ATE177099T1 - Diazabicyclische neurokinin antagonisten - Google Patents

Diazabicyclische neurokinin antagonisten

Info

Publication number
ATE177099T1
ATE177099T1 AT94931148T AT94931148T ATE177099T1 AT E177099 T1 ATE177099 T1 AT E177099T1 AT 94931148 T AT94931148 T AT 94931148T AT 94931148 T AT94931148 T AT 94931148T AT E177099 T1 ATE177099 T1 AT E177099T1
Authority
AT
Austria
Prior art keywords
diazabicyclic
neurokinin antagonists
compounds
formula
disorders
Prior art date
Application number
AT94931148T
Other languages
English (en)
Inventor
Harry R Howard Jr
Kevin D Shenk
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE177099T1 publication Critical patent/ATE177099T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, ***e
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT94931148T 1993-12-29 1994-11-14 Diazabicyclische neurokinin antagonisten ATE177099T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17503493A 1993-12-29 1993-12-29

Publications (1)

Publication Number Publication Date
ATE177099T1 true ATE177099T1 (de) 1999-03-15

Family

ID=22638565

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94931148T ATE177099T1 (de) 1993-12-29 1994-11-14 Diazabicyclische neurokinin antagonisten

Country Status (26)

Country Link
US (2) US5854239A (de)
EP (1) EP0737194B1 (de)
JP (1) JP2895630B2 (de)
KR (1) KR100197454B1 (de)
CN (1) CN1046515C (de)
AT (1) ATE177099T1 (de)
AU (1) AU699465B2 (de)
BR (1) BR9408450A (de)
CA (1) CA2180263C (de)
CO (1) CO4230019A1 (de)
CZ (1) CZ282567B6 (de)
DE (1) DE69416869T2 (de)
DK (1) DK0737194T3 (de)
ES (1) ES2127946T3 (de)
FI (1) FI108296B (de)
GR (1) GR3029853T3 (de)
HU (1) HUT74682A (de)
IL (1) IL112118A (de)
NO (1) NO305600B1 (de)
NZ (1) NZ274915A (de)
PE (1) PE49395A1 (de)
PL (1) PL179435B1 (de)
RU (1) RU2124014C1 (de)
TW (1) TW369526B (de)
WO (1) WO1995018129A1 (de)
ZA (1) ZA9410339B (de)

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FR2848210B1 (fr) * 2002-12-06 2007-10-19 Aventis Pharma Sa Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases
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PL179435B1 (pl) * 1993-12-29 2000-09-29 Pfizer Diazabicykliczni antagonisci neurokininy PL

Also Published As

Publication number Publication date
GR3029853T3 (en) 1999-07-30
DE69416869D1 (de) 1999-04-08
HU9601790D0 (en) 1996-09-30
RU2124014C1 (ru) 1998-12-27
CO4230019A1 (es) 1995-10-19
NO962742D0 (no) 1996-06-28
AU8002194A (en) 1995-07-17
JPH09500904A (ja) 1997-01-28
CZ188696A3 (en) 1996-10-16
US5854239A (en) 1998-12-29
PL179435B1 (pl) 2000-09-29
IL112118A0 (en) 1995-03-15
DE69416869T2 (de) 1999-07-01
ES2127946T3 (es) 1999-05-01
ZA9410339B (en) 1996-06-28
NO962742L (no) 1996-06-28
PE49395A1 (es) 1996-01-06
CN1046515C (zh) 1999-11-17
PL315193A1 (en) 1996-10-14
AU699465B2 (en) 1998-12-03
US6110919A (en) 2000-08-29
FI946140A0 (fi) 1994-12-28
IL112118A (en) 1998-10-30
EP0737194B1 (de) 1999-03-03
EP0737194A1 (de) 1996-10-16
NO305600B1 (no) 1999-06-28
KR100197454B1 (ko) 1999-06-15
HUT74682A (en) 1997-01-28
FI946140A (fi) 1995-06-30
FI108296B (fi) 2001-12-31
JP2895630B2 (ja) 1999-05-24
CZ282567B6 (cs) 1997-08-13
DK0737194T3 (da) 1999-09-27
BR9408450A (pt) 1997-08-05
CA2180263C (en) 2000-05-16
CN1139434A (zh) 1997-01-01
WO1995018129A1 (en) 1995-07-06
NZ274915A (en) 1997-11-24
TW369526B (en) 1999-09-11

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