BR112014024064B8 - Métodos para preparação de 3-substituída-6-triflúormetil piridinas e para formação de 3-halo-6-triflúormetil piridina - Google Patents
Métodos para preparação de 3-substituída-6-triflúormetil piridinas e para formação de 3-halo-6-triflúormetil piridinaInfo
- Publication number
- BR112014024064B8 BR112014024064B8 BR112014024064A BR112014024064A BR112014024064B8 BR 112014024064 B8 BR112014024064 B8 BR 112014024064B8 BR 112014024064 A BR112014024064 A BR 112014024064A BR 112014024064 A BR112014024064 A BR 112014024064A BR 112014024064 B8 BR112014024064 B8 BR 112014024064B8
- Authority
- BR
- Brazil
- Prior art keywords
- pyridine
- substituted
- trifluormethyl
- methods
- formation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/26—Radicals substituted by halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
Abstract
MÉTODOS PARA PREPARAR 6-TRIFLUOROMETIL-3-PIRIDINAS SUBSTITUÍDAS E MÉTODOS PARA USAR 6-TRICLOROMETIL PIRIDINAS HALOGENADAS. A presente invenção refere-se às 6-trifluorometil-3-piridinas substituídas são intermediários sintéticos úteis na preparação de N-(6- haloalquilpiridinil-3) alquil sulfoximinas substituídas, que são úteis na formação de inseticidas potentes. Os métodos para formar tais 6-trifluorometil-3-piridinas substituídas são aqui divulgados. Também são divulgados métodos usando a 6-triclorometil piridina halogenada para formar as 6-trifluorometil-3-piridinas substituídas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261618370P | 2012-03-30 | 2012-03-30 | |
PCT/US2013/032270 WO2013148338A1 (en) | 2012-03-30 | 2013-03-15 | Methods for preparing 3-substituted-6-trifluoromethyl pyridines and methods for using 6-trichloromethyl halogenated pyridines |
Publications (2)
Publication Number | Publication Date |
---|---|
BR112014024064B1 BR112014024064B1 (pt) | 2020-01-14 |
BR112014024064B8 true BR112014024064B8 (pt) | 2022-10-11 |
Family
ID=49235880
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014024064A BR112014024064B8 (pt) | 2012-03-30 | 2013-03-15 | Métodos para preparação de 3-substituída-6-triflúormetil piridinas e para formação de 3-halo-6-triflúormetil piridina |
Country Status (14)
Country | Link |
---|---|
US (1) | US8785650B2 (pt) |
EP (1) | EP2831044B1 (pt) |
JP (1) | JP6219922B2 (pt) |
KR (1) | KR20140145176A (pt) |
CN (1) | CN104321310B (pt) |
AR (1) | AR093745A1 (pt) |
BR (1) | BR112014024064B8 (pt) |
CA (1) | CA2867155C (pt) |
CO (1) | CO7180217A2 (pt) |
ES (1) | ES2848700T3 (pt) |
IL (1) | IL234820A (pt) |
IN (1) | IN2014DN08373A (pt) |
MX (1) | MX354136B (pt) |
WO (1) | WO2013148338A1 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN105541698B (zh) * | 2015-12-23 | 2018-07-10 | 滨海康杰化学有限公司 | 一种5-溴-2-三氟甲基吡啶的制备方法 |
CN105820112A (zh) * | 2016-06-06 | 2016-08-03 | 山东福尔有限公司 | 一种2-氯-5-三氟甲基吡啶的制备方法 |
EP3694322B1 (en) | 2017-10-09 | 2024-07-03 | Terumo BCT Biotechnologies, LLC | Lyophilization container and method of using same |
WO2020185916A1 (en) | 2019-03-14 | 2020-09-17 | Terumo Bct Biotechnologies, Llc | Lyophilization container fill fixture, system and method of use |
CN115282879B (zh) * | 2022-08-08 | 2024-04-05 | 单县欣润化工有限公司 | 2-氯-5-三氟甲基吡啶合成的原料供应***及工艺 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2516402A (en) * | 1945-09-04 | 1950-07-25 | Purdue Research Foundation | Fluoromethylpyridines |
US4127575A (en) * | 1976-10-20 | 1978-11-28 | The Dow Chemical Company | Preparation of chloro substituted pyridines |
GB2068365B (en) * | 1980-02-05 | 1983-12-14 | Dow Chemical Co | Fungicidal pyridyl arylureas |
US4567273A (en) * | 1982-04-16 | 1986-01-28 | The Dow Chemical Company | Liquid phase halogen exchange of (trichloromethyl) pyridines to (trifluoromethyl)pyridines |
US4480102A (en) * | 1982-07-23 | 1984-10-30 | The Dow Chemical Company | 2,3-Difluoro-5-(trifluoromethyl)pyridine and methods of making and using the same |
IL70307A (en) * | 1982-11-26 | 1987-02-27 | Dow Chemical Co | Preparation of(trifluoromethyl)pyridines |
US4590279A (en) * | 1982-11-26 | 1986-05-20 | The Dow Chemical Company | Preparation of (trifluoromethyl)pyridines under liquid phase conditions |
US5886210A (en) * | 1996-08-22 | 1999-03-23 | Rohm And Haas Company | Method for preparing aromatic compounds |
AU7286598A (en) * | 1997-05-09 | 1998-11-27 | Dow Agrosciences Llc | Preparation of 2,5-dichloro-(3-trifluoromethyl)pyridine |
WO1998051152A1 (fr) * | 1997-05-15 | 1998-11-19 | Sagami Chemical Research Center | Insecticides/acaricides |
SK15432003A3 (sk) * | 2001-05-22 | 2004-05-04 | Neurogen Corporation | 5-Substituované 2-arylpyridíny |
EP1729771B1 (en) * | 2004-03-22 | 2009-10-14 | Eli Lilly & Company | Pyridyl derivatives and their use as mglu5 receptor antagonists |
TW201309635A (zh) | 2006-02-10 | 2013-03-01 | Dow Agrosciences Llc | 殺蟲性之n-取代(6-鹵烷基吡啶-3-基)烷基磺醯亞胺(二) |
MX2011000196A (es) * | 2008-07-01 | 2011-03-24 | Dow Agrosciences Llc | Proceso mejorado para la preparacion de alquilpiridinas 2-trifluorometil-5-(1-sustituidas). |
CN102395564A (zh) * | 2009-04-17 | 2012-03-28 | 石原产业株式会社 | 2-卤代-6-取代-4-三氟甲基吡啶的生产方法 |
CN102093288B (zh) * | 2011-01-11 | 2012-08-29 | 衢州恒顺化工有限公司 | 一种水合三氯吡啶肼的制备方法 |
BR112013026137B1 (pt) * | 2011-04-19 | 2020-12-01 | Nerviano Medical Sciences S.R.L | pirimidinil-pirróis substituídos ativos como inibidores da quinase |
-
2013
- 2013-03-15 WO PCT/US2013/032270 patent/WO2013148338A1/en active Application Filing
- 2013-03-15 KR KR1020147030039A patent/KR20140145176A/ko not_active Application Discontinuation
- 2013-03-15 BR BR112014024064A patent/BR112014024064B8/pt active IP Right Grant
- 2013-03-15 JP JP2015503335A patent/JP6219922B2/ja active Active
- 2013-03-15 CA CA2867155A patent/CA2867155C/en active Active
- 2013-03-15 US US13/839,373 patent/US8785650B2/en active Active
- 2013-03-15 EP EP13767953.6A patent/EP2831044B1/en active Active
- 2013-03-15 ES ES13767953T patent/ES2848700T3/es active Active
- 2013-03-15 IN IN8373DEN2014 patent/IN2014DN08373A/en unknown
- 2013-03-15 MX MX2014011833A patent/MX354136B/es active IP Right Grant
- 2013-03-15 CN CN201380026384.8A patent/CN104321310B/zh active Active
- 2013-03-27 AR ARP130101041A patent/AR093745A1/es active IP Right Grant
-
2014
- 2014-09-23 IL IL234820A patent/IL234820A/en active IP Right Grant
- 2014-10-28 CO CO14237884A patent/CO7180217A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
AR093745A1 (es) | 2015-06-24 |
MX354136B (es) | 2018-02-14 |
MX2014011833A (es) | 2014-12-10 |
EP2831044A1 (en) | 2015-02-04 |
JP6219922B2 (ja) | 2017-10-25 |
IN2014DN08373A (pt) | 2015-05-08 |
CA2867155A1 (en) | 2013-10-03 |
IL234820A (en) | 2017-06-29 |
EP2831044B1 (en) | 2020-11-11 |
BR112014024064B1 (pt) | 2020-01-14 |
ES2848700T3 (es) | 2021-08-11 |
EP2831044A4 (en) | 2015-11-11 |
JP2015514711A (ja) | 2015-05-21 |
US8785650B2 (en) | 2014-07-22 |
CN104321310B (zh) | 2017-02-22 |
US20130261310A1 (en) | 2013-10-03 |
CN104321310A (zh) | 2015-01-28 |
CA2867155C (en) | 2021-06-08 |
KR20140145176A (ko) | 2014-12-22 |
WO2013148338A1 (en) | 2013-10-03 |
CO7180217A2 (es) | 2015-02-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 15/03/2013, OBSERVADAS AS CONDICOES LEGAIS. |
|
B25D | Requested change of name of applicant approved |
Owner name: CORTEVA AGRISCIENCE LLC (US) |