BR112015021186A2 - processo para a preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octano - Google Patents
processo para a preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octanoInfo
- Publication number
- BR112015021186A2 BR112015021186A2 BR112015021186A BR112015021186A BR112015021186A2 BR 112015021186 A2 BR112015021186 A2 BR 112015021186A2 BR 112015021186 A BR112015021186 A BR 112015021186A BR 112015021186 A BR112015021186 A BR 112015021186A BR 112015021186 A2 BR112015021186 A2 BR 112015021186A2
- Authority
- BR
- Brazil
- Prior art keywords
- carbonyl
- sulfoxy
- diaza
- bicyclo
- pyrrolidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
resumo patente de invenção: "processo para a preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octano". é divulgado um processo para preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octano incluindo a reação de um composto de fórmula (ii) com um composto de fórmula (iii) para obter um composto de fórmula (iv). o produto final cristalino é conforme reivindicado.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN715MU2013 | 2013-03-08 | ||
PCT/IB2013/059327 WO2014135932A1 (en) | 2013-03-08 | 2013-10-12 | A process for preparation of (2s, 5r)-7-oxo-6-sulphooxy-2-[((3r)-pyrrolidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015021186A2 true BR112015021186A2 (pt) | 2017-07-18 |
Family
ID=54250567
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015021186A BR112015021186A2 (pt) | 2013-03-08 | 2013-10-12 | processo para a preparação de (2s,5r)-7-oxo-6-sulfóxi-2-[((3r)-pirrolidina-3-carbonil)-hidrazino carbonil]-1,6-diaza-biciclo[3.2.1]octano |
Country Status (13)
Country | Link |
---|---|
US (1) | US9624222B2 (pt) |
EP (1) | EP3013830A1 (pt) |
JP (2) | JP6285970B2 (pt) |
KR (1) | KR101774133B1 (pt) |
CN (1) | CN105008359B (pt) |
AU (1) | AU2013380575B2 (pt) |
BR (1) | BR112015021186A2 (pt) |
CA (1) | CA2904082C (pt) |
MX (1) | MX2015011721A (pt) |
NZ (1) | NZ711328A (pt) |
RU (1) | RU2625304C2 (pt) |
WO (1) | WO2014135932A1 (pt) |
ZA (1) | ZA201506342B (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI565707B (zh) * | 2012-05-30 | 2017-01-11 | 明治製菓藥業股份有限公司 | 新穎β-內醯胺酶抑制劑及其製造方法 |
NZ711329A (en) * | 2013-03-08 | 2016-06-24 | Wockhardt Ltd | A process for preparation of (2s, 5r)- sulfuric acid mono-{ [(4-aminopiperidin-4-yl) carbonyl]-7-oxo-1,6-diaza-bicyclo[3.2.1]-oct-6-yl} ester |
WO2014135930A1 (en) * | 2013-03-08 | 2014-09-12 | Wockhardt Limited | A process for sodium salt of (2s, 5r)-2-carboxamido-7-oxo-6-sulfooxy -1,6-diaza-bicyclo[3.2.1]octane |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2895630B2 (ja) * | 1993-12-29 | 1999-05-24 | フアイザー・インコーポレイテツド | ジアザビシクロニューロキニンアンタゴニスト |
ES2533826T3 (es) * | 2008-01-18 | 2015-04-15 | Merck Sharp & Dohme Corp. | Inhibidores de beta-lactamasa |
FR2951171A1 (fr) * | 2009-10-09 | 2011-04-15 | Novexel | Nouveau sel de sodium d'un compose azabicyclique sous forme enantiomere cristallisee et nouvelles formes polymorphes et pseudopolymorphes ainsi que leur preparation |
JP2011160817A (ja) * | 2010-02-04 | 2011-08-25 | Univ Of Tokyo | 移植支援材料 |
CA2822758C (en) | 2010-12-22 | 2018-03-20 | Meiji Seika Pharma Co., Ltd. | Optically active diazabicyclooctane derivative and process for preparing the same |
MX348974B (es) * | 2011-08-27 | 2017-07-04 | Wockhardt Ltd | Derivados 1,6 - diazabiciclo [3,2,1] octan-7-ona y su uso en el tratamiento de infecciones bacterianas. |
-
2013
- 2013-10-12 JP JP2015560792A patent/JP6285970B2/ja not_active Expired - Fee Related
- 2013-10-12 AU AU2013380575A patent/AU2013380575B2/en not_active Ceased
- 2013-10-12 WO PCT/IB2013/059327 patent/WO2014135932A1/en active Application Filing
- 2013-10-12 MX MX2015011721A patent/MX2015011721A/es unknown
- 2013-10-12 US US14/769,810 patent/US9624222B2/en not_active Expired - Fee Related
- 2013-10-12 CA CA2904082A patent/CA2904082C/en not_active Expired - Fee Related
- 2013-10-12 CN CN201380074308.4A patent/CN105008359B/zh not_active Expired - Fee Related
- 2013-10-12 NZ NZ711328A patent/NZ711328A/en not_active IP Right Cessation
- 2013-10-12 RU RU2015142483A patent/RU2625304C2/ru not_active IP Right Cessation
- 2013-10-12 KR KR1020157027179A patent/KR101774133B1/ko active IP Right Grant
- 2013-10-12 EP EP13812119.9A patent/EP3013830A1/en not_active Withdrawn
- 2013-10-12 BR BR112015021186A patent/BR112015021186A2/pt not_active Application Discontinuation
-
2015
- 2015-08-28 ZA ZA2015/06342A patent/ZA201506342B/en unknown
-
2017
- 2017-12-21 JP JP2017245132A patent/JP2018058895A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
KR101774133B1 (ko) | 2017-09-01 |
AU2013380575B2 (en) | 2016-07-07 |
CA2904082A1 (en) | 2014-09-12 |
NZ711328A (en) | 2016-06-24 |
EP3013830A1 (en) | 2016-05-04 |
JP6285970B2 (ja) | 2018-02-28 |
JP2016515102A (ja) | 2016-05-26 |
WO2014135932A1 (en) | 2014-09-12 |
KR20150123320A (ko) | 2015-11-03 |
MX2015011721A (es) | 2015-12-01 |
CN105008359A (zh) | 2015-10-28 |
CN105008359B (zh) | 2018-01-23 |
US9624222B2 (en) | 2017-04-18 |
CA2904082C (en) | 2017-10-03 |
US20160002234A1 (en) | 2016-01-07 |
ZA201506342B (en) | 2016-12-21 |
RU2625304C2 (ru) | 2017-07-13 |
JP2018058895A (ja) | 2018-04-12 |
RU2015142483A (ru) | 2017-04-13 |
AU2013380575A1 (en) | 2015-09-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according art. 34 industrial property law | ||
B06F | Objections, documents and/or translations needed after an examination request according art. 34 industrial property law | ||
B06I | Technical and formal requirements: publication cancelled |
Free format text: ANULADA A PUBLICACAO CODIGO 6.6.1 NA RPI NO 2462 DE 13/03/2018 POR TER SIDO INDEVIDA. |
|
B07E | Notice of approval relating to section 229 industrial property law | ||
B06U | Preliminary requirement: requests with searches performed by other patent offices: suspension of the patent application procedure | ||
B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |