BE857541A - Derives d'acide prostanoique et leur procede de preparation - Google Patents

Derives d'acide prostanoique et leur procede de preparation

Info

Publication number: BE857541A
Authority: BE; Belgium
Prior art keywords: preparation process; acid derivatives; prostanoic acid; prostanoic; derivatives
Prior art date: 1976-08-06

Application number

BE179954A

Other languages

English (en)

French (fr)

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-08-06

Filing date

1977-08-05

Publication date

1978-02-06

1977-08-05 Application filed by Schering Ag filed Critical Schering Ag

1978-02-06 Publication of BE857541A publication Critical patent/BE857541A/xx

Links

238000002360 preparation method Methods 0.000 title 1
WGJJROVFWIXTPA-OALUTQOASA-N prostanoic acid Chemical class CCCCCCCC[C@H]1CCC[C@@H]1CCCCCCC(O)=O WGJJROVFWIXTPA-OALUTQOASA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
- C07D307/935—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
- C07C405/0008—Analogues having the carboxyl group in the side-chains replaced by other functional groups
- C07C405/0016—Analogues having the carboxyl group in the side-chains replaced by other functional groups containing only hydroxy, etherified or esterified hydroxy groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
- C07C405/0008—Analogues having the carboxyl group in the side-chains replaced by other functional groups
- C07C405/0025—Analogues having the carboxyl group in the side-chains replaced by other functional groups containing keto groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
- C07C405/0008—Analogues having the carboxyl group in the side-chains replaced by other functional groups
- C07C405/0041—Analogues having the carboxyl group in the side-chains replaced by other functional groups containing nitrogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/377—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by splitting-off hydrogen or functional groups; by hydrogenolysis of functional groups
- C07C51/38—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by splitting-off hydrogen or functional groups; by hydrogenolysis of functional groups by decarboxylation
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
- C07C57/03—Monocarboxylic acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
- C07C57/13—Dicarboxylic acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/52—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing halogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/535—Organo-phosphoranes
- C07F9/5352—Phosphoranes containing the structure P=C-

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Oil, Petroleum & Natural Gas (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Ink Jet (AREA)
Materials For Photolithography (AREA)
Polarising Elements (AREA)

BE179954A 1976-08-06 1977-08-05 Derives d'acide prostanoique et leur procede de preparation BE857541A (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19762635985 DE2635985A1 (de)	1976-08-06	1976-08-06	Prostansaeurederivat und verfahren zu ihrer herstellung

Publications (1)

Publication Number	Publication Date
BE857541A true BE857541A (fr)	1978-02-06

Family

ID=5985150

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BE179954A BE857541A (fr)	1976-08-06	1977-08-05	Derives d'acide prostanoique et leur procede de preparation

Country Status (12)

