BR9709676A - Novos derivados aromáticos substituìdos por uma ribose, seu processo de preparação e sua aplicação como medicamentos - Google Patents

Novos derivados aromáticos substituìdos por uma ribose, seu processo de preparação e sua aplicação como medicamentos

Info

Publication number
BR9709676A
BR9709676A BR9709676-8A BR9709676A BR9709676A BR 9709676 A BR9709676 A BR 9709676A BR 9709676 A BR9709676 A BR 9709676A BR 9709676 A BR9709676 A BR 9709676A
Authority
BR
Brazil
Prior art keywords
alkyl
ribose
medicines
application
preparation process
Prior art date
Application number
BR9709676-8A
Other languages
English (en)
Inventor
Michel Klich
Patrick Laurin
Laurent Schio
Branislav Musicki
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of BR9709676A publication Critical patent/BR9709676A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/06—Benzopyran radicals
    • C07H17/065—Benzo[b]pyrans
    • C07H17/075—Benzo[b]pyran-2-ones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: <B>''NOVOS DERIVADOS AROMáTICOS SUBSTITUìDOS POR UMA RIBOSE, SEU PROCESSO DE PREPARAçãO E SUA APLICAçãO COMO MEDICAMENTOS''<D>. A invenção tem por objeto os compostos de fórmula (I), na qual R1= H, OH, alquila, alquenila ou alquinila, eventualmente substituído ou alcóxi; R2= H, Hal; R3= H, alquila, Hal; R4 = (a), Rg e RH: H, alquila, arila heterociclo; R5= H ou O-alquila; R6 = alquila; R6 = alquila; R7 = H ou alquila. Os compostos de fórmula (I) apresentam propriedades antibióticas.
BR9709676-8A 1996-06-11 1997-06-10 Novos derivados aromáticos substituìdos por uma ribose, seu processo de preparação e sua aplicação como medicamentos BR9709676A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9607207A FR2749585B1 (fr) 1996-06-11 1996-06-11 Nouveaux derives aromatiques substitues par un ribose, leur procede de preparation et leur application comme medicaments
PCT/FR1997/001022 WO1997047634A1 (fr) 1996-06-11 1997-06-10 Nouveaux derives aromatiques substitues par un ribose, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
BR9709676A true BR9709676A (pt) 2000-05-09

Family

ID=9492918

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9709676-8A BR9709676A (pt) 1996-06-11 1997-06-10 Novos derivados aromáticos substituìdos por uma ribose, seu processo de preparação e sua aplicação como medicamentos

Country Status (24)

Country Link
US (2) US6350733B1 (pt)
EP (1) EP0906326B1 (pt)
JP (1) JP2000511920A (pt)
CN (1) CN1308342C (pt)
AR (1) AR008228A1 (pt)
AT (1) ATE209212T1 (pt)
AU (1) AU712665B2 (pt)
BR (1) BR9709676A (pt)
CA (1) CA2258152C (pt)
CZ (1) CZ296204B6 (pt)
DE (1) DE69709732T2 (pt)
DK (1) DK0906326T3 (pt)
ES (1) ES2165067T3 (pt)
FR (1) FR2749585B1 (pt)
HU (1) HU222787B1 (pt)
IL (3) IL127133A0 (pt)
NO (1) NO313638B1 (pt)
PL (1) PL187204B1 (pt)
PT (1) PT906326E (pt)
RU (1) RU2194052C2 (pt)
TR (1) TR199802555T2 (pt)
TW (1) TW561159B (pt)
WO (1) WO1997047634A1 (pt)
ZA (1) ZA974840B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW538046B (en) * 1998-01-08 2003-06-21 Hoechst Marion Roussel Inc Aromatic amides having antiobiotic activities and the preparation processes, intermediates and pharmaceutical composition thereof
FR2784681B1 (fr) * 1998-10-15 2003-01-17 Hoechst Marion Roussel Inc Nouveaux amides aromatiques, leur procede de preparation et leur application comme medicaments
AU2002300839B2 (en) * 1998-01-08 2004-04-29 Novexel Novel aromatic amides, preparation method and application as medicines
FR2773369B1 (fr) * 1998-01-08 2001-02-16 Hoechst Marion Roussel Inc Nouveaux amides aromatiques, leur procede de preparation et leur application comme medicaments
FR2844273B1 (fr) * 2002-09-05 2008-04-04 Aventis Pharma Sa Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens.
US7439253B2 (en) * 2002-12-06 2008-10-21 Novexel Heterocyclic compounds, their preparation and their use as medicaments, in particular as antibacterials and beta-lactamase inhibitors
AU2005233614C1 (en) * 2004-04-08 2012-07-19 Armetheon, Inc. Materials and methods for treating coagulation disorders
AU2006343604A1 (en) * 2006-05-15 2007-11-22 Xtl Biopharmaceuticals, Ltd. 3,4-disubstituted coumarin and quinolone compounds

