AU2002218365A1 - Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents - Google Patents

Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents

Info

Publication number: AU2002218365A1
Authority: AU; Australia
Prior art keywords: antimicrobial agents; piperidine derivatives; heterocyclylalkyl piperidine; heterocyclylalkyl; derivatives
Prior art date: 2000-11-15
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2002218365A

Other versions

AU2002218365B2 (en

Inventor

Eric Bacque

Jean-Christophe Carry

Youssef El Ahmad

Michel Evers

Philippe Hubert

Jean-Luc Malleron

Serge Mignani

Guy Pantel

Michel Tabart

Fabrice Viviani

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Novexel SA

Original Assignee

Novexel SA

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2001-11-14

Publication date

2002-08-01

2000-11-15 Priority claimed from FR0014738A external-priority patent/FR2816618B1/en

2001-11-14 Application filed by Novexel SA filed Critical Novexel SA

2002-08-01 Publication of AU2002218365A1 publication Critical patent/AU2002218365A1/en

2006-12-14 Assigned to NOVEXEL reassignment NOVEXEL Request for Assignment Assignors: AVENTIS PHARMA S.A.

2007-07-05 Application granted granted Critical

2007-07-05 Publication of AU2002218365B2 publication Critical patent/AU2002218365B2/en

2007-10-05 Priority to AU2007226805A priority Critical patent/AU2007226805A1/en

2021-11-14 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Links

-1 Heterocyclylalkyl piperidine derivatives Chemical class 0.000 title 1
239000004599 antimicrobial Substances 0.000 title 1

AU2002218365A 2000-11-15 2001-11-14 Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents Ceased AU2002218365B2 (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
AU2007226805A AU2007226805A1 (en)	2000-11-15	2007-10-05	Heterocyclylalkyl piperidine derivatives

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR00/14738		2000-11-15
FR0014738A FR2816618B1 (en)	2000-11-15	2000-11-15	HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM
PCT/FR2001/003559 WO2002040474A2 (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents

Related Child Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2007226805A Division AU2007226805A1 (en)	2000-11-15	2007-10-05	Heterocyclylalkyl piperidine derivatives

Publications (2)

Publication Number	Publication Date
AU2002218365A1 true AU2002218365A1 (en)	2002-08-01
AU2002218365B2 AU2002218365B2 (en)	2007-07-05

Family

ID=8856503

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2002218365A Ceased AU2002218365B2 (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents
AU1836502A Pending AU1836502A (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU1836502A Pending AU1836502A (en)	2000-11-15	2001-11-14	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same

Country Status (28)

Country	Link
EP (2)	EP1695964A1 (en)
JP (1)	JP2004514661A (en)
KR (1)	KR100849608B1 (en)
CN (1)	CN1483031A (en)
AR (1)	AR034006A1 (en)
AT (1)	ATE337311T1 (en)
AU (2)	AU2002218365B2 (en)
BG (1)	BG107793A (en)
BR (1)	BR0115312A (en)
CA (1)	CA2429311A1 (en)
CZ (1)	CZ20031316A3 (en)
DE (1)	DE60122567T2 (en)
DK (1)	DK1337529T3 (en)
EA (1)	EA200300568A1 (en)
EE (1)	EE200300207A (en)
ES (1)	ES2271119T3 (en)
FR (1)	FR2816618B1 (en)
HR (1)	HRP20030379A2 (en)
HU (1)	HUP0303758A3 (en)
IL (1)	IL155841A0 (en)
NO (2)	NO20032187L (en)
PL (1)	PL363004A1 (en)
PT (1)	PT1337529E (en)
SK (1)	SK5822003A3 (en)
TN (1)	TNSN01160A1 (en)
WO (1)	WO2002040474A2 (en)
YU (1)	YU46803A (en)
ZA (1)	ZA200303794B (en)

