BR0009277A - Processo de preparação de ácido propiÈnico de 3s-3-amino-3-arila e derivados deste - Google Patents

Processo de preparação de ácido propiÈnico de 3s-3-amino-3-arila e derivados deste

Info

Publication number
BR0009277A
BR0009277A BR0009277-0A BR0009277A BR0009277A BR 0009277 A BR0009277 A BR 0009277A BR 0009277 A BR0009277 A BR 0009277A BR 0009277 A BR0009277 A BR 0009277A
Authority
BR
Brazil
Prior art keywords
derivatives
amino
propionic acid
preparation process
aryl propionic
Prior art date
Application number
BR0009277-0A
Other languages
English (en)
Inventor
Lorraine Scott
Frank John Villani Jr
Donald G Walker
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of BR0009277A publication Critical patent/BR0009277A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/55—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom

Abstract

Patente de Invenção: "PROCESSO DE PREPARAçãO DE áCIDO PROPIÈNICO DE 3S-3-AMINO-3-ARILA E DERIVADOS DESTE". A presente invenção é direcionada para um processo para preparação de ácido propiónico de 3S-3-amino-3-arila e derivados destes.
BR0009277-0A 1999-03-22 2000-03-21 Processo de preparação de ácido propiÈnico de 3s-3-amino-3-arila e derivados deste BR0009277A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12622799P 1999-03-22 1999-03-22
PCT/US2000/007492 WO2000056715A1 (en) 1999-03-22 2000-03-21 Process of preparing 3s-3-amino-3-aryl propionic acid and derivatives thereof

Publications (1)

Publication Number Publication Date
BR0009277A true BR0009277A (pt) 2002-02-05

Family

ID=22423697

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0009277-0A BR0009277A (pt) 1999-03-22 2000-03-21 Processo de preparação de ácido propiÈnico de 3s-3-amino-3-arila e derivados deste

Country Status (17)

Country Link
US (3) US6673926B2 (pt)
EP (1) EP1163222A1 (pt)
JP (1) JP2002540100A (pt)
KR (1) KR20020016617A (pt)
CN (1) CN1362948A (pt)
AU (1) AU3906300A (pt)
BR (1) BR0009277A (pt)
CA (1) CA2367969A1 (pt)
CZ (1) CZ20013403A3 (pt)
HR (1) HRP20010766A2 (pt)
HU (1) HUP0201347A3 (pt)
MX (1) MXPA01009621A (pt)
NZ (1) NZ514383A (pt)
RU (1) RU2228929C2 (pt)
SK (1) SK13582001A3 (pt)
WO (1) WO2000056715A1 (pt)
YU (1) YU74401A (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6306909B1 (en) 1997-03-12 2001-10-23 Queen's University At Kingston Anti-epileptogenic agents
HUP0201263A3 (en) 1999-03-22 2003-05-28 Ortho Mcneil Pharm Inc Synthesis of 3-amino-3-aryl propanoates and intermediates
YU74401A (sh) * 1999-03-22 2004-07-15 Ortho-Mcneil Pharmaaceutical Postupak za dobijanje 2s-3-amino-3-arilpropionske kiseline i njenih derivata
EP1397136A1 (en) * 2001-05-25 2004-03-17 Queen's University At Kingston Heterocyclic beta-aminoacids and their use as anti-epileptogenic agents
CN101982458B (zh) * 2010-09-14 2013-11-06 北京欧凯纳斯科技有限公司 3-氨基-3-芳基丙酸及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE58243B1 (en) 1983-12-07 1993-08-11 Lonza Ag A process for the preparation of optically-active 3-amino carboxylic acids
US5254573A (en) 1991-10-15 1993-10-19 Monsanto Company Substituted heterocyclic derivatives useful as platelet aggregation inhibitors
JP4328387B2 (ja) * 1996-05-01 2009-09-09 オーソ―マクニール・フアーマシユーチカル・インコーポレーテツド 血栓形成疾患の処置のためのピロリジン、ピペリジン及びヘキサヒドロアゼピンのカルボキサミド誘導体
EP0912495B1 (en) 1996-07-12 2001-11-21 G.D. SEARLE & CO. Asymetric synthesis of chiral beta-amino acids
YU74401A (sh) * 1999-03-22 2004-07-15 Ortho-Mcneil Pharmaaceutical Postupak za dobijanje 2s-3-amino-3-arilpropionske kiseline i njenih derivata
DE10111877A1 (de) * 2001-03-10 2002-09-12 Aventis Pharma Gmbh Neue Imidazolidinderivate, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate

Also Published As

Publication number Publication date
MXPA01009621A (es) 2003-07-21
KR20020016617A (ko) 2002-03-04
US20030176471A1 (en) 2003-09-18
HUP0201347A3 (en) 2002-12-28
CZ20013403A3 (cs) 2002-07-17
AU3906300A (en) 2000-10-09
NZ514383A (en) 2004-01-30
US20020068829A1 (en) 2002-06-06
WO2000056715A1 (en) 2000-09-28
RU2228929C2 (ru) 2004-05-20
YU74401A (sh) 2004-07-15
US6673926B2 (en) 2004-01-06
CA2367969A1 (en) 2000-09-28
US20040063960A1 (en) 2004-04-01
HUP0201347A2 (en) 2002-09-28
CN1362948A (zh) 2002-08-07
HRP20010766A2 (en) 2002-12-31
SK13582001A3 (sk) 2003-02-04
JP2002540100A (ja) 2002-11-26
EP1163222A1 (en) 2001-12-19

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Free format text: JOHNSON & JOHNSON INDUSTRIAL LTDA. (BR/SP)

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O E 13 DA LPI

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.