AR112795A1 - Compuestos heterocíclicos fungicidas de tiazol - Google Patents
Compuestos heterocíclicos fungicidas de tiazolInfo
- Publication number
- AR112795A1 AR112795A1 ARP180102550A ARP180102550A AR112795A1 AR 112795 A1 AR112795 A1 AR 112795A1 AR P180102550 A ARP180102550 A AR P180102550A AR P180102550 A ARP180102550 A AR P180102550A AR 112795 A1 AR112795 A1 AR 112795A1
- Authority
- AR
- Argentina
- Prior art keywords
- ring
- 6alquilo
- alkyl
- membered
- isoxazolyl
- Prior art date
Links
- 239000000417 fungicide Substances 0.000 title abstract 2
- FZWLAAWBMGSTSO-UHFFFAOYSA-N Thiazole Chemical compound C1=CSC=N1 FZWLAAWBMGSTSO-UHFFFAOYSA-N 0.000 title 1
- 230000000855 fungicidal effect Effects 0.000 title 1
- 150000002391 heterocyclic compounds Chemical class 0.000 title 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 16
- 229910052799 carbon Inorganic materials 0.000 abstract 13
- 229910052717 sulfur Inorganic materials 0.000 abstract 13
- 125000004122 cyclic group Chemical group 0.000 abstract 12
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 10
- 229910052757 nitrogen Inorganic materials 0.000 abstract 10
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 9
- IKHGUXGNUITLKF-UHFFFAOYSA-N Acetaldehyde Chemical compound CC=O IKHGUXGNUITLKF-UHFFFAOYSA-N 0.000 abstract 9
- 229910052739 hydrogen Inorganic materials 0.000 abstract 9
- 239000001257 hydrogen Substances 0.000 abstract 9
- 229910020008 S(O) Inorganic materials 0.000 abstract 8
- 229910052736 halogen Inorganic materials 0.000 abstract 8
- 150000002367 halogens Chemical class 0.000 abstract 8
- 125000000446 sulfanediyl group Chemical group *S* 0.000 abstract 8
- -1 cyano, hydroxy Chemical group 0.000 abstract 7
- 125000000623 heterocyclic group Chemical group 0.000 abstract 7
- 150000002431 hydrogen Chemical class 0.000 abstract 7
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 6
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 6
- 125000003118 aryl group Chemical group 0.000 abstract 6
- 125000001072 heteroaryl group Chemical group 0.000 abstract 6
- 125000000262 haloalkenyl group Chemical group 0.000 abstract 5
- 125000001424 substituent group Chemical group 0.000 abstract 5
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000000232 haloalkynyl group Chemical group 0.000 abstract 4
- 125000005842 heteroatom Chemical group 0.000 abstract 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 4
- 229920006395 saturated elastomer Polymers 0.000 abstract 4
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 3
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 3
- 125000004916 (C1-C6) alkylcarbonyl group Chemical group 0.000 abstract 3
- 125000006570 (C5-C6) heteroaryl group Chemical group 0.000 abstract 3
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 3
- NBBJYMSMWIIQGU-UHFFFAOYSA-N Propionic aldehyde Chemical compound CCC=O NBBJYMSMWIIQGU-UHFFFAOYSA-N 0.000 abstract 3
- 150000001299 aldehydes Chemical class 0.000 abstract 3
- 125000004457 alkyl amino carbonyl group Chemical group 0.000 abstract 3
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000006583 (C1-C3) haloalkyl group Chemical group 0.000 abstract 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 abstract 2
- KHBQMWCZKVMBLN-UHFFFAOYSA-N Benzenesulfonamide Chemical compound NS(=O)(=O)C1=CC=CC=C1 KHBQMWCZKVMBLN-UHFFFAOYSA-N 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000004414 alkyl thio group Chemical group 0.000 abstract 2