Country	Link
US (3)	US4284646A (xx)
JP (1)	JPS5340740A (xx)
BE (1)	BE857541A (xx)
CH (2)	CH637376A5 (xx)
DE (1)	DE2635985A1 (xx)
DK (1)	DK334577A (xx)
FR (1)	FR2392971A1 (xx)
GB (1)	GB1590654A (xx)
IE (1)	IE45863B1 (xx)
IT (1)	IT1085354B (xx)
LU (1)	LU77916A1 (xx)
NL (1)	NL7708741A (xx)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1078774B (it) *	1976-09-07	1985-05-08	Lpb Ist Farm	Derivato dell acido 19 metil 9 cheto 15 idrossi prost 18 enoico
US4257983A (en) *	1979-04-02	1981-03-24	The Upjohn Company	2-Decarboxy-2-aminomethyl-19,20-didehydro-PG1 compounds
US4257981A (en) *	1979-04-02	1981-03-24	The Upjohn Company	2-Decarboxy-2-aminomethyl-19,20-didehydro-PG2 compounds
US4276427A (en) *	1979-04-02	1981-06-30	The Upjohn Company	19,20-Didehydro-PG1 compounds
US4259529A (en) *	1979-04-02	1981-03-31	The Upjohn Company	2-Decarboxy-2-hydroxymethyl-19,20-didehydro-13,14-dihydro-PG1 compounds
US4257982A (en) *	1979-04-02	1981-03-24	The Upjohn Company	2-Decarboxy-2-aminomethyl-19,20-didehydro-13,14-dihydro-PG2 compounds
US4276428A (en) *	1979-04-02	1981-06-30	The Upjohn Company	19,20-Didehydro-13,14-dihydro-PG1 compounds
US4284795A (en) *	1979-04-02	1981-08-18	The Upjohn Company	19,20-Didehydro-PG2 compounds
US4257980A (en) *	1979-04-02	1981-03-24	The Upjohn Company	2-Decarboxy-2-aminomethyl-19,20-didehydro-13,14-dihydro-PG1 compounds
US4243611A (en) *	1979-04-02	1981-01-06	The Upjohn Company	2-Decarboxy-2-hydroxymethyl-19,20-didehydro PG2 compounds
US4269995A (en) *	1979-04-02	1981-05-26	The Upjohn Company	19,20-Didehydro-13,14-dihydro-PG2 compounds
US4257979A (en) *	1979-04-02	1981-03-24	The Upjohn Company	2-Decarboxy-2-aminomethyl-19-hydroxy-19-methyl-PG compounds
US4278818A (en) *	1979-04-02	1981-07-14	The Upjohn Company	2-Decarboxy-2-hydroxymethyl-19,20-didehydro-13,14-dihydro-PG2 compounds
US4251463A (en) *	1979-05-01	1981-02-17	The Upjohn Company	2-Decarboxy-2-aminomethyl-9-deoxy-9-methylene-5,6-didehydro-PGF1 compounds
US4254058A (en) *	1979-07-05	1981-03-03	The Upjohn Company	2-Decarboxy-2-aminomethyl-19-hydroxy-6a-carba-PGI2 compounds
US4256667A (en) *	1979-07-05	1981-03-17	The Upjohn Company	2-Decarboxy-2-aminomethyl-19-hydroxy-19-methyl-6a-carba-PGI2 compounds
US4251464A (en) *	1979-07-05	1981-02-17	The Upjohn Company	2-Decarboxy-2-aminomethyl-19-hydroxy-6-oxo-PGE1 compounds
US4255354A (en) *	1979-07-05	1981-03-10	The Upjohn Company	2-Decarboxy-2-aminomethyl-19-hydroxy-19-methyl-6-oxo-PGF1 compounds
FI71308C (fi) *	1981-02-13	1986-12-19	Schering Ag	Analogifoerfarande foer framstaellning av terapeutiskt anvaendbara (13e)-(8r,11r,12r)-11,15-dihydroxi-16,19-dimetyl-9-oxo-13,18-prostadiensyraderivat och av deras salter
CA2109109A1 (en) *	1991-04-22	1992-10-23	Fumie Sato	Prostaglandin e1 analogues
CA2088128C (en) *	1992-01-31	2002-10-29	Katsuhiro Imaki	Salts of glucopyranose derivatives and its intermediate
US5545665A (en)	1993-12-28	1996-08-13	Allergan	Cyclopentane(ene) heptenoic or heptanoic acids and derivatives thereof useful as therapeutic agents
JP4834224B2 (ja)	1999-03-05	2011-12-14	デュークユニバーシティ	Ｃ１６不飽和ｆｐ−選択的プロスタグランジン類縁体
US6894175B1 (en) *	1999-08-04	2005-05-17	The Procter & Gamble Company	2-Decarboxy-2-phosphinico prostaglandin derivatives and methods for their preparation and use
US20020172693A1 (en)	2000-03-31	2002-11-21	Delong Michell Anthony	Compositions and methods for treating hair loss using non-naturally occurring prostaglandins
US20020037914A1 (en)	2000-03-31	2002-03-28	Delong Mitchell Anthony	Compositions and methods for treating hair loss using C16-C20 aromatic tetrahydro prostaglandins
US20020013294A1 (en)	2000-03-31	2002-01-31	Delong Mitchell Anthony	Cosmetic and pharmaceutical compositions and methods using 2-decarboxy-2-phosphinico derivatives
US20090148527A1 (en) *	2007-12-07	2009-06-11	Robinson Michael R	Intraocular formulation
US8722739B2 (en) *	2008-10-29	2014-05-13	Novaer Holdings, Inc.	Amino acid salts of prostaglandins
US8623918B2 (en) *	2008-10-29	2014-01-07	Novaer Holdings, Inc.	Amino acid salts of prostaglandins
US10486881B2 (en)	2016-12-09	2019-11-26	Fres-Co System Usa, Inc.	Flexible packages with clog resistant degassing valve and methods of making the same

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3419285A (en) *	1967-05-02	1968-12-31	Earl P. Morehouse	Towing hitch
US3919285A (en) *	1971-02-02	1975-11-11	Upjohn Co	PGE{HD 3 {B analogs
US3932479A (en) *	1973-04-27	1976-01-13	American Cyanamid Company	Lithium 3-triphenylmethoxy-1-trans-alkenyl-dialkyl alanates
US4064351A (en) *	1974-09-19	1977-12-20	Sankyo Company Limited	9-OXO-15 ξ-HYDROXY-20-ALKYLIDENEPROST-13(TRANS)-ENOIC ACID DERIVATIVES
GB1499018A (en) *	1974-09-19	1978-01-25	Sankyo Co	Pharmaceutically useful prostenoic acid derivatives
IT1078774B (it) *	1976-09-07	1985-05-08	Lpb Ist Farm	Derivato dell acido 19 metil 9 cheto 15 idrossi prost 18 enoico

