AT348981B - Verfahren zur herstellung neuer 5-sulfonamido- 2-amino-benzoesaeurederivate sowie ihrer saeureadditonssalze - Google Patents
Verfahren zur herstellung neuer 5-sulfonamido- 2-amino-benzoesaeurederivate sowie ihrer saeureadditonssalzeInfo
- Publication number
- AT348981B AT348981B AT180277A AT180277A AT348981B AT 348981 B AT348981 B AT 348981B AT 180277 A AT180277 A AT 180277A AT 180277 A AT180277 A AT 180277A AT 348981 B AT348981 B AT 348981B
- Authority
- AT
- Austria
- Prior art keywords
- sulfonamido
- amino
- new
- production
- benzoic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19762611705 DE2611705A1 (de) | 1976-03-18 | 1976-03-18 | N-5-(nitrofurfuryliden-)-1-amino- hydantoin enthaltende kristalloesungsmittel |
HU76GO00001334A HU172949B (hu) | 1976-03-18 | 1976-03-18 | Sposob poluchenija novykh proizvodnykh sul'fonamido-benzojnoj kisloty |
Publications (2)
Publication Number | Publication Date |
---|---|
ATA180277A ATA180277A (de) | 1978-08-15 |
AT348981B true AT348981B (de) | 1979-03-12 |
Family
ID=25770228
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT180277A AT348981B (de) | 1976-03-18 | 1977-03-16 | Verfahren zur herstellung neuer 5-sulfonamido- 2-amino-benzoesaeurederivate sowie ihrer saeureadditonssalze |
Country Status (9)
Country | Link |
---|---|
US (1) | US4244871A (de) |
JP (1) | JPS52136146A (de) |
AT (1) | AT348981B (de) |
CA (1) | CA1092111A (de) |
DE (2) | DE2611705A1 (de) |
FR (1) | FR2344531A1 (de) |
GB (1) | GB1561243A (de) |
NL (1) | NL7702991A (de) |
SE (1) | SE7703068L (de) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS58192820A (ja) * | 1982-05-06 | 1983-11-10 | Mochida Pharmaceut Co Ltd | 抗ウイルス作用を有する医薬組成物 |
IT1176613B (it) * | 1984-08-14 | 1987-08-18 | Ravizza Spa | Derivati piperazinici farmacologicamente attivi e processo per la loro preparazione |
JPS61134382A (ja) * | 1984-12-04 | 1986-06-21 | Kyorin Pharmaceut Co Ltd | 新規なスルファモイル安息香酸誘導体およびその製造法 |
JP2001508811A (ja) * | 1998-04-20 | 2001-07-03 | 藤沢薬品工業株式会社 | cGMP−ホスホジエステラーゼ阻害剤としてのアントラニル酸誘導体 |
BRPI0413536B8 (pt) * | 2003-09-09 | 2021-05-25 | Hoffmann La Roche | derivados de 1-benzoil-piperazina, seu uso e medicamento que os compreende |
BRPI0414209B8 (pt) * | 2003-09-09 | 2021-05-25 | Hoffmann La Roche | derivados de 1-(2-amino-benzol)-piperazina, seus processos de preparação e seu uso, e medicamento |
CA2589192C (en) * | 2004-12-09 | 2014-04-22 | F. Hoffmann-La Roche Ag | Phenyl-piperazin methanone derivatives |
WO2006063709A1 (en) * | 2004-12-15 | 2006-06-22 | F.Hoffmann-La Roche Ag | Bi- and tricyclic substituted phenyl methanones as glycine transporter i (glyt-1) inhibitors for the treatment of alzheimer’s disease |
US7485637B2 (en) * | 2005-01-04 | 2009-02-03 | Hoffmann-La Roche Inc. | Benzoyl-tetrahydropiperidine derivatives |
JP2008526795A (ja) * | 2005-01-06 | 2008-07-24 | エフ.ホフマン−ラ ロシュ アーゲー | 神経障害および神経精神疾患を処置するためのグリシントランスポータ1(glyt−1)阻害物質としての、スルファニル置換フェニルメタノン |
DE602005022113D1 (de) * | 2005-01-07 | 2010-08-12 | Hoffmann La Roche | Phenyl)methanon-derivate als glycin-transporter 1 (glyt-1) hemmer zur behandlung von neurologischen und neuropsychiatrischen erkrankungen |
