BR112014017902A2 - Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose - Google Patents
Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicoseInfo
- Publication number
- BR112014017902A2 BR112014017902A2 BR112014017902A BR112014017902A BR112014017902A2 BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2 BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2
- Authority
- BR
- Brazil
- Prior art keywords
- glucose metabolism
- therapeutic
- prophylactic agent
- disorders
- diseases caused
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
AGENTE TERAPÊUTICO OU PROFILÁTICO PARA DOENÇAS CAUSADAS POR DISTÚRBIOS DO METABOLISMO DE GLICOSE. O propósito da presente invenção é prover um novo agente terapêutico ou um novo agente profilático para doenças associadas com metabolismo anormal da glicose. A presente invenção é um agente terapêutico ou um agente profilático para doenças associadas com metabolismo anormal da glicose, que compreende um composto de 2-feniltiazol representado pela fórmula (I) ou um sal farmaceuticamente aceitável do mesmo como um ingrediente ativo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2012015351 | 2012-01-27 | ||
PCT/JP2013/051627 WO2013111870A1 (ja) | 2012-01-27 | 2013-01-25 | 糖尿病の治療薬 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112014017902A2 true BR112014017902A2 (pt) | 2017-08-22 |
Family
ID=48873581
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014017902A BR112014017902A2 (pt) | 2012-01-27 | 2013-01-25 | Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose |
Country Status (15)
Country | Link |
---|---|
US (1) | US20150005506A1 (pt) |
EP (1) | EP2808018B1 (pt) |
JP (1) | JP5924699B2 (pt) |
KR (1) | KR20140134266A (pt) |
CN (1) | CN104066430A (pt) |
AR (1) | AR089812A1 (pt) |
AU (1) | AU2013212865A1 (pt) |
BR (1) | BR112014017902A2 (pt) |
CA (1) | CA2862602A1 (pt) |
HK (1) | HK1201209A1 (pt) |
IN (1) | IN2014DN05972A (pt) |
MX (1) | MX2014008484A (pt) |
RU (1) | RU2014134845A (pt) |
TW (1) | TW201334779A (pt) |
WO (1) | WO2013111870A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104628671B (zh) * | 2015-02-10 | 2016-04-13 | 佛山市赛维斯医药科技有限公司 | 含苯基脒结构的硝基苯噻唑羧酸酰胺类化合物及用途 |
CN104610188B (zh) * | 2015-02-10 | 2016-07-27 | 佛山市赛维斯医药科技有限公司 | 含苯基脒结构的腈基苯噻唑羧酸酰胺类化合物、其制备及用途 |
CN104610190B (zh) * | 2015-02-10 | 2016-08-17 | 佛山市赛维斯医药科技有限公司 | 一类含环丙基脒结构的卤代苯基噻唑羧酸酰胺类化合物及用途 |
CN104628672A (zh) * | 2015-02-10 | 2015-05-20 | 佛山市赛维斯医药科技有限公司 | 一类含苯基脒结构的烷氧苯基噻唑羧酸酰胺类化合物及用途 |
CN104628673A (zh) * | 2015-02-10 | 2015-05-20 | 佛山市赛维斯医药科技有限公司 | 一类含叔丁基脒结构的腈基苯噻唑羧酸酰胺类化合物及用途 |
KR102473677B1 (ko) * | 2015-08-17 | 2022-12-02 | 삼성디스플레이 주식회사 | 액정 표시 장치 |
US11344539B2 (en) | 2016-02-19 | 2022-05-31 | National University Corporation Tottori University | Therapeutic or prophylactic drug for dementia |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100221041B1 (ko) * | 1990-11-30 | 1999-09-15 | 야스이 쇼사꾸 | 2-아릴티아졸 유도체 및 그의 약제학적 조성물 |
HUP9902721A2 (hu) * | 1997-11-25 | 1999-12-28 | The Procter & Gamble Co. | Tömény textillágyító készítmény és ehhez alkalmazható magas telítetlenségű textillágyító vegyület |
US20050074442A1 (en) * | 2002-03-13 | 2005-04-07 | Natarajan Ranganathan | Compositions and methods for augmenting kidney function |
WO2006012438A2 (en) * | 2004-07-21 | 2006-02-02 | University Of Florida Research Foundation, Inc. | Compositions and methods for treatment and prevention of insulin resistance |
