BG97014A - Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им - Google Patents

Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им

Info

Publication number
BG97014A
BG97014A BG097014A BG9701492A BG97014A BG 97014 A BG97014 A BG 97014A BG 097014 A BG097014 A BG 097014A BG 9701492 A BG9701492 A BG 9701492A BG 97014 A BG97014 A BG 97014A
Authority
BG
Bulgaria
Prior art keywords
preparation
application
benzothiazepinone
derivatives
benzothiazepinone derivatives
Prior art date
Application number
BG097014A
Other languages
English (en)
Inventor
Aldo Salimbeni
Elso Manghisi
Saturnino Caliari
Francesco Fici
Original Assignee
Istituto Luso Farmaco D'italia S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Istituto Luso Farmaco D'italia S.P.A. filed Critical Istituto Luso Farmaco D'italia S.P.A.
Publication of BG97014A publication Critical patent/BG97014A/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/12Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
BG097014A 1990-04-27 1992-10-22 Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им BG97014A (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT20160A IT1240686B (it) 1990-04-27 1990-04-27 Derivati 1,5-benzotiazepinonici, loro preparazione e uso farmaceutico
PCT/EP1991/000742 WO1991017153A1 (en) 1990-04-27 1991-04-18 1,5-benzothiazepinone derivatives, their preparations and pharmaceutical use

Publications (1)

Publication Number Publication Date
BG97014A true BG97014A (bg) 1993-12-24

Family

ID=11164306

Family Applications (1)

Application Number Title Priority Date Filing Date
BG097014A BG97014A (bg) 1990-04-27 1992-10-22 Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им

Country Status (20)

Country Link
US (1) US5571807A (bg)
EP (1) EP0526495A1 (bg)
JP (1) JPH05506654A (bg)
CN (1) CN1056101A (bg)
AU (1) AU645317B2 (bg)
BG (1) BG97014A (bg)
BR (1) BR9106372A (bg)
CA (1) CA2081204A1 (bg)
CS (1) CS120991A2 (bg)
FI (1) FI924756A0 (bg)
HU (1) HU9203326D0 (bg)
IE (1) IE71033B1 (bg)
IL (1) IL97859A0 (bg)
IN (1) IN172160B (bg)
IT (1) IT1240686B (bg)
MA (1) MA22143A1 (bg)
PT (1) PT97508A (bg)
RO (1) RO111269B1 (bg)
WO (1) WO1991017153A1 (bg)
ZA (1) ZA913171B (bg)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0702009T3 (da) * 1994-09-16 1999-02-01 Orion Corp Fermion Fremgangsmåde til fremstilling af farmaceutisk aktive benzothiazepinderivater
US5559229A (en) * 1995-06-01 1996-09-24 Acic (Canada) Inc. Method for the manufacture of benzothiazepine
WO1996038429A1 (en) * 1995-06-01 1996-12-05 Acic (Canada) Inc. Method for the manufacture of benzothiazepine derivatives
WO2006079077A2 (en) * 2005-01-20 2006-07-27 Acadia Pharmaceuticals Inc. Use of diltiazem or analogs thereof as modulators of ghrelin receptor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3562257A (en) * 1967-10-28 1971-02-09 Tanabe Seiyaku Co Benzothiazepine derivatives
IT1206505B (it) * 1983-07-22 1989-04-27 Schiapparelli Farma Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono.
EP0256888B1 (en) * 1986-08-20 1991-07-03 McNeilab, Inc. Benzothiazepine vasodilators having aralkyl substitution
US4902684A (en) * 1988-06-20 1990-02-20 E. R. Squibb & Sons, Inc. Benzazepine and benzothiazepine derivatives
US4902687A (en) * 1989-03-27 1990-02-20 Eli Lilly And Company Excitatory amino acid receptor antagonists
ES2069003T3 (es) * 1989-04-28 1995-05-01 Tanabe Seiyaku Co Procedimiento para preparar derivados de 1,5-benzotiazepina.
JPH085869B2 (ja) * 1990-03-08 1996-01-24 田辺製薬株式会社 1,5−ベンゾチアゼピン誘導体の製法