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4226978A (en) * 1978-03-13 1980-10-07 Miles Laboratories, Inc. β-Galactosyl-umbelliferone-labeled aminoglycoside antibiotics and intermediates in their preparation
EP0654479B1 (en) * 1993-11-15 2000-03-15 Kureha Chemical Industry Co., Ltd. Esculetin derivatives and method for manufacture thereof, use thereof, and pharmaceutical composition
TW538046B (en) * 1998-01-08 2003-06-21 Hoechst Marion Roussel Inc Aromatic amides having antiobiotic activities and the preparation processes, intermediates and pharmaceutical composition thereof

Also Published As

Publication number Publication date
DE69709732T2 (de) 2002-08-08
FR2749585A1 (fr) 1997-12-12
IL146925A (en) 2006-10-05
ZA974840B (en) 1998-11-20
PL330550A1 (en) 1999-05-24
AR008228A1 (es) 1999-12-29
CA2258152C (fr) 2006-08-29
HUP9902925A3 (en) 2000-06-28
ES2165067T3 (es) 2002-03-01
CN1227564A (zh) 1999-09-01
IL127133A0 (en) 1999-09-22
EP0906326B1 (fr) 2001-11-21
PT906326E (pt) 2002-05-31
PL187204B1 (pl) 2004-06-30
CZ296204B6 (cs) 2006-02-15
US6350733B1 (en) 2002-02-26
FR2749585B1 (fr) 1998-08-14
JP2000511920A (ja) 2000-09-12
NO985790L (no) 1999-02-10
DK0906326T3 (da) 2002-05-21
DE69709732D1 (de) 2002-02-21
US20020010322A1 (en) 2002-01-24
CA2258152A1 (fr) 1997-12-18
NO313638B1 (no) 2002-11-04
CN1308342C (zh) 2007-04-04
CZ406998A3 (cs) 1999-04-14
RU2194052C2 (ru) 2002-12-10
WO1997047634A1 (fr) 1997-12-18
HU222787B1 (hu) 2003-10-28
TW561159B (en) 2003-11-11
TR199802555T2 (xx) 1999-04-21
EP0906326A1 (fr) 1999-04-07
US6812331B2 (en) 2004-11-02
AU3265997A (en) 1998-01-07
AU712665B2 (en) 1999-11-11
NO985790D0 (no) 1998-12-10
IL127133A (en) 2006-08-01
ATE209212T1 (de) 2001-12-15

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: AVENTIS PHARMA S.A. (FR)

Free format text: TRANSFERIDO POR FUSAO DE: HOECHST MARION ROUSSEL

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B25A Requested transfer of rights approved

Owner name: NOVEXEL (FR)

Free format text: TRANSFERIDO DE: AVENTIS PHARMA S.A.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: DE ACORDO COM O ART. 37, INDEFIRO O PRESENTE PEDIDO, TENDO POR BASE O ART. 8O COMBINADO COM ART. 13 DA LPI.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.