- 125000004429 atom Chemical group 0.000 abstract 2
- 125000002837 carbocyclic group Chemical group 0.000 abstract 2
- 150000001721 carbon Chemical group 0.000 abstract 2
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 2
- 230000001351 cycling effect Effects 0.000 abstract 2
- 239000012634 fragment Substances 0.000 abstract 2
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000003261 o-tolyl group Chemical group [H]C1=C([H])C(*)=C(C([H])=C1[H])C([H])([H])[H] 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 abstract 1
- 125000004454 (C1-C6) alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004739 (C1-C6) alkylsulfonyl group Chemical group 0.000 abstract 1
- 125000004845 (C1-C6) alkylsulfonylamino group Chemical group 0.000 abstract 1
- 125000004737 (C1-C6) haloalkoxy group Chemical group 0.000 abstract 1
- 125000004741 (C1-C6) haloalkylsulfonyl group Chemical group 0.000 abstract 1
- 125000006636 (C3-C8) cycloalkylcarbonyl group Chemical group 0.000 abstract 1
- 125000001054 5 membered carbocyclic group Chemical group 0.000 abstract 1
- 125000004008 6 membered carbocyclic group Chemical group 0.000 abstract 1
- 125000001960 7 membered carbocyclic group Chemical group 0.000 abstract 1
- 101100495917 Arabidopsis thaliana ATRX gene Proteins 0.000 abstract 1
- 125000003320 C2-C6 alkenyloxy group Chemical group 0.000 abstract 1
- 150000001204 N-oxides Chemical class 0.000 abstract 1
- 125000005193 alkenylcarbonyloxy group Chemical group 0.000 abstract 1
- 125000004450 alkenylene group Chemical group 0.000 abstract 1
- 125000006193 alkinyl group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000003806 alkyl carbonyl amino group Chemical group 0.000 abstract 1
- 125000005130 alkyl carbonyl thio group Chemical group 0.000 abstract 1
- 125000005196 alkyl carbonyloxy group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000005133 alkynyloxy group Chemical group 0.000 abstract 1
- 125000006615 aromatic heterocyclic group Chemical group 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 125000002619 bicyclic group Chemical group 0.000 abstract 1
- 229910002091 carbon monoxide Inorganic materials 0.000 abstract 1
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 1
- 125000006310 cycloalkyl amino group Chemical group 0.000 abstract 1
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 abstract 1
- 125000005221 halo alkyl carbonyl amino group Chemical group 0.000 abstract 1
- 125000005291 haloalkenyloxy group Chemical group 0.000 abstract 1
- 125000004993 haloalkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004692 haloalkylcarbonyl group Chemical group 0.000 abstract 1
- 125000004664 haloalkylsulfonylamino group Chemical group 0.000 abstract 1
- 125000005292 haloalkynyloxy group Chemical group 0.000 abstract 1
- 125000006769 halocycloalkoxy group Chemical group 0.000 abstract 1
- 125000005347 halocycloalkyl group Chemical group 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000002088 tosyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1C([H])([H])[H])S(*)(=O)=O 0.000 abstract 1
- 125000004665 trialkylsilyl group Chemical group 0.000 abstract 1
Classifications
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
- A01N43/78—1,3-Thiazoles; Hydrogenated 1,3-thiazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
