BR112015015250A2 - derivados de pirrolidina, composições farmacêuticas e usos dos mesmos - Google Patents
derivados de pirrolidina, composições farmacêuticas e usos dos mesmosInfo
- Publication number
- BR112015015250A2 BR112015015250A2 BR112015015250A BR112015015250A BR112015015250A2 BR 112015015250 A2 BR112015015250 A2 BR 112015015250A2 BR 112015015250 A BR112015015250 A BR 112015015250A BR 112015015250 A BR112015015250 A BR 112015015250A BR 112015015250 A2 BR112015015250 A2 BR 112015015250A2
- Authority
- BR
- Brazil
- Prior art keywords
- pharmaceutical compositions
- pyrrolidine derivatives
- derivatives
- pyrrolidine
- medicaments
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Abstract
resumo patente de invenção: "derivados de pirrolidina, composições farmacêuticas e usos dos mesmos". a presente invenção refere-se a novos derivados de pirrolidina da fórmula (i), , a seu uso como medicamentos, a métodos para seu uso terapêutico e a composições farmacêuticas que os contêm.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP13152734 | 2013-01-25 | ||
PCT/EP2014/050981 WO2014114578A1 (en) | 2013-01-25 | 2014-01-20 | Pyrrolidine derivatives, pharmaceutical compositions and uses thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015015250A2 true BR112015015250A2 (pt) | 2017-07-11 |
Family
ID=47630189
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015015250A BR112015015250A2 (pt) | 2013-01-25 | 2014-01-20 | derivados de pirrolidina, composições farmacêuticas e usos dos mesmos |
Country Status (7)
Country | Link |
---|---|
US (1) | US8877741B2 (pt) |
EP (1) | EP2948442B1 (pt) |
JP (1) | JP6047825B2 (pt) |
AU (1) | AU2014210013A1 (pt) |
BR (1) | BR112015015250A2 (pt) |
IL (1) | IL238851A0 (pt) |
WO (1) | WO2014114578A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10150728B2 (en) | 2013-10-17 | 2018-12-11 | Shionogi & Co., Ltd. | Alkylene derivatives |
WO2016201662A1 (en) * | 2015-06-18 | 2016-12-22 | Eli Lilly And Company | Fluoropyridyl pyrazol compounds |
WO2018095344A1 (en) * | 2016-11-24 | 2018-05-31 | Shanghai Meton Pharmaceutical Co., Ltd | Isocitrate dehydrogenase (idh) inhibitor |
US20220055992A1 (en) | 2018-12-21 | 2022-02-24 | Saltigo Gmbh | Process for preparing 2-alkoxy-4-amino-5-methyl-pyridines and/or 2-alkoxy-4-alkylamino-5-methyl-pyridines |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1997028128A1 (en) | 1996-02-02 | 1997-08-07 | Zeneca Limited | Heterocyclic compounds useful as pharmaceutical agents |
BRPI0907584A2 (pt) * | 2008-02-22 | 2015-07-21 | Irm Llc | Composto e composições como moduladores de atividade de gpr119 |
WO2012090219A2 (en) * | 2010-12-31 | 2012-07-05 | Jubilant Biosys Ltd. | Thiazole compounds useful as acetyl-coa carboxylase (acc) inhibitors |
US8530460B2 (en) * | 2011-12-19 | 2013-09-10 | Boehringer Ingelheim International Gmbh | Azetidine derivatives |
-
2014
- 2014-01-20 BR BR112015015250A patent/BR112015015250A2/pt not_active IP Right Cessation
- 2014-01-20 JP JP2015554114A patent/JP6047825B2/ja active Active
- 2014-01-20 EP EP14701328.8A patent/EP2948442B1/en active Active
- 2014-01-20 AU AU2014210013A patent/AU2014210013A1/en not_active Abandoned
- 2014-01-20 WO PCT/EP2014/050981 patent/WO2014114578A1/en active Application Filing
- 2014-01-22 US US14/161,256 patent/US8877741B2/en active Active
-
2015
- 2015-05-17 IL IL238851A patent/IL238851A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
US8877741B2 (en) | 2014-11-04 |
EP2948442A1 (en) | 2015-12-02 |
EP2948442B1 (en) | 2016-10-26 |
JP2016509598A (ja) | 2016-03-31 |
JP6047825B2 (ja) | 2016-12-21 |
WO2014114578A1 (en) | 2014-07-31 |
US20140213568A1 (en) | 2014-07-31 |
IL238851A0 (en) | 2015-06-30 |
AU2014210013A1 (en) | 2015-06-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |