BR9503468A - Composto composiçao farmacêutica processo para preparaçao do composto seu uso e processo para tratar um animal afetado por ou em risco de contrair uma doença viral ou relacionada - Google Patents

Composto composiçao farmacêutica processo para preparaçao do composto seu uso e processo para tratar um animal afetado por ou em risco de contrair uma doença viral ou relacionada

Info

Publication number
BR9503468A
BR9503468A BR9503468A BR9503468A BR9503468A BR 9503468 A BR9503468 A BR 9503468A BR 9503468 A BR9503468 A BR 9503468A BR 9503468 A BR9503468 A BR 9503468A BR 9503468 A BR9503468 A BR 9503468A
Authority
BR
Brazil
Prior art keywords
compound
contracting
viral
treat
risk
Prior art date
Application number
BR9503468A
Other languages
English (en)
Inventor
John J Nestor
Scott W Womble
Hans Maag
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23079211&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9503468(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR9503468A publication Critical patent/BR9503468A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
BR9503468A 1994-07-28 1995-07-27 Composto composiçao farmacêutica processo para preparaçao do composto seu uso e processo para tratar um animal afetado por ou em risco de contrair uma doença viral ou relacionada BR9503468A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US28189394A 1994-07-28 1994-07-28

Publications (1)

Publication Number Publication Date
BR9503468A true BR9503468A (pt) 1996-02-27

Family

ID=23079211

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9503468A BR9503468A (pt) 1994-07-28 1995-07-27 Composto composiçao farmacêutica processo para preparaçao do composto seu uso e processo para tratar um animal afetado por ou em risco de contrair uma doença viral ou relacionada

Country Status (33)

