BR112022012130A2 - Compostos antelmínticos compreendendo uma estrutura azaindólica - Google Patents

Compostos antelmínticos compreendendo uma estrutura azaindólica

Info

Publication number
BR112022012130A2
BR112022012130A2 BR112022012130A BR112022012130A BR112022012130A2 BR 112022012130 A2 BR112022012130 A2 BR 112022012130A2 BR 112022012130 A BR112022012130 A BR 112022012130A BR 112022012130 A BR112022012130 A BR 112022012130A BR 112022012130 A2 BR112022012130 A2 BR 112022012130A2
Authority
BR
Brazil
Prior art keywords
compounds
azaindolic
antelminthic
dirofilaria
helminths
Prior art date
Application number
BR112022012130A
Other languages
English (en)
Inventor
Berger Michael
Linder Michael
Schneider Carolin
Tanzler Janina
Sondern Ulrich
Original Assignee
Intervet Int Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intervet Int Bv filed Critical Intervet Int Bv
Publication of BR112022012130A2 publication Critical patent/BR112022012130A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P5/00—Nematocides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

COMPOSTOS ANTELMÍNTICOS COMPREENDENDO UMA ESTRUTURA AZAINDÓLICA. A presente invenção se refere a novos compostos antelmínticos. Estes compostos podem, por exemplo, serem usados no tratamento do tipo doença parasitária causada por helmintos, tais como Dirofilaria, em particular Dirofilaria immitis.
BR112022012130A 2019-12-18 2020-12-17 Compostos antelmínticos compreendendo uma estrutura azaindólica BR112022012130A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP19217671 2019-12-18
EP20213299 2020-12-11
PCT/EP2020/086660 WO2021122906A1 (en) 2019-12-18 2020-12-17 Anthelmintic compounds comprising azaindoles structure

Publications (1)

Publication Number Publication Date
BR112022012130A2 true BR112022012130A2 (pt) 2022-08-30

Family

ID=74106031

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112022012130A BR112022012130A2 (pt) 2019-12-18 2020-12-17 Compostos antelmínticos compreendendo uma estrutura azaindólica

Country Status (9)

Country Link
US (1) US20230110397A1 (pt)
EP (1) EP4077322A1 (pt)
JP (1) JP2023506303A (pt)
CN (1) CN114846014A (pt)
AU (1) AU2020404100A1 (pt)
BR (1) BR112022012130A2 (pt)
CA (1) CA3164104A1 (pt)
MX (1) MX2022007671A (pt)
WO (1) WO2021122906A1 (pt)

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JP2022526901A (ja) 2019-03-19 2022-05-27 ベーリンガー インゲルハイム アニマル ヘルス ユーエスエイ インコーポレイテッド 駆虫性アザベンゾチオフェンおよびアザベンゾフラン化合物
PE20231205A1 (es) 2020-05-29 2023-08-17 Boehringer Ingelheim Animal Health Usa Inc Compuestos heterociclicos como anthelminticos
AR127495A1 (es) 2021-11-01 2024-01-31 Boehringer Ingelheim Vetmedica Gmbh Compuestos de pirrolopiridazina como antihelmínticos
CN116969976A (zh) * 2022-04-28 2023-10-31 杭州普济远成生物医药科技有限公司 去泛素化酶抑制剂及其应用

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Also Published As

Publication number Publication date
WO2021122906A1 (en) 2021-06-24
CA3164104A1 (en) 2021-06-24
JP2023506303A (ja) 2023-02-15
US20230110397A1 (en) 2023-04-13
CN114846014A (zh) 2022-08-02
EP4077322A1 (en) 2022-10-26
AU2020404100A1 (en) 2022-06-09
MX2022007671A (es) 2022-07-19

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