Also Published As

Publication number Publication date
MA22143A1 (fr) 1991-12-31
FI924756A (fi) 1992-10-20
IT9020160A0 (it) 1990-04-27
EP0526495A1 (en) 1993-02-10
IE71033B1 (en) 1997-01-15
RO111269B1 (ro) 1996-08-30
IT1240686B (it) 1993-12-17
BR9106372A (pt) 1993-04-27
AU645317B2 (en) 1994-01-13
FI924756A0 (fi) 1992-10-20
PT97508A (pt) 1992-01-31
CN1056101A (zh) 1991-11-13
CA2081204A1 (en) 1991-10-28
IE911411A1 (en) 1991-11-06
JPH05506654A (ja) 1993-09-30
ZA913171B (en) 1992-02-26
HU9203326D0 (en) 1993-01-28
IN172160B (bg) 1993-04-17
IT9020160A1 (it) 1991-10-27
WO1991017153A1 (en) 1991-11-14
CS120991A2 (en) 1991-12-17
US5571807A (en) 1996-11-05
AU7695491A (en) 1991-11-27
IL97859A0 (en) 1992-06-21

Similar Documents

Publication Publication Date Title
BG97198A (bg) Диалкокси-пиридинил-бензимидазолови производни, метод за получаването им и тяхното фармацевтично приложение
TR25002A (tr) Kristalik natrinyumsilikatlarin hazirlanis yöntemi
BG97200A (bg) Заместени бензимидазоли,метод за получаването им и тяхното фармацевтично приложение
DE69009315D1 (de) Cinnamamidderivate.
DE69125099D1 (de) Indolderivate
ATE144765T1 (de) Hiv-hemmende benzenacetamidderivate
NO913745L (no) Fremgangsmaate for fremstilling av 1,3-benzoksazinderivater
DE69130255T2 (de) Oxadolderivate
DK0472733T3 (da) Phenantrenderivater
FI95036B (fi) Tieno-triatsolo-diatsepiinijohdosten valmistusmenetelmä
KR900701751A (ko) 치환 알릴아민 유도체, 그의 제조방법 및 그의 용도
FI894546A (fi) Menetelmä uusien 2'-halogeenimetylideeni-, 2'-etenylideeni- ja 2'-etynyyliadenosiinijohdannaisten valmistamiseksi
MX9101516A (es) Derivados de 1,2,5,6-tetrahidropiridin 3-cetoxima y-3-aldoxina y procedimiento para su preparacion
KR900700477A (ko) 3'- 아지도-3'- 디옥시디미딘 및 유사화합물을 합성하기 위한 방법
EE03027B1 (et) Meetod 8-klorokinolooni derivaatide valmistamiseks
DE69122555D1 (de) 2,4-Dihydroxyadipinsäurederivate
BG92749A (bg) Производни на аминопропанола,метод за тяхното получаване и фармацетични състави,съдържащи тези производни
BG97014A (bg) Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им
BG95668A (bg) Трет-бутилоксикарбонил-l-тирозил- пептидогликанов мономер, 125 горе i - белязано негово производно и метод за получаването му
MC2108A1 (fr) Derives de quinoleine
FI943833A0 (fi) Menetelmä 2,3,5,6-tetraklooripyridiinin valmistamiseksi
FI891111A (fi) Menetelmä 1,4-dihydropyridiinijohdannaisten valmistamiseksi
BG90160A (bg) Метод за получаване на 4'-деметилепиподофилотоксин- глюкозиди
FI904673A0 (fi) 2,6-dioksopiperidiinijohdannaisten valmistus
FR2602233B1 (fr) Derives de l'isoquinoleine