Country Link
EP (1) EP0694547B1 (pt)
JP (1) JP3090305B2 (pt)
KR (1) KR100358626B1 (pt)
CN (1) CN1045089C (pt)
AT (1) ATE179173T1 (pt)
AU (1) AU697107B2 (pt)
BR (1) BR9503468A (pt)
CA (1) CA2154721C (pt)
CO (1) CO4410181A1 (pt)
CY (2) CY2180B1 (pt)
CZ (1) CZ290511B6 (pt)
DE (3) DE69509173T2 (pt)
DK (1) DK0694547T3 (pt)
ES (1) ES2083348T3 (pt)
FI (1) FI112080B (pt)
GR (2) GR960300021T1 (pt)
HK (1) HK1012339A1 (pt)
HU (1) HU216867B (pt)
IL (1) IL114735A (pt)
LU (1) LU91136I2 (pt)
MA (1) MA23631A1 (pt)
MY (1) MY114393A (pt)
NL (1) NL300071I2 (pt)
NO (2) NO312899B1 (pt)
NZ (1) NZ272652A (pt)
PE (1) PE32296A1 (pt)
PL (1) PL180609B1 (pt)
RU (1) RU2133749C1 (pt)
SA (1) SA95160158B1 (pt)
TR (1) TR199500895A2 (pt)
TW (1) TW434242B (pt)
UY (1) UY24006A1 (pt)
ZA (1) ZA956228B (pt)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6458772B1 (en) 1909-10-07 2002-10-01 Medivir Ab Prodrugs
US5700936A (en) * 1996-01-26 1997-12-23 Syntex (U.S.A.) Inc. Process for preparing a 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl) methoxy-1,3-propanediol valinate
US5840890A (en) * 1996-01-26 1998-11-24 Syntex (U.S.A.) Inc. Process for preparing a 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl)methoxy-1,3-propanediol derivative
WO1997027198A1 (en) * 1996-01-26 1997-07-31 F.Hoffmann-La Roche Ag Process for preparing purine derivatives
WO1997027194A1 (en) * 1996-01-26 1997-07-31 F. Hoffmann-La Roche Ag Process for preparing purine derivatives
US5756736A (en) * 1996-01-26 1998-05-26 Syntex (U.S.A.) Inc. Process for preparing a 2-(2-amino-1,6-dihydro-6-oxo-purin-9-yl)methoxy-1,3-propanediol derivative
US6703394B2 (en) 1996-02-16 2004-03-09 Medivir Ab Acyclic nucleoside derivatives
US5869493A (en) * 1996-02-16 1999-02-09 Medivir Ab Acyclic nucleoside derivatives
ES2186127T3 (es) * 1997-02-10 2003-05-01 Medivir Ab Sintesis de derivados de nucleosidos aciclicos.
US6184376B1 (en) 1997-02-10 2001-02-06 Mediver Ab Synthesis of acyclic nucleoside derivatives
CZ300757B6 (cs) * 1997-08-15 2009-08-05 Medivir Ab Nukleosidové analogy, jako jsou antivirální cinidla obsahující inhibitory retrovirální reverzní transkriptázy a DNA polymerázy viru hepatitidy B (HBV)
WO1999032490A1 (en) * 1997-12-19 1999-07-01 Bristol-Myers Squibb Company Prodrugs of lobucavir and methods of use
WO1999051613A1 (en) * 1998-04-03 1999-10-14 Medivir Ab Prodrugs of phosphorous-containing pharmaceuticals
KR20030015655A (ko) * 2001-08-17 2003-02-25 한미약품공업 주식회사 항암제의 경구흡수율을 증가시키는 인단계 화합물의결정성 산부가염, 이의 제조방법 및 이를 함유하는 약학적조성물
WO2003091214A1 (en) * 2002-04-23 2003-11-06 Aventis Pharmaceuticals Inc. 3-substituted amino-1h-indole-2-carboxylic acid and 3-substituted amino-benzo
EP1552833B1 (en) 2002-10-16 2016-12-28 Takeda Pharmaceutical Company Limited Process for producing an amorphous optically active isomer of lansoprazole
EP3025718A1 (en) 2003-01-14 2016-06-01 Gilead Sciences, Inc. Compositions and methods for combination antiviral therapy
CA2537132A1 (en) * 2003-08-28 2005-03-10 Ranbaxy Laboratories Limited Amorphous valganciclovir hydrochloride
JP5563735B2 (ja) 2004-06-16 2014-07-30 タケダ ファーマシューティカルズ ユー.エス.エー. インコーポレイティド Ppi多回剤形
CA2580313C (en) * 2004-07-19 2016-03-15 Biocon Limited Insulin-oligomer conjugates, formulations and uses thereof
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
ZA200702234B (en) * 2006-03-21 2008-07-30 Cipla Ltd Preparation of ester of purine derivatives
US8173158B2 (en) 2007-10-12 2012-05-08 Takeda Pharmaceuticals U.S.A., Inc. Methods of treating gastrointestinal disorders independent of the intake of food
EP2714691B1 (en) * 2011-05-31 2016-09-07 Pharmathen S.A. Process for the preparation of 2-amino-9-((2-phenyl-1,3-dioxan-5-yloxy)methyl)-1h-purin-6(9h)-one compound useful in the preparation of valganciclovir
KR102312533B1 (ko) 2021-02-24 2021-10-15 주식회사 이웅 자동 스패너

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8202626A (nl) * 1982-06-29 1984-01-16 Stichting Rega V Z W Derivaten van 9-(2-hydroxyethoxymethyl)guanine.
IE842642L (en) * 1983-10-31 1985-04-30 Harvard College Purine Derivatives
ES8705889A1 (es) * 1984-12-12 1987-06-01 Syntex Inc Un metodo para preparar eteres alcaximetilicos y esteres alcoximetilicos de derivados de guananina.
AP55A (en) * 1987-08-15 1989-09-26 The Wellcome Foundation Ltd Therapeutic Acyclic Nucleosides
CA2005815C (en) * 1988-12-19 1999-08-03 Wellcome Foundation Limited (The) Antiviral acyclic nucleoside derivatives

