ATA813278A - METHOD FOR PRODUCING SALTS OF N- (PHOSPHONOACETYL) -L-ASPARAGIC ACID (PALA) AND THEIR SOLVATES - Google Patents

METHOD FOR PRODUCING SALTS OF N- (PHOSPHONOACETYL) -L-ASPARAGIC ACID (PALA) AND THEIR SOLVATES

Info

Publication number
ATA813278A
ATA813278A AT0813278A AT813278A ATA813278A AT A813278 A ATA813278 A AT A813278A AT 0813278 A AT0813278 A AT 0813278A AT 813278 A AT813278 A AT 813278A AT A813278 A ATA813278 A AT A813278A
Authority
AT
Austria
Prior art keywords
phosphonoacetyl
pala
solvates
asparagic acid
producing salts
Prior art date
Application number
AT0813278A
Other languages
German (de)
Other versions
AT374485B (en
Original Assignee
Starks Ass
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Starks Ass filed Critical Starks Ass
Publication of ATA813278A publication Critical patent/ATA813278A/en
Application granted granted Critical
Publication of AT374485B publication Critical patent/AT374485B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3808Acyclic saturated acids which can have further substituents on alkyl
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/28Phosphorus compounds with one or more P—C bonds
    • C07F9/38Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40Esters thereof
    • C07F9/4003Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006Esters of acyclic acids which can have further substituents on alkyl

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT0813278A 1977-11-14 1978-11-14 METHOD FOR PRODUCING SALTS OF N- (PHOSPHONOACETYL) -L-ASPARAGIC ACID (PALA) AND THEIR SOLVATES AT374485B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US85138277A 1977-11-14 1977-11-14

Publications (2)

Publication Number Publication Date
ATA813278A true ATA813278A (en) 1983-09-15
AT374485B AT374485B (en) 1984-04-25

Family

ID=25310650

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0813278A AT374485B (en) 1977-11-14 1978-11-14 METHOD FOR PRODUCING SALTS OF N- (PHOSPHONOACETYL) -L-ASPARAGIC ACID (PALA) AND THEIR SOLVATES

Country Status (14)

Country Link
JP (1) JPS5492920A (en)
AT (1) AT374485B (en)
AU (1) AU520966B2 (en)
CA (1) CA1110266A (en)
CH (1) CH636595A5 (en)
DE (1) DE2849396A1 (en)
DK (1) DK149134C (en)
FI (1) FI65261C (en)
FR (1) FR2408617A1 (en)
GB (2) GB2008118B (en)
GR (1) GR65247B (en)
NL (1) NL7811252A (en)
NZ (1) NZ188909A (en)
SE (1) SE439774B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4284579A (en) * 1979-07-17 1981-08-18 The United States Of America As Represented By The Of The Department Of Health & Human Services (N-Phosphonacetyl-L-aspartato)(1,2-diaminocyclchexane)platinum(II) or alkali metal salt

Also Published As

Publication number Publication date
GR65247B (en) 1980-07-31
DK506278A (en) 1979-05-15
GB2008118B (en) 1982-08-04
NL7811252A (en) 1979-05-16
DK149134B (en) 1986-02-10
FI65261B (en) 1983-12-30
AT374485B (en) 1984-04-25
SE439774B (en) 1985-07-01
FI65261C (en) 1984-04-10
GB2051070A (en) 1981-01-14
CA1110266A (en) 1981-10-06
DK149134C (en) 1986-07-14
DE2849396A1 (en) 1979-05-17
AU4152878A (en) 1979-05-24
GB2051070B (en) 1982-08-04
NZ188909A (en) 1980-10-08
GB2008118A (en) 1979-05-31
CH636595A5 (en) 1983-06-15
FR2408617A1 (en) 1979-06-08
AU520966B2 (en) 1982-03-11
FI783467A (en) 1979-05-15
JPS5492920A (en) 1979-07-23
SE7811736L (en) 1979-05-15
FR2408617B1 (en) 1983-11-18