- A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La presente se refiere a un compuesto y a un proceso para prepararlo. Composiciones y usos como fungicidas. Reivindicación 1: Un compuesto seleccionado de la fórmula (1), donde, T se selecciona de un anillo de arilo de 5 ó 6 miembros o un anillo cíclico saturado o parcialmente saturado de 5 ó 6 miembros o un anillo heteroarilo de 5 ó 6 miembros o un anillo heterocíclico saturado o parcialmente saturado de 5 ó 6 miembros, en el que cada el miembro del anillo del anillo heteroarilo se selecciona de C, N, O y S, y en el que cada miembro del anillo, del anillo heterocíclico se selecciona de C, N, O, S(O)ₐ, C=O, C=S, S=NR⁶ y S(O)=NR⁶, y T está opcionalmente sustituido con uno o más R¹ᵃ en los miembros del anillo de carbono y uno o más R¹ᵇ en los miembros del anillo del heteroátomo; L¹ es O, S, NR²³, donde, R²³ se selecciona de hidrógeno, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, alcoxi C₁₋₆alquilo C₁₋₆, alquiltio C₁₋₆alquilo C₁₋₆, alquilsulfinilo C₁₋₆alquilo C₁₋₆, alquilsulfonilo C₁₋₆alquilo C₁₋₆, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆alquilo C₁₋₆, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆, alquilsulfonilo C₁₋₆ y haloalquilsulfonilo C₁₋₆; A es C(R¹⁵)₂ o C(R¹⁵)₂-C(R¹⁵)₂; donde, R¹⁵ se selecciona independientemente de hidrógeno, halógeno, ciano, hidroxi, aldehído, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, alcoxi C₁₋₆alquilo C₁₋₆, alquiltio C₁₋₆alquilo C₁₋₆, alquilsulfinilo C₁₋₆alquilo C₁₋₆, alquilsulfonilo C₁₋₆alquilo C₁₋₆, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆, alcoxicarbonil C₁₋₆alquilo C₁₋₆, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆, alcoxilo C₁₋₆, haloalcoxilo C₁₋₆, alquiltio C₁₋₆, haloalquiltio C₁₋₆, alquilsulfinilo C₁₋₆, haloalquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆ y haloalquilsulfonilo C₁₋₆; W es O ó S; Z es C o N; la presentación ⁻ ⁻ ⁻ ⁻ ⁻ en el anillo D es un enlace simple cuando Z es N y es un enlace simple o doble cuando Z es C; n es un número entero que varía de 0 a 9 con la condición de que cuando Z es N, n es un número entero que varía de 0 a 8; y cuando la presentación ⁻ ⁻ ⁻ ⁻ ⁻ en el anillo D es un enlace doble, entonces n es un número entero que va de 0 a 7; G es un anillo heteroarilo de 5 ó 6 miembros opcionalmente sustituido o un anillo heterocíclico saturado o parcialmente saturado de 5 ó 6 miembros, cada miembro del anillo del anillo heteroarilo se selecciona de C, N, O y S; y cada miembro del anillo del anillo heterocíclico se selecciona de C, N, O, S(O)ₐ, C(=O), C(=S), S(=NR⁶) y S(O)=NR⁶; donde los miembros del anillo de carbono están sustituidos con uno o más miembros del anillo de R³ᵃ y heteroátomo están sustituidos con uno o más R¹¹ᵃ; donde, R³ᵃ es hidrógeno o R³ᵇ; R³ᵇ es alquilo C₁₋₃, haloalquilo C₁₋₃, halógeno, un fenilo o anillo heteroaromático de 5 ó 6 miembros, en el que el fenilo o el anillo heteroaromático de 5 ó 6 miembros está opcionalmente sustituido con uno o más sustituyentes seleccionados independientemente de R⁴ᵃ en los miembros del anillo de carbono y R⁴ᵇ en los miembros del anillo de nitrógeno, R⁴ᵃ se selecciona independientemente de alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, cicloalquilo C₃₋₆, cicloalquil C₃₋₆alquilo C₁₋₆, alquilo C₁₋₆cicloalquilo C₃₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, halocicloalquilo C₃₋₆, halógeno, hidroxi, amino, ciano, nitro, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alquiltio C₁₋₆, alquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, haloalquiltio C₁₋₆, haloalquilsulfinilo C₁₋₆, haloalquilsulfonilo C₁₋₆, alquilamino C₁₋₆, dialquilamino