AR220539A1 - Procedimiento para obtener 7 beta-aril-malonamido-7 alpha-metoxi-3-(tiadiazoliltio)1-oxadetiacefalosporinas y sus sales - Google Patents

Procedimiento para obtener 7 beta-aril-malonamido-7 alpha-metoxi-3-(tiadiazoliltio)1-oxadetiacefalosporinas y sus sales

Info

Publication number
AR220539A1
AR220539A1 AR273406A AR27340678A AR220539A1 AR 220539 A1 AR220539 A1 AR 220539A1 AR 273406 A AR273406 A AR 273406A AR 27340678 A AR27340678 A AR 27340678A AR 220539 A1 AR220539 A1 AR 220539A1
Authority
AR
Argentina
Prior art keywords
tiadiazoliltio
oxadetiacefalosporinas
malonamido
metoxi
aril
Prior art date
Application number
AR273406A
Other languages
English (en)
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Application granted granted Critical
Publication of AR220539A1 publication Critical patent/AR220539A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D505/00Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AR273406A 1977-08-25 1978-08-23 Procedimiento para obtener 7 beta-aril-malonamido-7 alpha-metoxi-3-(tiadiazoliltio)1-oxadetiacefalosporinas y sus sales AR220539A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP52102261A JPS609718B2 (ja) 1977-08-25 1977-08-25 チアジアゾリルチオセフアロスポリン類縁抗生物質

Publications (1)

Publication Number Publication Date
AR220539A1 true AR220539A1 (es) 1980-11-14

Family

ID=14322642

Family Applications (1)

Application Number Title Priority Date Filing Date
AR273406A AR220539A1 (es) 1977-08-25 1978-08-23 Procedimiento para obtener 7 beta-aril-malonamido-7 alpha-metoxi-3-(tiadiazoliltio)1-oxadetiacefalosporinas y sus sales

Country Status (34)

Country Link
US (1) US4201782A (es)
JP (1) JPS609718B2 (es)
AR (1) AR220539A1 (es)
AT (1) AT361121B (es)
AU (1) AU517618B2 (es)
BE (1) BE869955A (es)
BG (1) BG34338A3 (es)
CA (1) CA1101417A (es)
CH (1) CH637396A5 (es)
CS (1) CS203927B2 (es)
DD (1) DD137230A5 (es)
DE (1) DE2837264A1 (es)
DK (1) DK372878A (es)
ES (1) ES472817A1 (es)
FI (1) FI65432C (es)
FR (1) FR2401165A1 (es)
GB (1) GB1576796A (es)
GR (1) GR70260B (es)
HU (1) HU177900B (es)
IE (1) IE47630B1 (es)
IL (1) IL55429A0 (es)
IT (1) IT1118098B (es)
MX (1) MX5328E (es)
NL (1) NL190554C (es)
NO (1) NO782866L (es)
NZ (1) NZ188173A (es)
PH (1) PH17508A (es)
PL (1) PL110656B1 (es)
PT (1) PT68434A (es)
RO (1) RO75070A (es)
SE (1) SE452010B (es)
SU (1) SU812182A3 (es)
YU (1) YU43999B (es)
ZA (1) ZA784753B (es)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4259485A (en) * 1979-04-24 1981-03-31 Eli Lilly And Company Crystallization process
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
DE3373475D1 (en) * 1982-12-14 1987-10-15 Beecham Group Plc Process for the preparation of beta-lactam compounds
JPS60123490A (ja) * 1983-12-07 1985-07-02 Shionogi & Co Ltd マロニルオキサセフェムカルボン酸誘導体
US6013835A (en) * 1995-06-07 2000-01-11 Hfm International, Inc. Method and apparatus for preparing purified terephthalic acid
US6197794B1 (en) 1998-01-08 2001-03-06 Celltech Therapeutics Limited Phenylalanine derivatives
US6329372B1 (en) 1998-01-27 2001-12-11 Celltech Therapeutics Limited Phenylalanine derivatives
ATE273273T1 (de) 1998-02-26 2004-08-15 Celltech Therapeutics Ltd Phenylalaninderivate als inhibitoren von alpha4 integrinen
GB9805655D0 (en) 1998-03-16 1998-05-13 Celltech Therapeutics Ltd Chemical compounds
US6521626B1 (en) 1998-03-24 2003-02-18 Celltech R&D Limited Thiocarboxamide derivatives
GB9811159D0 (en) 1998-05-22 1998-07-22 Celltech Therapeutics Ltd Chemical compounds
GB9811969D0 (en) 1998-06-03 1998-07-29 Celltech Therapeutics Ltd Chemical compounds
GB9812088D0 (en) 1998-06-05 1998-08-05 Celltech Therapeutics Ltd Chemical compounds
GB9814414D0 (en) 1998-07-03 1998-09-02 Celltech Therapeutics Ltd Chemical compounds
GB9821061D0 (en) 1998-09-28 1998-11-18 Celltech Therapeutics Ltd Chemical compounds
GB9821222D0 (en) 1998-09-30 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9821406D0 (en) * 1998-10-01 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9825652D0 (en) 1998-11-23 1999-01-13 Celltech Therapeutics Ltd Chemical compounds
US6518283B1 (en) 1999-05-28 2003-02-11 Celltech R&D Limited Squaric acid derivatives
US6534513B1 (en) 1999-09-29 2003-03-18 Celltech R&D Limited Phenylalkanoic acid derivatives
US6455539B2 (en) 1999-12-23 2002-09-24 Celltech R&D Limited Squaric acid derivates
EP1332132B1 (en) 2000-04-17 2007-10-10 UCB Pharma, S.A. Enamine derivatives as cell adhesion molecules
US6545013B2 (en) 2000-05-30 2003-04-08 Celltech R&D Limited 2,7-naphthyridine derivatives
US6403608B1 (en) 2000-05-30 2002-06-11 Celltech R&D, Ltd. 3-Substituted isoquinolin-1-yl derivatives
AU2001267753A1 (en) 2000-07-07 2002-01-21 Celltech R And D Limited Squaric acid derivatives containing a bicyclic heteroaromatic ring as integrin antagonists
US6649756B2 (en) * 2000-07-13 2003-11-18 Wyeth, Five Giralda Farms Process improvement in the preparation of (4r, 5s, 6s)-3-[[(2r,3r)-2-[[[(s)-2-amino-3-methyl-1-oxobutyl]amino]methyl]tetrahydro-3-furanyl]thio]-6-[(r)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
AU2001275724A1 (en) 2000-08-02 2002-02-13 Celltech R&D Limited 3-substituted isoquinolin-1-yl derivatives
CN102827191B (zh) * 2012-09-24 2015-03-11 浙江东邦药业有限公司 一种氧头孢类化合物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL178005C (nl) * 1972-11-06 1986-01-02 Merck & Co Inc Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
US4045438A (en) * 1975-10-24 1977-08-30 Yeda Research And Development Co. Ltd. Cephalosporin antibiotics
US4031083A (en) * 1975-10-24 1977-06-21 Yeda Research And Development Co., Ltd. Cephalosporin antibiotics
CA1070688A (en) * 1975-11-12 1980-01-29 Mitsuru Yoshioka Cephalosporin analogues
CA1085392A (en) * 1976-03-25 1980-09-09 Masayuki Narisada Arylmalonamido-1-oxadethiacephalosporins

