEROCìCLICOSSUBSTITUìDOS DE CINCO MEMBROS, COMPOSIçõESFUNGICIDAS CONTENDO OS MESMOS E PROCESSOS PARAA PRODUçãO DOS MESMOS". O composto fungicida4,5-dimetil-N-2-propenil-2-(trimetilsilil)-3tiofenocarboxamida (fórmula(I)) tem mostrado controle superior e inesperado do crescimento defungos de origem no solo Gaeumannomyces graminis (Gg). Apresente invenção provê um novo composto para sintetizar ocomposto de fórmula (1) que usa o composto alilamida de ácido4-hidróxi-4,5-dimetil-2-trimetilsilanil-dihidrotiofeno-3-carboxílico(fórmula (II)), assim como novos compostos de síntese de alilamida.Além disso, a própria fórmula (II) foi inesperadamente verificadacomo provendo controle de Gg. Assim, os compostos tendofórmula (III) ou sais agronómicos e composições dos mesmos sãoesperados como também provendo este controle; em que Q é -NH,S ou O; W é O ou S, X é -OH, -OAc, -OR, onde R é alquila inferior,Y é S, O ou -NH; Z é -Si(R)~ 3~, -C(R)~ 3~, onde R é alquilainferior, R~ 1~ é uma alquila inferior, alila ou propargila, R~ 2~ éuma alquila inferior ou arila, e R~ 3~ e R~ 4~ sãoindependentemente escolhidos dentre hidrogênio, alquila inferior earila; opcionalmente, R~ 2~ e R~ 3~ juntos formam um anel de 5ou 6 membros.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8839898P | 1998-06-05 | 1998-06-05 | |
| PCT/US1999/012502 WO1999062915A1 (en) | 1998-06-05 | 1999-06-04 | Substituted five-membered heterocyclic compounds, fungicidal compositions containing them and methods of making thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BR9911624A true BR9911624A (pt) | 2001-10-30 |
| BR9911624B1 BR9911624B1 (pt) | 2010-07-13 |
Family
ID=22211142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI9911624-3A BR9911624B1 (pt) | 1998-06-05 | 1999-06-04 | processos para sintetizar um fungicida e para controlar doença em uma planta, compostos heterocìclicos substituìdos de cinco membros e composição fungicida contendo os mesmos. |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US6140511A (pt) |
| EP (1) | EP1084130B1 (pt) |
| CN (2) | CN1182142C (pt) |
| AT (1) | ATE223422T1 (pt) |
| AU (1) | AU762985B2 (pt) |
| BR (1) | BR9911624B1 (pt) |
| CA (1) | CA2334221C (pt) |
| CZ (1) | CZ299799B6 (pt) |
| DE (1) | DE69902782T2 (pt) |
| DK (1) | DK1084130T3 (pt) |
| ES (1) | ES2183568T3 (pt) |
| PL (1) | PL199097B1 (pt) |
| PT (1) | PT1084130E (pt) |
| RU (1) | RU2220973C2 (pt) |
| UA (1) | UA58598C2 (pt) |
| WO (1) | WO1999062915A1 (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1275301A1 (en) | 2001-07-10 | 2003-01-15 | Bayer CropScience S.A. | Trisubstituted heterocyclic compounds and their use as fungicides |
| US7582589B2 (en) * | 2003-05-07 | 2009-09-01 | Syngenta Crop Protection, Inc. | 3-carbonylaminothiophenes and their use as fungicides |
| DE102011017541A1 (de) | 2010-04-29 | 2011-11-10 | Basf Se | Synergistische fungizide Mischungen |
| CN103044479B (zh) * | 2012-12-12 | 2015-09-02 | 河南农业大学 | 杀菌剂硅噻菌胺的合成方法 |