C₁₋₆, cicloalquilamino C₃₋₆, alcoxi C₁₋₆alquilo C₁₋₆, hidroxialquilo C₁₋₆, alquilcarbonilo C₁₋₆, alcoxicarbonilo C₁₋₆, alquilcarboniloxi C₁₋₆, alquilcarboniltio C₁₋₆, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆ y trialquilsililo C₁₋₆; R⁴ᵇ se selecciona independientemente de alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, cicloalquilo C₃₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, halocicloalquilo C₃₋₆ y alcoxi C₁₋₆alquilo C₁₋₆; R¹¹ᵃ es hidrógeno o R¹¹ᵇ, en donde R¹¹ᵇ se selecciona independientemente entre alquilo C₁₋₃, cicloalquilo C₃₋₆, haloalquilo C₁₋₆, halocicloalquilo C₃₋₆; J es un anillo carbocíclico o heterocíclico de 5, 6 ó 7 miembros, un sistema de anillo bicíclico carbocíclico o heterocíclico de 8 a 11 miembros o un sistema de anillo espirocíclico carbocíclico o heterocíclico de 7 a 11 miembros, cada miembro del anillo del el anillo heterocíclico o sistema de anillo se selecciona de C, N, O, S(O)ₐ, C(=O), C(=S), y cada anillo o sistema de anillo está opcionalmente sustituido con uno o más sustituyentes seleccionados independientemente de R⁵, o J se selecciona del grupo de fórmulas (2) donde W¹ es C(R⁵)₂ o CO ó O ó S o SO o SO₂ o NR⁵; R⁵ se selecciona independientemente de hidrógeno, halógeno, ciano, hidroxi, nitro, aldehído, ácido carboxílico, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, cicloalquilo C₃₋₆, halocicloalquilo C₃₋₆, alquilo C₁₋₆cicloalquilo C₃₋₆, cicloalquilo C₃₋₆alquilo C₁₋₆, cicloalquilo C₃₋₆cicloalquilo C₃₋₆, halociclo C₃₋₆alquilo C₁₋₆, cicloalquenilo C₃₋₆, halocicloalquenilo C₃₋₆, alcoxi C₁₋₆alquilo C₁₋₆, cicloalcoxi C₃₋₆alquilo C₁₋₆, alquiltio C₁₋₆alquilo C₁₋₆, alquilsulfinilo C₁₋₆alquilo C₁₋₆, alquilsulfonilo C₁₋₆alquilo C₁₋₆, alquilamino C₁₋₆alquilo C₁₋₆, dialquilamino C₁₋₆alquilo C₁₋₆, haloalquilamino C₁₋₆alquilo C₁₋₆, cicloalquilamino C₁₋₆alquilo C₁₋₆, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, cicloalquilcarbonilo C₃₋₆, alcoxicarbonilo C₁₋₆, cicloalcoxicarbonilo C₃₋₆, cicloalquil C₃₋₆alcoxicarbonilo C₁₋₆, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆, cicloalquilaminocarbonilo C₃₋₆, haloalcoxi C₁₋₆alquilo C₁₋₆, hidroxialquilo C₁₋₆, alcoxi C₁₋₆, haloalcoxi C₁₋₆, cicloalcoxi C₃₋₆, halocicloalcoxi C₃₋₆, cicloalquil C₃₋₆alcoxi C₁₋₆, alqueniloxi C₂₋₆, haloalqueniloxi C₂₋₆, alquiniloxi C₂₋₆, haloalquiniloxi C₂₋₆, alcoxi C₁₋₆alcoxi C₁₋₆, alquilcarboniloxi C₁₋₆, haloalquilcarboniloxi C₁₋₆, cicloalquilcarboniloxi C₃₋₆, alquil C₁₋₆carboniloalcoxi C₁₋₆, alquiltio C₁₋₆, haloalquiltio C₁₋₆, cicloalquiltio C₃₋₆, alquilsulfinilo C₁₋₆, haloalquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, haloalquilsulfonilo C₁₋₆, cicloalquilsulfonilo C₃₋₆, trialquilsililo C₁₋₆, alquilsulfonilamino C₁₋₆, haloalquilsulfonilamino C₁₋₆ o -Z²Q, donde, Z¹ y Z² son independientemente un enlace directo, O, C=O, C=S, S(O)ₐ, CHR²⁰ o NR²¹; donde, R²⁰ se selecciona independientemente de hidrógeno, alquilo C₁₋₄ o haloalquilo C₁₋₄; y R²¹ se selecciona independientemente de hidrógeno, alquilo C₁₋₃, haloalquilo C₁₋₃, cicloalquilo C₃₋₈, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₈, alcoxicarbonilo C₁₋₈ o haloalcoxicarbonilo C₁₋₈; Q se selecciona independientemente de fenilo, bencilo, naftilo, un anillo de arilo de 5 ó 6 miembros, un sistema de anillo arílico multi-cíclico de 8 a 11 miembros, un sistema de anillo condensado con arilo de 8 a 11 miembros, un anillo heteroarilo de 5 ó 6 miembros, un sistema de anillo multi-cíclico heteroarílico de 8 a 11 miembros o un