BRPI0606730A2 (pt) * | 2005-01-18 | 2009-07-14 | Hoffmann La Roche | derivados de fenil metanona 2,5-di-substituìdos como inibidores do transportador de glicina 1 (glyt-1) para o tratamento de distúbios neurológicos e neuropsiquiátricos |
RU2007126951A (ru) * | 2005-01-26 | 2009-03-10 | Ф.Хоффманн-Ля Рош Аг (Ch) | Производные фенилметанона и их применение в качестве ингибиторов переносчика глицина 1 |
KR100928599B1 (ko) * | 2005-02-07 | 2009-11-26 | 에프. 호프만-라 로슈 아게 | 글라이신 트랜스포터 1의 저해제로서의 헤테로환상 치환된페닐 메탄온 |
GB0505086D0 (en) * | 2005-03-11 | 2005-04-20 | Glaxo Group Ltd | Compounds |
MX2011000051A (es) * | 2008-07-07 | 2011-07-28 | Fasgen Inc | Nuevos compuestos, composiciones farmaceuticas que contienen los mismos, metodos para usar los mismos, y metodos para preparar los mismos. |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2910488A (en) * | 1958-01-22 | 1959-10-27 | Merck & Co Inc | Aniline derivatives |
US3346568A (en) * | 1961-09-14 | 1967-10-10 | Ciba Geigy Corp | 2-amino-5-sulfamyl-benzoic acid hydrazides |
FR1403935A (fr) * | 1963-06-05 | 1965-06-25 | Ciba Geigy | Nouveaux amides d'acides anthraniliques |
US3839321A (en) * | 1966-07-21 | 1974-10-01 | Smithkline Corp | 5-sulfamoyl-n-(2-substituted-ethyl) anthranilic acids |
US3522274A (en) * | 1967-05-24 | 1970-07-28 | American Home Prod | 2,3-dihydro-1-alkyl-7-sulfamoyl-4,1-benzoxazepin-5(1h)-ones |
US3843662A (en) * | 1971-12-09 | 1974-10-22 | Pfizer | 2-halo-5-(substituted piperidino sulfonyl)benzoic acids |
DE2232457A1 (de) * | 1972-07-01 | 1974-01-10 | Boehringer Mannheim Gmbh | Neue 3-alkyl-4-sulfamoylanilinderivate |
DE2423847A1 (de) * | 1973-05-28 | 1975-01-02 | Ciba Geigy Ag | Neue sulfamoylbenzoesaeureamide |
CH590261A5 (de) * | 1973-07-10 | 1977-07-29 | Ciba Geigy Ag |
-
1976
- 1976-03-18 DE DE19762611705 patent/DE2611705A1/de active Pending
-
1977
- 1977-03-16 FR FR7707839A patent/FR2344531A1/fr active Granted
- 1977-03-16 AT AT180277A patent/AT348981B/de not_active IP Right Cessation
- 1977-03-17 CA CA274,162A patent/CA1092111A/en not_active Expired
- 1977-03-17 SE SE7703068A patent/SE7703068L/xx not_active Application Discontinuation
- 1977-03-17 GB GB11472/77A patent/GB1561243A/en not_active Expired
- 1977-03-18 NL NL7702991A patent/NL7702991A/xx not_active Application Discontinuation
- 1977-03-18 JP JP2938777A patent/JPS52136146A/ja active Pending
- 1977-03-18 DE DE19772712023 patent/DE2712023A1/de not_active Withdrawn
-
1979
- 1979-07-12 US US06/058,363 patent/US4244871A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
ATA180277A (de) | 1978-08-15 |
GB1561243A (en) | 1980-02-13 |
US4244871A (en) | 1981-01-13 |
DE2712023A1 (de) | 1977-10-06 |
CA1092111A (en) | 1980-12-23 |
FR2344531A1 (fr) | 1977-10-14 |
SE7703068L (sv) | 1977-09-19 |
JPS52136146A (en) | 1977-11-14 |
FR2344531B1 (de) | 1980-04-04 |
DE2611705A1 (de) | 1977-09-22 |
NL7702991A (nl) | 1977-09-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ELJ | Ceased due to non-payment of the annual fee | ||
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |