AU3124300A - Inhibitors of beta-lactamases and uses therefor - Google Patents
Inhibitors of beta-lactamases and uses thereforInfo
- Publication number
- AU3124300A AU3124300A AU31243/00A AU3124300A AU3124300A AU 3124300 A AU3124300 A AU 3124300A AU 31243/00 A AU31243/00 A AU 31243/00A AU 3124300 A AU3124300 A AU 3124300A AU 3124300 A AU3124300 A AU 3124300A
- Authority
- AU
- Australia
- Prior art keywords
- lactamases
- inhibitors
- beta
- uses therefor
- therefor
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/69—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11244898P | 1998-12-16 | 1998-12-16 | |
US60112448 | 1998-12-16 | ||
PCT/US1999/029958 WO2000035904A1 (en) | 1998-12-16 | 1999-12-16 | INHIBITORS OF β-LACTAMASES AND USES THEREFOR |
Publications (1)
Publication Number | Publication Date |
---|---|
AU3124300A true AU3124300A (en) | 2000-07-03 |
Family
ID=22343962
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU31243/00A Abandoned AU3124300A (en) | 1998-12-16 | 1999-12-16 | Inhibitors of beta-lactamases and uses therefor |
Country Status (2)
Country | Link |
---|---|
AU (1) | AU3124300A (en) |
WO (1) | WO2000035904A1 (en) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6858592B2 (en) | 2001-06-29 | 2005-02-22 | Genzyme Corporation | Aryl boronic acids for treating obesity |
US7041280B2 (en) | 2001-06-29 | 2006-05-09 | Genzyme Corporation | Aryl boronate functionalized polymers for treating obesity |
US7112572B2 (en) | 2002-09-09 | 2006-09-26 | Trigen Limited | Multivalent metal salts of boronic acids |
PT2603514T (en) | 2010-08-10 | 2018-11-09 | Rempex Pharmaceuticals Inc | Cyclic boronic acid ester derivatives and therapeutic uses thereof |
US9012491B2 (en) | 2011-08-31 | 2015-04-21 | Rempex Pharmaceuticals, Inc. | Heterocyclic boronic acid ester derivatives and therapeutic uses thereof |
US9156858B2 (en) | 2012-05-23 | 2015-10-13 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
US10561675B2 (en) | 2012-06-06 | 2020-02-18 | Rempex Pharmaceuticals, Inc. | Cyclic boronic acid ester derivatives and therapeutic uses thereof |
AU2014204045B2 (en) | 2013-01-04 | 2018-10-18 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
US9101638B2 (en) | 2013-01-04 | 2015-08-11 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
CA2894892A1 (en) | 2013-01-04 | 2014-07-10 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
US9241947B2 (en) | 2013-01-04 | 2016-01-26 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
LT3604316T (en) | 2014-05-05 | 2024-02-26 | Melinta Therapeutics, Inc. | Synthesis of boronate salts |
WO2015171398A1 (en) | 2014-05-05 | 2015-11-12 | Rempex Pharmaceuticals, Inc. | Salts and polymorphs of cyclic boronic acid ester derivatives and therapeutic uses thereof |
WO2015179308A1 (en) | 2014-05-19 | 2015-11-26 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
WO2016003929A1 (en) | 2014-07-01 | 2016-01-07 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
WO2016081297A1 (en) | 2014-11-18 | 2016-05-26 | Rempex Pharmaceuticals, Inc. | Cyclic boronic acid ester derivatives and therapeutic uses thereof |
US20180051041A1 (en) | 2015-03-17 | 2018-02-22 | Rempex Pharmaceuticals, Inc. | Boronic acid derivatives and therapeutic uses thereof |
DK3478693T3 (en) | 2016-06-30 | 2021-09-20 | Qpex Biopharma Inc | BORONIC ACID DERIVATIVES AND THERAPEUTIC USES THEREOF |
US11286270B2 (en) | 2017-10-11 | 2022-03-29 | Qpex Biopharma, Inc. | Boronic acid derivatives and synthesis thereof |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5612378A (en) * | 1995-06-06 | 1997-03-18 | 3-Dimensional Pharmaceuticals, Inc. | Bis-arylsulfonylaminobenzamide derivatives and the use thereof as factor Xa inhibitors |
US6008377A (en) * | 1996-03-19 | 1999-12-28 | Eli Lilly And Company | Synthesis of 3-[4-(2-aminoethoxy)-benzoyl]-2-aryl-6-hydroxy-benzo[B]thiophenes |
-
1999
- 1999-12-16 AU AU31243/00A patent/AU3124300A/en not_active Abandoned
- 1999-12-16 WO PCT/US1999/029958 patent/WO2000035904A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2000035904A1 (en) | 2000-06-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |