BG97014A - Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им - Google Patents
Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението имInfo
- Publication number
- BG97014A BG97014A BG097014A BG9701492A BG97014A BG 97014 A BG97014 A BG 97014A BG 097014 A BG097014 A BG 097014A BG 9701492 A BG9701492 A BG 9701492A BG 97014 A BG97014 A BG 97014A
- Authority
- BG
- Bulgaria
- Prior art keywords
- preparation
- application
- benzothiazepinone
- derivatives
- benzothiazepinone derivatives
- Prior art date
Links
- IENUYWJQEOAHFA-UHFFFAOYSA-N 1$l^{4},5-benzothiazepine 1-oxide Chemical class O=S1C=CC=NC2=CC=CC=C12 IENUYWJQEOAHFA-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
- A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT20160A IT1240686B (it) | 1990-04-27 | 1990-04-27 | Derivati 1,5-benzotiazepinonici, loro preparazione e uso farmaceutico |
PCT/EP1991/000742 WO1991017153A1 (en) | 1990-04-27 | 1991-04-18 | 1,5-benzothiazepinone derivatives, their preparations and pharmaceutical use |
Publications (1)
Publication Number | Publication Date |
---|---|
BG97014A true BG97014A (bg) | 1993-12-24 |
Family
ID=11164306
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG097014A BG97014A (bg) | 1990-04-27 | 1992-10-22 | Производни на 1,5-бензотиазепинон,метод за тяхното получаване и приложението им |
Country Status (20)
Country | Link |
---|---|
US (1) | US5571807A (bg) |
EP (1) | EP0526495A1 (bg) |
JP (1) | JPH05506654A (bg) |
CN (1) | CN1056101A (bg) |
AU (1) | AU645317B2 (bg) |
BG (1) | BG97014A (bg) |
BR (1) | BR9106372A (bg) |
CA (1) | CA2081204A1 (bg) |
CS (1) | CS120991A2 (bg) |
FI (1) | FI924756A0 (bg) |
HU (1) | HU9203326D0 (bg) |
IE (1) | IE71033B1 (bg) |
IL (1) | IL97859A0 (bg) |
IN (1) | IN172160B (bg) |
IT (1) | IT1240686B (bg) |
MA (1) | MA22143A1 (bg) |
PT (1) | PT97508A (bg) |
RO (1) | RO111269B1 (bg) |
WO (1) | WO1991017153A1 (bg) |
ZA (1) | ZA913171B (bg) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0702009T3 (da) * | 1994-09-16 | 1999-02-01 | Orion Corp Fermion | Fremgangsmåde til fremstilling af farmaceutisk aktive benzothiazepinderivater |
US5559229A (en) * | 1995-06-01 | 1996-09-24 | Acic (Canada) Inc. | Method for the manufacture of benzothiazepine |
WO1996038429A1 (en) * | 1995-06-01 | 1996-12-05 | Acic (Canada) Inc. | Method for the manufacture of benzothiazepine derivatives |
WO2006079077A2 (en) * | 2005-01-20 | 2006-07-27 | Acadia Pharmaceuticals Inc. | Use of diltiazem or analogs thereof as modulators of ghrelin receptor |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3562257A (en) * | 1967-10-28 | 1971-02-09 | Tanabe Seiyaku Co | Benzothiazepine derivatives |
IT1206505B (it) * | 1983-07-22 | 1989-04-27 | Schiapparelli Farma | Nuovi derivati benzotiazepinonici, metodo per la loro preparazione e composizioni farmaceutiche che licontengono. |
EP0256888B1 (en) * | 1986-08-20 | 1991-07-03 | McNeilab, Inc. | Benzothiazepine vasodilators having aralkyl substitution |
US4902684A (en) * | 1988-06-20 | 1990-02-20 | E. R. Squibb & Sons, Inc. | Benzazepine and benzothiazepine derivatives |
US4902687A (en) * | 1989-03-27 | 1990-02-20 | Eli Lilly And Company | Excitatory amino acid receptor antagonists |
ES2069003T3 (es) * | 1989-04-28 | 1995-05-01 | Tanabe Seiyaku Co | Procedimiento para preparar derivados de 1,5-benzotiazepina. |
JPH085869B2 (ja) * | 1990-03-08 | 1996-01-24 | 田辺製薬株式会社 | 1,5−ベンゾチアゼピン誘導体の製法 |
-
1990
- 1990-04-27 IT IT20160A patent/IT1240686B/it active IP Right Grant
-
1991
- 1991-04-15 IN IN296/MAS/91A patent/IN172160B/en unknown
- 1991-04-16 IL IL97859A patent/IL97859A0/xx unknown
- 1991-04-18 AU AU76954/91A patent/AU645317B2/en not_active Expired - Fee Related
- 1991-04-18 HU HU923326A patent/HU9203326D0/hu unknown
- 1991-04-18 EP EP91907834A patent/EP0526495A1/en not_active Withdrawn
- 1991-04-18 JP JP91507700A patent/JPH05506654A/ja active Pending
- 1991-04-18 BR BR919106372A patent/BR9106372A/pt not_active Application Discontinuation
- 1991-04-18 WO PCT/EP1991/000742 patent/WO1991017153A1/en not_active Application Discontinuation
- 1991-04-18 CA CA002081204A patent/CA2081204A1/en not_active Abandoned
- 1991-04-18 RO RO92-01339A patent/RO111269B1/ro unknown
- 1991-04-26 MA MA22413A patent/MA22143A1/fr unknown
- 1991-04-26 CS CS911209A patent/CS120991A2/cs unknown
- 1991-04-26 ZA ZA913171A patent/ZA913171B/xx unknown
- 1991-04-26 PT PT97508A patent/PT97508A/pt not_active Application Discontinuation
- 1991-04-26 IE IE141191A patent/IE71033B1/en not_active IP Right Cessation
- 1991-04-27 CN CN91102741A patent/CN1056101A/zh active Pending
-
1992
- 1992-10-20 FI FI924756A patent/FI924756A0/fi not_active Application Discontinuation
- 1992-10-22 BG BG097014A patent/BG97014A/bg unknown
-
1995
- 1995-03-31 US US08/397,904 patent/US5571807A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
MA22143A1 (fr) | 1991-12-31 |
FI924756A (fi) | 1992-10-20 |
IT9020160A0 (it) | 1990-04-27 |
EP0526495A1 (en) | 1993-02-10 |
IE71033B1 (en) | 1997-01-15 |
RO111269B1 (ro) | 1996-08-30 |
IT1240686B (it) | 1993-12-17 |
BR9106372A (pt) | 1993-04-27 |
AU645317B2 (en) | 1994-01-13 |
FI924756A0 (fi) | 1992-10-20 |
PT97508A (pt) | 1992-01-31 |
CN1056101A (zh) | 1991-11-13 |
CA2081204A1 (en) | 1991-10-28 |
IE911411A1 (en) | 1991-11-06 |
JPH05506654A (ja) | 1993-09-30 |
ZA913171B (en) | 1992-02-26 |
HU9203326D0 (en) | 1993-01-28 |
IN172160B (bg) | 1993-04-17 |
IT9020160A1 (it) | 1991-10-27 |
WO1991017153A1 (en) | 1991-11-14 |
CS120991A2 (en) | 1991-12-17 |
US5571807A (en) | 1996-11-05 |
AU7695491A (en) | 1991-11-27 |
IL97859A0 (en) | 1992-06-21 |
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