Similar Documents

Publication Publication Date Title
AT363457B (en) METHOD FOR PRODUCING NEW SUBSTITUTED 1- (3-AMINOSULFONYLPHENYL) -2-ALKYLAMINOAETHANOLS AND THEIR ACID ADDITION SALTS
ATA921778A (en) METHOD FOR PRODUCING NEW DERIVATIVES OF HYDROXYCARBONYLPHOSPHONIC ACID, AND THEIR SALTS AND OPTICAL ANTIPODES
AT361937B (en) METHOD FOR PRODUCING NEW 4-ACYL-AMINOPHENYL-AETHANOLAMINES AND THEIR ACID ADDITION SALTS
AT359522B (en) METHOD FOR PRODUCING NEW 6-AMINO-ALKYLAMINOURACILES AND THEIR ACID ADDITION SALTS
AT365175B (en) METHOD FOR PRODUCING 5 (6) -THIOBENZIMIDAZOLE DERIVATIVES AND THEIR SALTS
AT366666B (en) METHOD FOR PRODUCING NEW AMIDINOSULPHONE ACID DERIVATIVES AND THEIR SALTS
AT354436B (en) METHOD FOR PRODUCING NEW 2-BROMO-6-FLUOR-N-2-IMIDAZOLIDINYLIDENE-BENZAMINE AND ITS ACID ADDITION SALTS
AT375363B (en) METHOD FOR PRODUCING 1- (8-CHINOLYL) 2-PYRROLIDINONE AND ITS ACID ADDITION SALTS
AT370421B (en) METHOD FOR THE PRODUCTION OF ALCALOIDS OF THE LEUROSIN TYPE AND THEIR SALTS
AT363065B (en) METHOD FOR PRODUCING NEW QUATERNAUS AMMONIUM SALTS OF PHENYLPROPYLAMINES AND PHENYLBUTYLAMINES
AT363923B (en) METHOD FOR PRODUCING NEW 8-AMINO-ALKYLTETRACYCLONONANS AND THEIR ACID ADDITION SALTS
AT361904B (en) METHOD FOR PRODUCING NEW 3-ANILINO-AETHYLAMINO-2-HYDROXY-1-PHENOXYPROPANES AND THEIR ACID ADDITION SALTS
AT374485B (en) METHOD FOR PRODUCING SALTS OF N- (PHOSPHONOACETYL) -L-ASPARAGIC ACID (PALA) AND THEIR SOLVATES
AT360033B (en) METHOD FOR PRODUCING NEW TETRAHYDRO- -S-TRIAZINTHIONS AND THEIR ACID ADDITION SALTS
AT359644B (en) METHOD FOR PRODUCING NEW OXIMES OF 7-AMINOTHIAZOLYLACETAMIDOCEPHALOSPORANIC ACID AND THEIR SALTS
ATA398678A (en) METHOD FOR PRODUCING NEW 4-ACETAMIDOPHENYL-ALPHA- (2-METHYL-IND (EN / OL) - -3-YL) -ACETATES AND THEIR ACID ADDITION SALTS
AT366042B (en) METHOD FOR PRODUCING NEW 2-METHYLTHIO -6-FLUOR-9- (1-METHYL-4-PIPERIDYLIDEN) -THIOXANTH N AND ITS NON-TOXIC ACID ADDITION SALTS
AT369740B (en) METHOD FOR PRODUCING NEW THIODIBENCE THIEPINES AND THEIR ACID ADDITION SALTS
ATA501078A (en) METHOD FOR PRODUCING BENZYLIDE AMINO-ALKANIC ACID AMIDES
AT365559B (en) METHOD FOR PRODUCING AMINOPROPANDIOLMONO ETHERS AND THEIR ACID ADDITION SALTS
AT357692B (en) METHOD FOR PRODUCING 4-DESACETOXY- -VINBLASTIN AND ITS ACID ADDITION SALTS
ATA59280A (en) METHOD FOR PRODUCING NEW 3-ANILINOAETHYLAMINO-2-HYDROXY-1-PHENOXYPROPANES AND THEIR ACID ADDITION SALTS
ATA330380A (en) METHOD FOR PRODUCING N-DESMETHYL-N-FORMYL-LEUROSIN AND ITS SALTS
ATA148580A (en) METHOD FOR PRODUCING NEW 4-ACYL-AMINOPHENYL-AETHANOLAMINES AND THEIR ACID ADDITION SALTS
AT364365B (en) METHOD FOR PRODUCING NEW SUBSTITUTED OCTAHYDROPYRAZINOPYRIMIDINONES AND THEIR ACID ADDITION SALTS