AU666740B2 - 5'-indolinyl oxazolidinones useful against (mycobacterium tuberculosis) - Google Patents

5'-indolinyl oxazolidinones useful against (mycobacterium tuberculosis) Download PDF

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Publication number
AU666740B2
AU666740B2 AU43865/93A AU4386593A AU666740B2 AU 666740 B2 AU666740 B2 AU 666740B2 AU 43865/93 A AU43865/93 A AU 43865/93A AU 4386593 A AU4386593 A AU 4386593A AU 666740 B2 AU666740 B2 AU 666740B2
Authority
AU
Australia
Prior art keywords
indolinyl
document
international
date
oxazolidinone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
AU43865/93A
Other languages
English (en)
Other versions
AU4386593A (en
Inventor
Steven Joseph Brickner
Gary Edward Zurenko
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of AU4386593A publication Critical patent/AU4386593A/en
Application granted granted Critical
Publication of AU666740B2 publication Critical patent/AU666740B2/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AU43865/93A 1992-07-08 1993-05-26 5'-indolinyl oxazolidinones useful against (mycobacterium tuberculosis) Expired - Fee Related AU666740B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US90938792A 1992-07-08 1992-07-08
US909387 1992-07-08
PCT/US1993/004850 WO1994001110A1 (en) 1992-07-08 1993-05-26 5'-INDOLINYL OXAZOLIDINONES USEFUL AGAINST $i(MYCOBACTERIUM TUBERCULOSIS)

Publications (2)

Publication Number Publication Date
AU4386593A AU4386593A (en) 1994-01-31
AU666740B2 true AU666740B2 (en) 1996-02-22

Family

ID=25427164

Family Applications (1)

Application Number Title Priority Date Filing Date
AU43865/93A Expired - Fee Related AU666740B2 (en) 1992-07-08 1993-05-26 5'-indolinyl oxazolidinones useful against (mycobacterium tuberculosis)

Country Status (9)

Country Link
EP (1) EP0648119A1 (ja)
JP (1) JPH07508985A (ja)
KR (1) KR950702417A (ja)
AU (1) AU666740B2 (ja)
CA (1) CA2136324A1 (ja)
IL (1) IL106220A0 (ja)
MX (1) MX9303764A (ja)
TW (1) TW260608B (ja)
WO (1) WO1994001110A1 (ja)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9717807D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
GB9725244D0 (en) 1997-11-29 1998-01-28 Zeneca Ltd Chemical compounds
CN1311787A (zh) 1998-06-05 2001-09-05 阿斯特拉曾尼卡有限公司 噁唑烷酮衍生物、其制备方法以及含有它们的药物组合物
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
US7141588B2 (en) 2002-02-25 2006-11-28 Pfizer, Inc. N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
AR038536A1 (es) 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
CA2491287A1 (en) 2002-08-12 2004-02-19 Pharmacia & Upjohn Company N-aryl-2-oxazolidinones and their derivatives
ES2271660T3 (es) 2002-11-21 2007-04-16 PHARMACIA & UPJOHN COMPANY LLC Derivados de n-(4-piperazin-1-il)-fenil-2-oxazolidinona-5-carboxamida y compuestos relacionados como agentes antibacterianos.
US7304050B2 (en) 2003-09-16 2007-12-04 Pfizer Inc. Antibacterial agents
KR20230052873A (ko) 2020-06-18 2023-04-20 아카제라 메디신즈, 인크. 옥사졸리디논 화합물, 옥사졸리디논 화합물을 포함하는 리포좀 조성물 및 이의 사용 방법

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990002744A1 (en) * 1988-09-15 1990-03-22 The Upjohn Company In position 3 substituted-5-beta-amidomethyl-oxazolidin-2-ones

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5314792A (en) * 1976-07-24 1978-02-09 Rubuobuna Buratsurabusukay Ara Copolymers of nnvinylmethylpyrazol and diivinyl crossslinking agent and process for producing same
JPS54110186A (en) * 1978-02-17 1979-08-29 Tokyo Yuuki Kagaku Kougiyou Kk Method of mamufacturing weak basic anion exchange resin
DE3324835A1 (de) * 1983-07-09 1985-01-17 Cassella Ag, 6000 Frankfurt Vernetztes copolymerisat, verfahren zu seiner herstellung und seine verwendung als sorptionsmittel
JPS6023854A (ja) * 1983-07-19 1985-02-06 Konishiroku Photo Ind Co Ltd 写真要素
DE3434137A1 (de) * 1984-09-18 1986-03-20 Basf Ag, 6700 Ludwigshafen Verfahren zur herstellung von unloeslichen, nur wenig quellbaren pulverfoermigen polymeren
JPS63130605A (ja) * 1986-11-20 1988-06-02 Tokuyama Soda Co Ltd 陰イオン交換体の製造方法
US4889632A (en) * 1987-12-10 1989-12-26 Ceskoslovenska Akademie Ved Macroporous polymeric membranes for the separation of polymers and a method of their application
GB8829835D0 (en) * 1988-12-21 1989-02-15 Smith Kline French Lab Compounds
JPH03708A (ja) * 1989-05-29 1991-01-07 Koei Chem Co Ltd 吸水性材料

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990002744A1 (en) * 1988-09-15 1990-03-22 The Upjohn Company In position 3 substituted-5-beta-amidomethyl-oxazolidin-2-ones

Also Published As

Publication number Publication date
AU4386593A (en) 1994-01-31
JPH07508985A (ja) 1995-10-05
IL106220A0 (en) 1993-11-15
EP0648119A1 (en) 1995-04-19
KR950702417A (ko) 1995-07-29
MX9303764A (es) 1994-01-31
WO1994001110A1 (en) 1994-01-20
TW260608B (ja) 1995-10-21
CA2136324A1 (en) 1994-01-20

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