BR9907233A - Polìmeros inibidores de lipase e seu uso - Google Patents

Polìmeros inibidores de lipase e seu uso

Info

Publication number
BR9907233A
BR9907233A BR9907233-5A BR9907233A BR9907233A BR 9907233 A BR9907233 A BR 9907233A BR 9907233 A BR9907233 A BR 9907233A BR 9907233 A BR9907233 A BR 9907233A
Authority
BR
Brazil
Prior art keywords
polymers
lipase
patient
inhibiting polymers
methods
Prior art date
Application number
BR9907233-5A
Other languages
English (en)
Inventor
W Harry Mandeville Iii
Molly Kate Boie
Venkata R Garigapati
Original Assignee
Geltex Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Geltex Pharma Inc filed Critical Geltex Pharma Inc
Publication of BR9907233A publication Critical patent/BR9907233A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)

Abstract

"POLìMEROS INIBIDORES DE LIPASE E SEU USO". A presente invenção descreve um método para tratar obesidade num paciente administrando-se ao paciente um polímero que tenha sido substituído com um ou mais grupos que inibem lipases, que são enzimas responsáveis pela hidrólise de gordura. A invenção refere-se ainda aos polímeros empregados nos métodos descritos na presente patente, bem como a intermediários e métodos novos para preparação dos polímeros.
BR9907233-5A 1998-01-09 1999-01-06 Polìmeros inibidores de lipase e seu uso BR9907233A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US537998A 1998-01-09 1998-01-09
US09/166,510 US6267952B1 (en) 1998-01-09 1998-10-05 Lipase inhibiting polymers
PCT/US1999/000195 WO1999034786A2 (en) 1998-01-09 1999-01-06 Lipase inhibiting polymers

Publications (1)

Publication Number Publication Date
BR9907233A true BR9907233A (pt) 2000-10-17

Family

ID=26674279

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9907233-5A BR9907233A (pt) 1998-01-09 1999-01-06 Polìmeros inibidores de lipase e seu uso

Country Status (20)

Country Link
US (6) US6267952B1 (pt)
EP (1) EP1043982B1 (pt)
JP (1) JP2002500182A (pt)
KR (1) KR100620634B1 (pt)
CN (2) CN1636574A (pt)
AT (1) ATE308979T1 (pt)
AU (1) AU747016B2 (pt)
BR (1) BR9907233A (pt)
CA (1) CA2318416A1 (pt)
DE (1) DE69928219T2 (pt)
DK (1) DK1043982T3 (pt)
ES (1) ES2253872T3 (pt)
HK (1) HK1079706A1 (pt)
HU (1) HUP0101128A3 (pt)
IL (1) IL137098A (pt)
NO (1) NO20003511L (pt)
NZ (1) NZ505296A (pt)
PL (1) PL193453B1 (pt)
RU (1) RU2207861C2 (pt)
WO (1) WO1999034786A2 (pt)

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Also Published As

Publication number Publication date
NO20003511D0 (no) 2000-07-07
PL193453B1 (pl) 2007-02-28
EP1043982B1 (en) 2005-11-09
US20050085535A1 (en) 2005-04-21
ES2253872T3 (es) 2006-06-01
US6875428B2 (en) 2005-04-05
PL344022A1 (en) 2001-09-24
IL137098A0 (en) 2001-06-14
DK1043982T3 (da) 2006-02-13
EP1043982A2 (en) 2000-10-18
ATE308979T1 (de) 2005-11-15
IL137098A (en) 2006-07-05
AU747016B2 (en) 2002-05-09
HUP0101128A2 (hu) 2002-01-28
KR20010034012A (ko) 2001-04-25
RU2207861C2 (ru) 2003-07-10
AU2105699A (en) 1999-07-26
NO20003511L (no) 2000-09-07
CN1636574A (zh) 2005-07-13
CN1287489A (zh) 2001-03-14
US20030185789A1 (en) 2003-10-02
HUP0101128A3 (en) 2003-01-28
US6572850B1 (en) 2003-06-03
WO1999034786A3 (en) 2000-02-03
US6267952B1 (en) 2001-07-31
HK1079706A1 (zh) 2006-04-13
DE69928219D1 (de) 2005-12-15
JP2002500182A (ja) 2002-01-08
NZ505296A (en) 2002-12-20
WO1999034786A2 (en) 1999-07-15
KR100620634B1 (ko) 2006-09-13
US6352692B1 (en) 2002-03-05
CA2318416A1 (en) 1999-07-15
DE69928219T2 (de) 2006-07-27
US6558657B1 (en) 2003-05-06

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