Also Published As

Publication number Publication date
NO952977D0 (no) 1995-07-27
RU2133749C1 (ru) 1999-07-27
NZ272652A (en) 1996-12-20
MA23631A1 (fr) 1996-04-01
FI112080B (fi) 2003-10-31
JP3090305B2 (ja) 2000-09-18
CY2004003I1 (el) 2009-11-04
HU216867B (hu) 1999-09-28
NL300071I2 (nl) 2002-03-01
HU9502238D0 (en) 1995-09-28
DE10299032I1 (de) 2003-01-23
TR199500895A2 (tr) 1996-06-21
FI953592A (fi) 1996-01-29
CO4410181A1 (es) 1997-01-09
CY2004003I2 (el) 2009-11-04
NO952977L (no) 1996-01-29
MY114393A (en) 2002-10-31
UY24006A1 (es) 2001-07-31
PL180609B1 (pl) 2001-03-30
CN1045089C (zh) 1999-09-15
HK1012339A1 (en) 1999-07-30
DE69509173T2 (de) 1999-10-21
JPH0841061A (ja) 1996-02-13
GR3030678T3 (en) 1999-11-30
KR100358626B1 (ko) 2003-01-14
CA2154721C (en) 2001-01-02
DK0694547T3 (da) 2000-01-03
DE10299032I2 (de) 2006-06-14
ATE179173T1 (de) 1999-05-15
PE32296A1 (es) 1996-08-07
PL309812A1 (en) 1996-02-05
LU91136I2 (fr) 2005-07-06
CA2154721A1 (en) 1996-01-29
EP0694547A3 (en) 1996-06-05
TW434242B (en) 2001-05-16
AU2719595A (en) 1996-02-08
KR960004345A (ko) 1996-02-23
EP0694547A2 (en) 1996-01-31
ES2083348T3 (es) 1999-08-01
CY2180B1 (en) 2002-08-23
RU95113148A (ru) 1997-06-27
HUT73246A (en) 1996-07-29
SA95160158B1 (ar) 2006-05-20
CZ193995A3 (en) 1996-02-14
ZA956228B (en) 1996-02-22
ES2083348T1 (es) 1996-04-16
AU697107B2 (en) 1998-09-24
NO2003001I2 (no) 2007-06-11
EP0694547B1 (en) 1999-04-21
GR960300021T1 (en) 1996-04-30
NO312899B1 (no) 2002-07-15
CN1122804A (zh) 1996-05-22
DE694547T1 (de) 1996-10-24
DE69509173D1 (de) 1999-05-27
IL114735A0 (en) 1995-11-27
NL300071I1 (nl) 2002-02-01
IL114735A (en) 1998-06-15
CZ290511B6 (cs) 2002-08-14
FI953592A0 (fi) 1995-07-27

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
HKFN Application deemed withdrawn (deleted)
FB36 Technical and formal requirements: requirement - article 36 of industrial property law
HJEG Technical examination (opinion): technical examination (opinion) related to article 229 of industrial property law
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15N Others concerning applications: notification of judicial decision

Free format text: INPI-52400.0615/2004 TRIBUNAL REGIONAL FEDERAL DA 2A REGIAO 13A VARA FEDERAL DO RIO DE JANEIRO PROCESSO:NO0506840-58.2004.4.02.5101 APELANTE: F HOFFMANN LA ROCHE AG E OUTRO APELADO: F HOFFMANN LA ROCHE AG E OUTROS DECISAO: IMPROCEDENTE O PEDIDO DA INICIAL E CONCLUINDO PELO INDEFERIMENTO DO PEDIDO DE PATENTE DE INVENCAO PI 9503468-4 DE TITULO ?COMPOSTO, COMPOSICAO FARMACEUTICA, PROCESSO PARA PREPARACAO DO COMPOSTO, SEU USO, E PROCESSO PARA TRATAR UM ANIMAL AFETADO POR, OU SEM RISCO DE CONTRAIR, UMA DOENCA VIRAL OU RELACIONADA?, POR NAO PREENCHER OS REQUISITOS LEGAIS DE ATIVIDADE INVENTIVA E DE SUFICIENCIA DESCRITIVA.