1976
- 1976-08-06 DE DE19762635985 patent/DE2635985A1/de not_active Ceased
1977
- 1977-07-25 DK DK334577A patent/DK334577A/da not_active Application Discontinuation
- 1977-08-02 CH CH950677A patent/CH637376A5/de not_active IP Right Cessation
- 1977-08-03 IE IE1613/77A patent/IE45863B1/en unknown
- 1977-08-04 LU LU77916A patent/LU77916A1/xx unknown
- 1977-08-05 JP JP9405577A patent/JPS5340740A/ja active Pending
- 1977-08-05 BE BE179954A patent/BE857541A/xx not_active IP Right Cessation
- 1977-08-05 GB GB32916/77A patent/GB1590654A/en not_active Expired
- 1977-08-05 IT IT26535/77A patent/IT1085354B/it active
- 1977-08-08 NL NL7708741A patent/NL7708741A/xx not_active Application Discontinuation
- 1977-08-08 FR FR7724385A patent/FR2392971A1/fr active Granted
1979
- 1979-08-24 US US06/069,193 patent/US4284646A/en not_active Expired - Lifetime
1981
- 1981-04-22 US US06/256,369 patent/US4359467A/en not_active Expired - Fee Related
1982
- 1982-09-01 US US06/413,940 patent/US4489092A/en not_active Expired - Lifetime
1983
- 1983-01-31 CH CH54183A patent/CH641158A5/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE45863L (en)	1978-02-06
NL7708741A (nl)	1978-02-08
US4359467A (en)	1982-11-16
FR2392971B1 (xx)	1980-02-15
CH637376A5 (de)	1983-07-29
JPS5340740A (en)	1978-04-13
FR2392971A1 (fr)	1978-12-29
US4489092A (en)	1984-12-18
LU77916A1 (xx)	1977-11-14
CH641158A5 (de)	1984-02-15
IE45863B1 (en)	1982-12-15
DK334577A (da)	1978-02-07
IT1085354B (it)	1985-05-28
US4284646A (en)	1981-08-18
GB1590654A (en)	1981-06-03
DE2635985A1 (de)	1978-02-09

Legal Events

Date

Code

Title

Description

1986-02-28

RE

Patent lapsed

Owner name: SCHERING A.G.

Effective date: 19850831

Publication	Publication Date	Title
BE857541A (fr)	1978-02-06	Derives d'acide prostanoique et leur procede de preparation
FR2296407A1 (fr)	1976-07-30	Derives d'acide benzoique, leur procede de preparation et leur application
FR2483409B1 (fr)	1986-05-09	Derives de l'acide 3-amino-2-hydroxy butanoylaminoacetique et leur procede de preparation
FR2468599B1 (fr)	1986-03-21	Derives d'acide thiazolylacetique et procede de preparation
FR2318627A1 (fr)	1977-02-18	Derives de l'acide phenylacetique et leur procede de preparation
BE887574R (fr)	1981-06-15	Derives de l'acide quinoleine-carboxylique et procede pour leur preparation
BE868417A (fr)	1978-12-27	Derives d'acide 1,2,3-thiadiazole-5-carboxylique leur procede de preparation et leur utilisation
BE864112A (fr)	1978-08-21	Derives d'acide benzoique, leur procede de preparation et leur application en therapeutique
FR2281340A1 (fr)	1976-03-05	Derives de l'acide folique, leur procede de preparation et leur application
BE859064A (fr)	1978-01-16	Derives d'acide folique a marquage radioactif et leur procede de preparation
BE818209A (fr)	1974-11-18	Derives de l'acide 7-acylamino-3-cephene-4-carboxylique et leur procede de preparation
BE882195A (fr)	1980-09-12	Derives d'acide 1,2,3-thiadiazole-5-carboxylique, leur procede de preparation et leur utilisation
BE822496A (fr)	1975-05-22	Derives d'acide hydratropique et leur procede de preparation
PT67088A (fr)	1977-10-01	Procede de preparation de derives de l'acide(phenyl-3-amino-2-propionyloxy)-2-acetique
BE856095A (fr)	1977-12-27	Nouveaux derives d'acide isophtalamique iode, leur procede de preparation et leur utilisation
FR2348226A1 (fr)	1977-11-10	Procede de preparation d'acides steroidecarboxyliques et de leurs esters
BE827870A (fr)	1975-10-13	Derives d'emidazole et leur procede de preparation
BE831298A (fr)	1976-01-12	Nouveaux derives d'acide prostanoique et leur procede de preparation
BE855532A (fr)	1977-12-09	1,1-dioxyde d'acide 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylique, son procede de preparation et son application
BE855822A (fr)	1977-12-19	Derives d'acide troponyl-oxamique et leur preparation
FR2353556A1 (fr)	1977-12-30	Derives de l'acide clavulanique, leur procede de preparation et leur application en therapeutique
BE841165A (fr)	1976-10-27	Derives d'acides 8-aza-prostanoiques et leur procede de preparation
BE856326A (fr)	1977-12-30	Nouveaux derives d'acide prostanoique et leur procede de preparation
BE837860A (fr)	1976-05-14	Derives d'acide glycyrrhetinique et procede pour leur preparation
BE846141A (fr)	1977-03-14	Procede de preparation de l'acide oxo-5 hexanoique et de ses derives