BG106868A - Pyrimidine carboxamides useful as inhibitors of pde4 isozymes - Google Patents

Pyrimidine carboxamides useful as inhibitors of pde4 isozymes

Info

Publication number
BG106868A
BG106868A BG106868A BG10686802A BG106868A BG 106868 A BG106868 A BG 106868A BG 106868 A BG106868 A BG 106868A BG 10686802 A BG10686802 A BG 10686802A BG 106868 A BG106868 A BG 106868A
Authority
BG
Bulgaria
Prior art keywords
inhibitors
chronic
pde4 isozymes
carboxamides useful
pyrimidine carboxamides
Prior art date
Application number
BG106868A
Other languages
Bulgarian (bg)
English (en)
Inventor
Robert Chambers
Thomas Magee
Anthony Marfat
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG106868A publication Critical patent/BG106868A/xx

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
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    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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  • Life Sciences & Earth Sciences (AREA)
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  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
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  • Virology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Biotechnology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
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BG106868A 2000-01-31 2002-06-24 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes BG106868A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17928200P 2000-01-31 2000-01-31
PCT/IB2001/000125 WO2001057025A1 (en) 2000-01-31 2001-01-30 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes

Publications (1)

Publication Number Publication Date
BG106868A true BG106868A (en) 2003-01-31

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Application Number Title Priority Date Filing Date
BG106868A BG106868A (en) 2000-01-31 2002-06-24 Pyrimidine carboxamides useful as inhibitors of pde4 isozymes

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US (1) US6740655B2 (xx)
EP (1) EP1252157B1 (xx)
JP (1) JP2003522165A (xx)
KR (1) KR20020071029A (xx)
CN (1) CN1404480A (xx)
AP (1) AP2002002590A0 (xx)
AR (1) AR027336A1 (xx)
AT (1) ATE269860T1 (xx)
AU (1) AU2700301A (xx)
BG (1) BG106868A (xx)
BR (1) BR0107934A (xx)
CA (1) CA2396458C (xx)
CO (1) CO5271669A1 (xx)
CR (1) CR6714A (xx)
CZ (1) CZ20022413A3 (xx)
DE (1) DE60103976T2 (xx)
DK (1) DK1252157T3 (xx)
DZ (1) DZ3406A1 (xx)
EA (1) EA005028B1 (xx)
EE (1) EE200200426A (xx)
ES (1) ES2223772T3 (xx)
GE (1) GEP20043385B (xx)
GT (1) GT200100023A (xx)
HK (1) HK1054232A1 (xx)
HN (1) HN2001000018A (xx)
HU (1) HUP0204271A3 (xx)
IL (1) IL150486A0 (xx)
IS (1) IS6444A (xx)
MA (1) MA26871A1 (xx)
MX (1) MXPA02007465A (xx)
NO (1) NO20023614L (xx)
NZ (1) NZ519726A (xx)
OA (1) OA12170A (xx)
PA (1) PA8511301A1 (xx)
PE (1) PE20011059A1 (xx)
PL (1) PL357555A1 (xx)
PT (1) PT1252157E (xx)
SK (1) SK10342002A3 (xx)
SV (1) SV2001000298A (xx)
TN (1) TNSN01019A1 (xx)
TR (1) TR200402292T4 (xx)
UY (1) UY26570A1 (xx)
WO (1) WO2001057025A1 (xx)
ZA (1) ZA200206034B (xx)

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ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
ES2238334T3 (es) * 1999-12-24 2005-09-01 Glaxo Group Limited Formulacion farmaceutica en aerosol de salmeterol y propionato de fluticasona.
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren
US7776315B2 (en) 2000-10-31 2010-08-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg Pharmaceutical compositions based on anticholinergics and additional active ingredients
YU39503A (sh) * 2000-11-22 2006-05-25 F. Hoffmann-La Roche Ag. Derivati pirimidina
ATE293109T1 (de) * 2001-01-31 2005-04-15 Pfizer Prod Inc Nikotinsäureamid-derivate und ihre mimetika als inhibitoren von pde4-isozyms
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