Also Published As

Publication number Publication date
NZ188173A (en) 1981-05-15
GB1576796A (en) 1980-10-15
ZA784753B (en) 1979-08-29
MX5328E (es) 1983-06-22
AT361121B (de) 1981-02-25
AU517618B2 (en) 1981-08-13
ES472817A1 (es) 1979-02-16
ATA620378A (de) 1980-07-15
NL190554B (nl) 1993-11-16
NL190554C (nl) 1994-04-18
NL7808802A (nl) 1979-02-27
DK372878A (da) 1979-02-26
YU43999B (en) 1990-02-28
RO75070A (ro) 1980-10-30
DD137230A5 (de) 1979-08-22
IL55429A0 (en) 1978-10-31
FR2401165A1 (fr) 1979-03-23
PH17508A (en) 1984-09-07
DE2837264A1 (de) 1979-03-01
AU3923878A (en) 1980-02-28
PT68434A (en) 1978-09-01
IE47630B1 (en) 1984-05-16
FI65432B (fi) 1984-01-31
CS203927B2 (en) 1981-03-31
NO782866L (no) 1979-02-27
US4201782A (en) 1980-05-06
GR70260B (es) 1982-09-02
DE2837264C2 (es) 1991-06-13
PL209215A1 (pl) 1979-06-04
PL110656B1 (en) 1980-07-31
BG34338A3 (en) 1983-08-15
IT1118098B (it) 1986-02-24
FI65432C (fi) 1984-05-10
IT7868975A0 (it) 1978-08-24
FR2401165B1 (es) 1982-06-25
CH637396A5 (de) 1983-07-29
JPS609718B2 (ja) 1985-03-12
YU202878A (en) 1982-10-31
SU812182A3 (ru) 1981-03-07
BE869955A (fr) 1978-12-18
CA1101417A (en) 1981-05-19
IE781703L (en) 1979-02-25
JPS5436288A (en) 1979-03-16
SE7808950L (sv) 1979-02-26
HU177900B (en) 1982-01-28
SE452010B (sv) 1987-11-09
FI782586A (fi) 1979-02-26

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