AR231537A1 - Procedimiento para la preparacion de derivados de la piridazina - Google Patents

Procedimiento para la preparacion de derivados de la piridazina

Info

Publication number
AR231537A1
AR231537A1 AR290279A AR29027982A AR231537A1 AR 231537 A1 AR231537 A1 AR 231537A1 AR 290279 A AR290279 A AR 290279A AR 29027982 A AR29027982 A AR 29027982A AR 231537 A1 AR231537 A1 AR 231537A1
Authority
AR
Argentina
Prior art keywords
piridazine
derivatives
procedure
preparation
Prior art date
Application number
AR290279A
Other languages
English (en)
Spanish (es)
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Application granted granted Critical
Publication of AR231537A1 publication Critical patent/AR231537A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/26Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
    • C07D237/30Phthalazines
    • C07D237/34Phthalazines with nitrogen atoms directly attached to carbon atoms of the nitrogen-containing ring, e.g. hydrazine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D237/00Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR290279A 1981-08-11 1982-08-10 Procedimiento para la preparacion de derivados de la piridazina AR231537A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8115546A FR2511366A1 (fr) 1981-08-11 1981-08-11 Nouveaux derives de la pyridazine, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent

Publications (1)

Publication Number Publication Date
AR231537A1 true AR231537A1 (es) 1984-12-28

Family

ID=9261385

Family Applications (1)

Application Number Title Priority Date Filing Date
AR290279A AR231537A1 (es) 1981-08-11 1982-08-10 Procedimiento para la preparacion de derivados de la piridazina

Country Status (30)

Country Link
US (1) US4710499A (de)
EP (1) EP0073161B1 (de)
JP (1) JPS5838263A (de)
KR (1) KR880002711B1 (de)
AR (1) AR231537A1 (de)
AT (1) ATE23042T1 (de)
AU (1) AU579570B2 (de)
CA (1) CA1179347A (de)
CS (1) CS239929B2 (de)
DD (1) DD202550A5 (de)
DE (1) DE3273893D1 (de)
DK (1) DK148596C (de)
EG (1) EG15749A (de)
ES (1) ES514887A0 (de)
FI (1) FI72970C (de)
FR (1) FR2511366A1 (de)
GR (1) GR76236B (de)
HU (1) HU189608B (de)
IE (1) IE53493B1 (de)
IL (1) IL66424A (de)
MA (1) MA19559A1 (de)
NO (1) NO158871C (de)
NZ (1) NZ201553A (de)
OA (1) OA07179A (de)
PH (1) PH18921A (de)
PL (1) PL137200B1 (de)
PT (1) PT75372B (de)
SU (1) SU1356960A3 (de)
YU (1) YU171682A (de)
ZA (1) ZA825515B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2539741A1 (fr) * 1983-01-21 1984-07-27 Sanofi Sa Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent
US5001125A (en) * 1984-03-26 1991-03-19 Janssen Pharmaceutica N.V. Anti-virally active pyridazinamines
JPS60218377A (ja) * 1984-04-16 1985-11-01 Mitsubishi Yuka Yakuhin Kk 4−フエニルフタラジン誘導体及びそれを有効成分とする循環改善剤
DE3664772D1 (en) * 1985-01-14 1989-09-07 Boehringer Ingelheim Kg 12-amino pyridazinoû4',5':3,4¨pyrroloû2,1-a¨isoquinolines, process for their preparation and use
US5106973A (en) * 1987-11-23 1992-04-21 Janssen Pharmaceutica N.V. Pyridzainamine derivatives
DK0628550T3 (da) * 1993-06-08 1998-09-28 Vertex Pharma Pyridazin som interleukin-1 beta-omdannede enzyminhibitorer
US20100210590A1 (en) * 1995-09-27 2010-08-19 Northwestern University Compositions and treatments for seizure-related disorders
GB9707693D0 (en) * 1997-04-16 1997-06-04 Smithkline Beecham Plc Novel method of treatment
US20030176437A1 (en) * 2001-08-31 2003-09-18 D.M. Watterson Anti-inflammatory and protein kinase inhibitor compositions and related methods for downregulation of detrimental cellular responses and inhibition of cell death
EP1812007B1 (de) * 2004-11-02 2011-09-07 Northwestern University Pyridazinverbindungen und verfahren
ES2441718T3 (es) 2004-11-02 2014-02-06 Northwestern University Compuestos de piridazina, composiciones y métodos
US20090325973A1 (en) * 2006-04-28 2009-12-31 Watterson D Martin Formulations containing pyridazine compounds
EP2015750A2 (de) * 2006-04-28 2009-01-21 Northwestern University Zusammensetzungen und behandlungen mit pyridazinverbindungen und cholisterinasehemmern
CA2650704A1 (en) * 2006-04-28 2007-11-08 Northwestern University Salts of pyridazine compounds
JP2010520223A (ja) * 2007-03-02 2010-06-10 ノースウェスタン ユニバーシティ 発作関連障害のための組成物および方法
WO2024148148A1 (en) * 2023-01-04 2024-07-11 The Trustees Of Columbia University In The City Of New York Pyridazine based small molecule inhibitor of cognitive impairment

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1345880A (en) * 1971-06-18 1974-02-06 Cepbepe Pyridazine derivatives
FR2473522A1 (fr) * 1980-01-16 1981-07-17 Synthelabo Nouveaux derives substitues de dihydro-2,3 imidazo(1,2-b)pyridazines et les medicaments, utiles notamment comme antidepresseurs, qui en contiennent

Also Published As

Publication number Publication date
ATE23042T1 (de) 1986-11-15
PT75372B (en) 1984-12-10
IL66424A (en) 1985-10-31
ES8305736A1 (es) 1983-04-16
NO158871B (no) 1988-08-01
US4710499A (en) 1987-12-01
KR840001147A (ko) 1984-03-28
DK358782A (da) 1983-02-12
OA07179A (fr) 1984-04-30
EP0073161A1 (de) 1983-03-02
CS239929B2 (en) 1986-01-16
PT75372A (en) 1982-09-01
SU1356960A3 (ru) 1987-11-30
JPS5838263A (ja) 1983-03-05
EG15749A (en) 1986-09-30
FR2511366A1 (fr) 1983-02-18
PH18921A (en) 1985-11-11
AU8702982A (en) 1983-05-12
AU579570B2 (en) 1988-12-01
NO158871C (no) 1988-11-09
EP0073161B1 (de) 1986-10-22
PL137200B1 (en) 1986-05-31
DD202550A5 (de) 1983-09-21
IL66424A0 (en) 1982-11-30
PL237836A1 (en) 1983-02-28
FI822768A0 (fi) 1982-08-09
IE53493B1 (en) 1988-11-23
FI72970C (fi) 1987-08-10
DK148596B (da) 1985-08-12
GR76236B (de) 1984-08-04
ZA825515B (en) 1983-06-29
JPH0456032B2 (de) 1992-09-07
IE821822L (en) 1983-02-11
CA1179347A (en) 1984-12-11
HU189608B (en) 1986-07-28
DK148596C (da) 1986-01-13
DE3273893D1 (en) 1986-11-27
KR880002711B1 (ko) 1988-12-26
YU171682A (en) 1985-03-20
MA19559A1 (fr) 1983-04-01
NZ201553A (en) 1985-08-16
NO822717L (no) 1983-02-14
FR2511366B1 (de) 1984-12-14
FI822768L (fi) 1983-02-11
FI72970B (fi) 1987-04-30
ES514887A0 (es) 1983-04-16

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