JP2009501795A (ja) * | 2005-07-21 | 2009-01-22 | ユニバーシティ オブ フロリダ リサーチファウンデーション インコーポレイティッド | 高尿酸血に関連する健康状態の治療及び予防のための組成物及び方法 |
CA2617248C (en) | 2005-08-03 | 2015-09-29 | Tap Pharmaceutical Products, Inc. | Methods for treating hypertension |
CA2630639A1 (en) * | 2005-11-21 | 2007-05-31 | Tap Pharmaceutical Products, Inc. | Treatment of qt interval prolongation and diseases associated therewith |
JP2007210978A (ja) | 2006-02-13 | 2007-08-23 | Hiroshima Univ | 耐糖能障害、ii型糖尿病、高脂血症、メタボリックシンドローム、内臓脂肪型肥満、脂肪肝または非アルコール性脂肪性肝炎の予防・治療剤 |
KR20160031040A (ko) | 2006-11-13 | 2016-03-21 | 다케다 파마슈티칼스 유에스에이, 인코포레이티드 | 크산틴 옥시도리덕타아제 억제제를 사용하여 신장 기능을 보존하는 방법 |
US8084483B2 (en) * | 2007-11-27 | 2011-12-27 | Ardea Biosciences, Inc. | Compounds and compositions and methods of use |
DK2266989T3 (en) * | 2008-03-31 | 2015-11-23 | C&C Res Lab | Heterocyclic derivatives |
EP2282736B1 (en) * | 2008-04-30 | 2015-11-11 | Wellstat Therapeutics Corporation | Tetrazole compounds for reducing uric acid |
EP2668953A1 (en) * | 2008-05-22 | 2013-12-04 | Bristol-Myers Squibb Company | Pharmaceutical compositions comprising an SGLT2 inhibitor with a supply of carbohydrate and/or an inhibitor of uric acid synthesis |
CN102256488A (zh) * | 2008-10-19 | 2011-11-23 | 理查德·J·约翰逊 | 伴随代谢失衡慢性肾病的治疗组合物和治疗方法 |
US20120219536A1 (en) * | 2009-08-24 | 2012-08-30 | Queensland University Of Technology | Purine-targeted diagnosis and therapy of wounds |
WO2011159745A1 (en) * | 2010-06-16 | 2011-12-22 | Takeda Pharmaceuticals North America, Inc. | Novel modified release dosage forms of xanthine oxidoreductase inhibitor or xanthine oxidase inhibitors |
JPWO2011162390A1 (ja) * | 2010-06-25 | 2013-08-22 | 帝人ファーマ株式会社 | 徐放性高血圧および腎機能障害治療剤 |
-
2013
- 2013-01-25 KR KR1020147020342A patent/KR20140134266A/ko not_active Application Discontinuation
- 2013-01-25 JP JP2013555326A patent/JP5924699B2/ja not_active Expired - Fee Related
- 2013-01-25 US US14/372,961 patent/US20150005506A1/en not_active Abandoned
- 2013-01-25 TW TW102102886A patent/TW201334779A/zh unknown
- 2013-01-25 BR BR112014017902A patent/BR112014017902A2/pt not_active IP Right Cessation
- 2013-01-25 CN CN201380006730.6A patent/CN104066430A/zh active Pending
- 2013-01-25 MX MX2014008484A patent/MX2014008484A/es unknown
- 2013-01-25 IN IN5972DEN2014 patent/IN2014DN05972A/en unknown
- 2013-01-25 RU RU2014134845A patent/RU2014134845A/ru not_active Application Discontinuation
- 2013-01-25 AR ARP130100233A patent/AR089812A1/es unknown
- 2013-01-25 AU AU2013212865A patent/AU2013212865A1/en not_active Abandoned
- 2013-01-25 WO PCT/JP2013/051627 patent/WO2013111870A1/ja active Application Filing
- 2013-01-25 EP EP13740913.2A patent/EP2808018B1/en not_active Not-in-force
- 2013-01-25 CA CA2862602A patent/CA2862602A1/en not_active Abandoned
-
2015
- 2015-02-25 HK HK15101890.2A patent/HK1201209A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
JP5924699B2 (ja) | 2016-05-25 |
AR089812A1 (es) | 2014-09-17 |
EP2808018A4 (en) | 2015-07-15 |
WO2013111870A1 (ja) | 2013-08-01 |
IN2014DN05972A (pt) | 2015-06-26 |
EP2808018B1 (en) | 2018-03-14 |
EP2808018A1 (en) | 2014-12-03 |
CN104066430A (zh) | 2014-09-24 |
KR20140134266A (ko) | 2014-11-21 |
MX2014008484A (es) | 2014-10-14 |
CA2862602A1 (en) | 2013-08-01 |
US20150005506A1 (en) | 2015-01-01 |
RU2014134845A (ru) | 2016-03-20 |
JPWO2013111870A1 (ja) | 2015-05-11 |
TW201334779A (zh) | 2013-09-01 |
AU2013212865A1 (en) | 2014-08-14 |
HK1201209A1 (en) | 2015-08-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |