ATE542812T1 - Substituierte indolylalkylaminoderivate als neue inhibitoren von histondeacetylase - Google Patents

Substituierte indolylalkylaminoderivate als neue inhibitoren von histondeacetylase

Info

Publication number
ATE542812T1
ATE542812T1 AT05767934T AT05767934T ATE542812T1 AT E542812 T1 ATE542812 T1 AT E542812T1 AT 05767934 T AT05767934 T AT 05767934T AT 05767934 T AT05767934 T AT 05767934T AT E542812 T1 ATE542812 T1 AT E542812T1
Authority
AT
Austria
Prior art keywords
indolylalkylamino
derivatives
substituted
histone deacetylase
new inhibitors
Prior art date
Application number
AT05767934T
Other languages
English (en)
Inventor
Marc Gustaaf C Verdonck
Patrick Rene Angibaud
Bruno Roux
Isabelle Noelle Constance Pilatte
Holte Peter Ten
Janine Arts
Emelen Kristof Van
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority claimed from PCT/EP2005/053612 external-priority patent/WO2006010750A1/en
Application granted granted Critical
Publication of ATE542812T1 publication Critical patent/ATE542812T1/de

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AT05767934T 2004-07-28 2005-07-25 Substituierte indolylalkylaminoderivate als neue inhibitoren von histondeacetylase ATE542812T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP04077172 2004-07-28
US59218204P 2004-07-29 2004-07-29
PCT/EP2005/053612 WO2006010750A1 (en) 2004-07-28 2005-07-25 Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase

Publications (1)

Publication Number Publication Date
ATE542812T1 true ATE542812T1 (de) 2012-02-15

Family

ID=34928411

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05767934T ATE542812T1 (de) 2004-07-28 2005-07-25 Substituierte indolylalkylaminoderivate als neue inhibitoren von histondeacetylase

Country Status (10)

Country Link
CN (1) CN1993353B (de)
AT (1) ATE542812T1 (de)
DK (1) DK1781639T3 (de)
ES (1) ES2381117T3 (de)
ME (1) ME01444B (de)
PT (1) PT1781639E (de)
RS (1) RS52304B (de)
SI (1) SI1781639T1 (de)
UA (1) UA93352C2 (de)
ZA (1) ZA200700764B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107095871A (zh) * 2016-02-22 2017-08-29 中国科学院上海巴斯德研究所 Quisinostat,一种新型的高效抗疟药物
CN107721980B (zh) * 2017-08-25 2019-07-12 南京医科大学 一类氟尿嘧啶和Quisinosta的乏氧靶向前药及其应用
CN112485233B (zh) * 2020-11-03 2022-08-26 山东师范大学 一种检测去乙酰化酶用纳米传感器及其检测方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ534831A (en) * 2002-03-13 2007-01-26 Janssen Pharmaceutica Nv Carbonylamino-derivatives having histone deacetylase (HDAC) inhibiting enzymatic activity

Also Published As

Publication number Publication date
CN1993353A (zh) 2007-07-04
PT1781639E (pt) 2012-05-02
DK1781639T3 (da) 2012-05-14
ZA200700764B (en) 2008-09-25
RS52304B (en) 2012-12-31
SI1781639T1 (sl) 2012-06-29
ME01444B (me) 2013-12-20
ES2381117T3 (es) 2012-05-23
CN1993353B (zh) 2010-12-01
UA93352C2 (ru) 2011-02-10

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