| CN105111229B (zh) * | 2015-06-08 | 2019-03-08 | 杭州师范大学 | 一种硅噻菌胺的合成方法 |
| CN106905357B (zh) * | 2017-03-09 | 2019-04-09 | 南京工业大学 | 一种硅噻菌胺关键中间体的制备方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU219131B (hu) * | 1991-10-18 | 2001-02-28 | Monsanto Co. | Módszer és fungicid készítmény növények torsgombabetegségének gátlására és a hatóanyagok |
| US5486621A (en) * | 1994-12-15 | 1996-01-23 | Monsanto Company | Fungicides for the control of take-all disease of plants |
-
1999
- 1999-04-06 UA UA2001010126A patent/UA58598C2/uk unknown
- 1999-06-04 ES ES99927224T patent/ES2183568T3/es not_active Expired - Lifetime
- 1999-06-04 CN CNB998093394A patent/CN1182142C/zh not_active Expired - Lifetime
- 1999-06-04 PT PT99927224T patent/PT1084130E/pt unknown
- 1999-06-04 DK DK99927224T patent/DK1084130T3/da active
- 1999-06-04 RU RU2001101165/04A patent/RU2220973C2/ru active
- 1999-06-04 EP EP99927224A patent/EP1084130B1/en not_active Expired - Lifetime
- 1999-06-04 PL PL345161A patent/PL199097B1/pl unknown
- 1999-06-04 US US09/326,225 patent/US6140511A/en not_active Expired - Lifetime
- 1999-06-04 CZ CZ20004529A patent/CZ299799B6/cs not_active IP Right Cessation
- 1999-06-04 WO PCT/US1999/012502 patent/WO1999062915A1/en active IP Right Grant
- 1999-06-04 BR BRPI9911624-3A patent/BR9911624B1/pt not_active IP Right Cessation
- 1999-06-04 AU AU44183/99A patent/AU762985B2/en not_active Expired
- 1999-06-04 DE DE69902782T patent/DE69902782T2/de not_active Expired - Lifetime
- 1999-06-04 AT AT99927224T patent/ATE223422T1/de active
- 1999-06-04 CN CNB2004100898232A patent/CN100503594C/zh not_active Expired - Lifetime
- 1999-06-04 CA CA002334221A patent/CA2334221C/en not_active Expired - Lifetime
-
2000
- 2000-07-05 US US09/609,211 patent/US6291513B1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| UA58598C2 (uk) | 2003-08-15 |
| CZ299799B6 (cs) | 2008-11-26 |
| RU2220973C2 (ru) | 2004-01-10 |
| CN100503594C (zh) | 2009-06-24 |
| EP1084130B1 (en) | 2002-09-04 |
| DE69902782T2 (de) | 2003-05-28 |
| WO1999062915A1 (en) | 1999-12-09 |
| PL345161A1 (en) | 2001-12-03 |
| ATE223422T1 (de) | 2002-09-15 |
| DE69902782D1 (de) | 2002-10-10 |
| CZ20004529A3 (en) | 2001-06-13 |
| US6291513B1 (en) | 2001-09-18 |
| PT1084130E (pt) | 2003-01-31 |
| CA2334221C (en) | 2008-12-23 |
| AU4418399A (en) | 1999-12-20 |
| CN1182142C (zh) | 2004-12-29 |
| ES2183568T3 (es) | 2003-03-16 |
| EP1084130A1 (en) | 2001-03-21 |
| BR9911624B1 (pt) | 2010-07-13 |
| CN1623995A (zh) | 2005-06-08 |
| CN1314907A (zh) | 2001-09-26 |
| PL199097B1 (pl) | 2008-08-29 |
| AU762985B2 (en) | 2003-07-10 |
| CA2334221A1 (en) | 1999-12-09 |
| US6140511A (en) | 2000-10-31 |
| DK1084130T3 (da) | 2002-10-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 13/07/2010, OBSERVADAS AS CONDICOES LEGAIS. |
|
| B25A | Requested transfer of rights approved |
Owner name: MITSUI AND CO., LTD. (JP) |
|
| B21A | Patent or certificate of addition expired [chapter 21.1 patent gazette] |
Free format text: PATENTE EXTINTA EM 13.07.2020 |