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AU2001289749B9 (en)	2000-07-26	2004-08-19	Smithkline Beecham P.L.C.	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
AR038240A1 (en)	2002-01-29	2005-01-05	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE FOR PREPARATION
EP1470131A2 (en)	2002-01-29	2004-10-27	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
AR040336A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND
FR2842807A1 (en) *	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (en)	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en) *	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
WO2004096982A2 (en)	2002-11-05	2004-11-11	Smithkline Beecham Corporation	Antibacterial agents
DE60324179D1 (en)	2002-12-04	2008-11-27	Glaxo Group Ltd	CHINOLINE AND NITROGENIC DERIVATEDAVAN AND THEIR USE AS ANTIBACTERIAL AGENTS
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR2862301B1 (en) *	2003-11-17	2007-12-21	Aventis Pharma Sa	NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) *	2004-03-12	2008-07-18	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
EP1846417A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	Antibacterial agents
US7709472B2 (en)	2005-01-25	2010-05-04	Glaxo Group Limited	Antibacterial agents
JP2008528586A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
US7592334B2 (en)	2005-01-25	2009-09-22	Glaxo Group Limited	Antibacterial agents
US7700595B2 (en)	2005-03-01	2010-04-20	Wyeth Llc	Cinnoline compounds
MY150958A (en)	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
JP2009524643A (en)	2006-01-26	2009-07-02	アクテリオンファーマシューティカルズリミテッド	Tetrahydropyran antibiotics
JP2009532423A (en)	2006-04-06	2009-09-10	グラクソグループリミテッド	Pyrrolo-quinoxalinone derivatives as antibacterial agents
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
WO2008152603A1 (en)	2007-06-15	2008-12-18	Actelion Pharmaceuticals Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
WO2010043714A1 (en)	2008-10-17	2010-04-22	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
JP5653935B2 (en)	2009-01-15	2015-01-14	グラクソグループリミテッドＧｌａｘｏＧｒｏｕｐＬｉｍｉｔｅｄ	Naphthyridin-2 (1H) -one compounds useful as antibacterial agents
US9273001B2 (en) *	2012-08-15	2016-03-01	Glaxo Group Limited	Chemical process
TW201618779A (en)	2014-08-22	2016-06-01	葛蘭素史克智慧財產發展有限公司	Methods
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
UY36851A (en)	2015-08-16	2017-03-31	Glaxosmithkline Ip Dev Ltd	COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS

Family Cites Families (6)

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Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (en)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en)	1988-07-29	1990-02-08	Origin Electric Co Ltd	Manufacture of hybrid integrated circuit
AU623474B2 (en)	1989-01-16	1992-05-14	Laboratoire Roger Bellon	New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
ES2201674T3 (en) *	1998-01-26	2004-03-16	Smithkline Beecham Plc	DERIVATIVES OF QUINOLINA WITH ANTIBACTERIAL PROPERTIES.
WO2000043383A1 (en) *	1999-01-20	2000-07-27	Smithkline Beecham P.L.C.	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en active IP Right Grant
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active IP Right Cessation
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation

Publication	Publication Date	Title
AU2002218365A1 (en)	2002-08-01	Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents
PL363004A1 (en)	2004-11-15	Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents
AU2001277754A1 (en)	2002-05-23	Proline derivatives and use thereof as drugs
AU2002226486A1 (en)	2002-07-08	Novel c-glycoside derivatives and use thereof
AU2001286878A1 (en)	2002-03-13	Oxazolidinones and their use as antibacterial agents
HUP0300746A3 (en)	2005-09-28	Proline derivatives and use thereof as drugs
AU2002226487A1 (en)	2002-07-08	Novel c-glycoside derivatives and use thereof
IL148720A0 (en)	2002-09-12	Quinolyl propyl piperidine derivatives and their use as antibacterial agents
PT1296974E (en)	2009-11-03	2-cyanopyrrolidine derivatives and their use as medicaments
AU2002235128A1 (en)	2002-05-27	Expression miniarrays and uses thereof
AU9025701A (en)	2002-04-15	Glucopyranosyloxybenzylbenzene derivatives and medicinal compositions containingthe same
AU2001294814A1 (en)	2002-04-08	Pumpcn compositions and uses thereof
HUP0204101A3 (en)	2004-05-28	3-aminoquinazolin-2,4-dione antibacterial agents, pharmaceutical compositions containing them and their use
AU2001277526A1 (en)	2002-01-30	Substituted benzo-nitro-heterocycles and use thereof as herbicides
AU4923200A (en)	2000-12-18	Isothiazolecarboxamides and their use as microbicides
AU2002214948A1 (en)	2002-02-18	Heterocyclylalkyl azole derivatives and use thereof as pesticidal agents
AU2001235437A1 (en)	2001-08-07	Isothiazolecarboxylic acid derivatives and their use as microbicides
AU2001227084A1 (en)	2001-08-07	N-arylhydrazide compounds and use thereof as drugs
AU5464901A (en)	2001-09-12	Dichloropyridyl- and dichloroisothiazolyl-thiocarboxamides and their use as microbicides
AU1152601A (en)	2001-05-08	Compositions and their use
AU2001237025A1 (en)	2001-08-27	Antimicrobial composition and articles
AU2001241037A1 (en)	2001-09-03	Use of piperidine benzoderivatives as fungicides
AU2002223655A1 (en)	2002-05-15	Indolylpiperidine derivatives as antihistaminic and antiallergic agents
AU4432001A (en)	2001-10-08	Trityl-type compounds and their use
AU2002220830A1 (en)	2002-06-03	Metal-chelating adsorbents and their use