BE764913A - Procede de preparation de derives de benzodiazepine - Google Patents

Procede de preparation de derives de benzodiazepine

Info

Publication number
BE764913A
BE764913A BE764913A BE764913A BE764913A BE 764913 A BE764913 A BE 764913A BE 764913 A BE764913 A BE 764913A BE 764913 A BE764913 A BE 764913A BE 764913 A BE764913 A BE 764913A
Authority
BE
Belgium
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
BE764913A
Other languages
English (en)
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2580570A external-priority patent/JPS5010316B1/ja
Priority claimed from JP2580470A external-priority patent/JPS4811112B1/ja
Priority claimed from JP3495070A external-priority patent/JPS5011920B1/ja
Priority claimed from JP4663770A external-priority patent/JPS4924060B1/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of BE764913A publication Critical patent/BE764913A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BE764913A 1970-03-27 1971-03-26 Procede de preparation de derives de benzodiazepine BE764913A (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2580570A JPS5010316B1 (fr) 1970-03-27 1970-03-27
JP2580470A JPS4811112B1 (fr) 1970-03-27 1970-03-27
JP3495070A JPS5011920B1 (fr) 1970-04-23 1970-04-23
JP4663770A JPS4924060B1 (fr) 1970-05-28 1970-05-28

Publications (1)

Publication Number Publication Date
BE764913A true BE764913A (fr) 1971-08-16

Family

ID=27458380

Family Applications (1)

Application Number Title Priority Date Filing Date
BE764913A BE764913A (fr) 1970-03-27 1971-03-26 Procede de preparation de derives de benzodiazepine

Country Status (14)

Country Link
US (1) US4102881A (fr)
BE (1) BE764913A (fr)
CA (2) CA922317A (fr)
CH (1) CH559188A5 (fr)
DE (1) DE2114441A1 (fr)
DK (1) DK131374B (fr)
FI (1) FI55334C (fr)
FR (1) FR2085748B1 (fr)
GB (1) GB1353486A (fr)
NL (1) NL7104132A (fr)
NO (1) NO132800C (fr)
PH (1) PH9214A (fr)
SE (1) SE400968B (fr)
YU (1) YU34997B (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2203782A1 (de) * 1971-02-09 1972-08-24 The Upjohn Co., Kalamazoo, Mich. (V.StA.) Verfahren zur Herstellung von Triazolobenzodiazepinen sowie neue Triazolobenzodiazepine und deren Zwischenprodukte

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines
US4755508A (en) * 1984-06-26 1988-07-05 Merck & Co., Inc. Benzodiazepine analogs and use as antogonists of gastrin and cholecystokinin
CA2269135A1 (fr) * 1996-10-31 1998-05-07 Merck & Co., Inc. Derives de benzodiazepine hydrazide utilises comme inhibiteurs de l'integrase du vih
US5939414A (en) * 1996-10-31 1999-08-17 Merck & Co., Inc. Benzodiazepine hydrazide derivatives as inhibitors of HIV integrase

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3462418A (en) * 1963-10-29 1969-08-19 Hoffmann La Roche Preparation of 1,4-benzodiazepin-2-one-4-oxide from 2-lower alkoxy-1,4-benzodiazepine-4-oxide
DK120901B (da) * 1965-09-17 1971-08-02 Rexolin Chem Fremgangsmåde til fremstilling af 7-chlor-1,3-dihydro-1-methyl-5-phenyl-2H-1,4-benzodiazepin-2-on.
US3987052A (en) * 1969-03-17 1976-10-19 The Upjohn Company 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines
ZA705076B (en) * 1969-07-30 1971-04-28 Grindstedvaerket As New 1,4-benzodiazepines
BE755139A (fr) * 1969-08-21 1971-02-22 Upjohn Co Derives de benzodiazepinones, leurs intermediaires, et leur preparatio
FR2022598A1 (en) * 1969-11-04 1970-07-31 Pakeda Chemical Ind Sedative chloro-phenyl-triazolobenzodiazepines

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2203782A1 (de) * 1971-02-09 1972-08-24 The Upjohn Co., Kalamazoo, Mich. (V.StA.) Verfahren zur Herstellung von Triazolobenzodiazepinen sowie neue Triazolobenzodiazepine und deren Zwischenprodukte

Also Published As

Publication number Publication date
CH559188A5 (fr) 1975-02-28
GB1353486A (en) 1974-05-15
CA922317A (en) 1973-03-06
US4102881A (en) 1978-07-25
NO132800C (fr) 1976-01-07
NL7104132A (fr) 1971-09-29
FI55334B (fi) 1979-03-30
YU34997B (en) 1980-06-30
DK131374B (da) 1975-07-07
PH9214A (en) 1975-07-10
YU73771A (en) 1979-12-31
NO132800B (fr) 1975-09-29
DK131374C (fr) 1975-12-01
DE2114441A1 (de) 1971-10-14
FI55334C (fi) 1979-07-10
CA936864A (en) 1973-11-13
FR2085748A1 (fr) 1971-12-31
FR2085748B1 (fr) 1974-08-02
SE400968B (sv) 1978-04-17

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