AR228442A1 - Procedimiento para la preparacion de 1-(8-quinolil)-2-pirrolidinona - Google Patents
Procedimiento para la preparacion de 1-(8-quinolil)-2-pirrolidinonaInfo
- Publication number
- AR228442A1 AR228442A1 AR283420A AR28342080A AR228442A1 AR 228442 A1 AR228442 A1 AR 228442A1 AR 283420 A AR283420 A AR 283420A AR 28342080 A AR28342080 A AR 28342080A AR 228442 A1 AR228442 A1 AR 228442A1
- Authority
- AR
- Argentina
- Prior art keywords
- pirrolidinone
- quinolyl
- procedure
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/40—Nitrogen atoms attached in position 8
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pain & Pain Management (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB7941409 | 1979-11-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR228442A1 true AR228442A1 (es) | 1983-03-15 |
Family
ID=10509524
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR283420A AR228442A1 (es) | 1979-11-30 | 1980-11-28 | Procedimiento para la preparacion de 1-(8-quinolil)-2-pirrolidinona |
Country Status (18)
Country | Link |
---|---|
US (1) | US4366158A (es) |
EP (1) | EP0030023A3 (es) |
JP (1) | JPS5699475A (es) |
KR (1) | KR830004293A (es) |
AR (1) | AR228442A1 (es) |
AT (1) | AT375363B (es) |
AU (1) | AU6495080A (es) |
CA (1) | CA1156235A (es) |
DK (1) | DK506480A (es) |
ES (1) | ES497242A0 (es) |
FI (1) | FI803704L (es) |
GB (1) | GB2063868B (es) |
GR (1) | GR71918B (es) |
HU (1) | HU185224B (es) |
IL (1) | IL61580A (es) |
IT (1) | IT1221040B (es) |
NZ (1) | NZ195688A (es) |
ZA (1) | ZA807467B (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MXPA06000795A (es) | 2003-07-22 | 2006-08-23 | Arena Pharm Inc | Derivados de diaril y arilheteroaril urea como moduladores del receptor 5-ht2a de serotonina utiles para la profilaxis y tratamiento de desordenes relacionados con el mismo. |
GB0507198D0 (en) * | 2005-04-08 | 2005-05-18 | Sb Pharmco Inc | Process for preparing bicyclic compounds |
GB0519758D0 (en) * | 2005-09-28 | 2005-11-09 | Glaxo Group Ltd | Novel process |
EP2508177A1 (en) | 2007-12-12 | 2012-10-10 | Glaxo Group Limited | Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
WO2009123714A2 (en) | 2008-04-02 | 2009-10-08 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
WO2010062321A1 (en) | 2008-10-28 | 2010-06-03 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2h-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)-urea and crystalline forms related thereto |
EP4119141A1 (en) | 2015-06-12 | 2023-01-18 | Axovant Sciences GmbH | Nelotanserin for the prophylaxis and treatment of rem sleep behavior disorder |
CA2992518A1 (en) | 2015-07-15 | 2017-01-19 | Axovant Sciences Gmbh | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of hallucinations associated with a neurodegenerative disease |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4143151A (en) * | 1978-07-03 | 1979-03-06 | The Dow Chemical Company | Method for treating hyperglycemia in mammals using arylamino benzoic acids |
-
1980
- 1980-11-24 US US06/209,426 patent/US4366158A/en not_active Expired - Lifetime
- 1980-11-26 GB GB8037872A patent/GB2063868B/en not_active Expired
- 1980-11-28 IT IT50277/80A patent/IT1221040B/it active
- 1980-11-28 AU AU64950/80A patent/AU6495080A/en not_active Abandoned
- 1980-11-28 ZA ZA00807467A patent/ZA807467B/xx unknown
- 1980-11-28 NZ NZ195688A patent/NZ195688A/en unknown
- 1980-11-28 HU HU802850A patent/HU185224B/hu unknown
- 1980-11-28 FI FI803704A patent/FI803704L/fi not_active Application Discontinuation
- 1980-11-28 KR KR1019800004552A patent/KR830004293A/ko unknown
- 1980-11-28 JP JP16791880A patent/JPS5699475A/ja active Pending
- 1980-11-28 AT AT0582780A patent/AT375363B/de not_active IP Right Cessation
- 1980-11-28 DK DK506480A patent/DK506480A/da not_active Application Discontinuation
- 1980-11-28 CA CA000365722A patent/CA1156235A/en not_active Expired
- 1980-11-28 ES ES497242A patent/ES497242A0/es active Granted
- 1980-11-28 AR AR283420A patent/AR228442A1/es active
- 1980-11-28 IL IL61580A patent/IL61580A/xx unknown
- 1980-11-28 EP EP80107463A patent/EP0030023A3/en not_active Ceased
- 1980-11-28 GR GR63493A patent/GR71918B/el unknown
Also Published As
Publication number | Publication date |
---|---|
ES8203882A1 (es) | 1982-04-01 |
IT8050277A0 (it) | 1980-11-28 |
EP0030023A2 (en) | 1981-06-10 |
GR71918B (es) | 1983-08-17 |
US4366158A (en) | 1982-12-28 |
ES497242A0 (es) | 1982-04-01 |
KR830004293A (ko) | 1983-07-09 |
IL61580A0 (en) | 1980-12-31 |
HU185224B (en) | 1984-12-28 |
ZA807467B (en) | 1982-07-28 |
ATA582780A (de) | 1983-12-15 |
IL61580A (en) | 1984-06-29 |
IT1221040B (it) | 1990-06-21 |
CA1156235A (en) | 1983-11-01 |
JPS5699475A (en) | 1981-08-10 |
AT375363B (de) | 1984-07-25 |
AU6495080A (en) | 1981-06-04 |
FI803704L (fi) | 1981-05-31 |
GB2063868A (en) | 1981-06-10 |
NZ195688A (en) | 1984-09-28 |
GB2063868B (en) | 1984-02-29 |
EP0030023A3 (en) | 1981-09-02 |
DK506480A (da) | 1981-05-31 |
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