sistema de anillo condensado heteroarílico de 8 a 11 miembros, cada miembro de anillo del anillo o sistema de anillo se selecciona de C, N, O y S, y cada sistema de anillo o anillo está opcionalmente sustituido con uno o más sustituyentes seleccionados independientemente entre R⁷ en los miembros del anillo del átomo de carbono y R¹² en los miembros del anillo del heteroátomo, o Q se selecciona independientemente de un anillo carbocíclico no aromático de 3 a 7 miembros, un anillo heterocíclico no aromático de 5, 6 ó 7 miembros, un sistema de anillo multi-cíclico no aromático de 8 a 15 miembros o un sistema de anillo fusionado no aromático de 8 a 15 miembros, cada miembro del anillo del anillo o sistema de anillos se selecciona de C, N, O, S(O)ₐ, C(=O), C(=S), S(=NR⁶) y S(=O)=NR⁶ y SiR¹⁶R¹⁷, y cada sistema de anillo o anillo está opcionalmente sustituido con uno o más sustituyentes seleccionados independientemente entre R⁷ en los miembros del anillo del átomo de carbono y R¹² en los miembros del anillo del heteroátomo; o J y Q juntos forman un fragmento seleccionado de los compuestos de fórmula (3) y (4); donde, x en los fragmentos de fórmula (3) y (4) es un número entero que varía de 0 a 2 e Y se selecciona de N, O y S, donde, R¹ᵃ, R¹ᵇ, R⁷ y R¹² se seleccionan independientemente entre hidrógeno, halógeno, hidroxi, ciano, nitro, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, alcanoalquinilo C₂₋₆, cicloalquilo C₃₋₈, halocicloalquilo C₃₋₈, alquilo C₁₋₆cicloalquilo C₃₋₈, cicloalquilo C₃₋₈alquilo C₁₋₆, cicloalquilo C₃₋₈cicloalquilo C₃₋₈, haloalquiloalquilo C₃₋₈alquilo C₁₋₆, alcoxi C₁₋₆alquilo C₁₋₆, cicloalcoxi C₃₋₈alquilo C₁₋₆, alquiltio C₁₋₆alquilo C₁₋₆, alquilsulfinilo C₁₋₆alquilo C₁₋₆, alquilsulfonilo C₁₋₆alquilo C₁₋₆, alquilamino C₁₋₆, dialquilamino C₁₋₆, alquilamino C₁₋₆alquilo C₁₋₆, dialquilamino C₁₋₆alquilo C₁₋₆, haloalquilamino C₁₋₆alquilo C₁₋₆, cicloalquilamino C₃₋₈, cicloalquilamino C₃₋₈alquilo C₁₋₆, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, cicloalquilcarbonilo C₃₋₈, alcoxicarbonilo C₁₋₆, cicloalcoxicarbonilo C₃₋₈, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆, cicloalquilaminocarbonilo C₃₋₈, haloalcoxi C₁₋₆alquilo C₁₋₆, hidroxialquilo C₁₋₆, hidroxialquenilo C₁₋₆, hidroxialquinilo C₁₋₆, alcoxilo C₁₋₆, haloalcoxilo C₁₋₆, cicloalcoxilo C₁₋₆, halocicloalcoxilo C₃₋₈, cicloalquilo C₁₋₈alcoxilo C₁₋₆, alqueniloxilo C₂₋₆, haloalqueniloxilo C₂₋₆, alquiniloxilo C₂₋₆, haloalquiniloxi C₂₋₆, alcoxi C₁₋₆alcoxi C₁₋₆, alquilcarboniloxi C₁₋₆, haloalquilcarboniloxi C₁₋₆, cicloalquilcarboniloxi C₃₋₆, alquil C₁₋₆carboniloalcoxi C₁₋₆, alquiltio C₁₋₆, haloalquiltio C₁₋₆, cicloalquiltio C₃₋₈, alquilsulfinilo C₁₋₆, haloalquilsulfinilo C₁₋₆, alquilsulfonilo C₁₋₆, haloalquilsulfonilo C₁₋₆, cicloalquilsulfonilo C₃₋₈, cicloalquilsulfinilo C₃₋₈, trialquilsililo C₁₋₆, alquilsulfonilamino C₁₋₆, haloalquilsulfonilamino C₁₋₆, alquilcarboniltio C₁₋₆, alquilsulfoniloxi C₁₋₆, alquilsulfiniloxi C₁₋₆, arilsulfoniloxi, arilsulfiniloxi, arilsulfonilo, arilsulfinilo, cianoalquilo C₁₋₆, alquenilcarboniloxi C₂₋₆, alcoxi C₁₋₆alquiltio C₁₋₆, alquiltio C₁₋₆alcoxi C₁₋₆, haloalquenilcarboniloxi C₂₋₆, alcoxi C₁₋₆alquinilo C₂₋₆, alquiniltio C₂₋₆, haloalcoalquilcarboniloxi C₃₋₈, alquenilamino C₂₋₆, alquinilamino C₂₋₆, haloalquilamino C₁₋₆, cicloalquil C₃₋₈alquilamino C₁₋₆, alcoxiamino C₁₋₆, haloalcoxiamino C₁₋₆, alquilcarbonilamino C₁₋₆, haloalquilcarbonilamino C₁₋₆, alcoxicarbonilamino C₁₋₆, alqueniltio C₂₋₆, haloalcoxicarbonilo C₁₋₆, alcoxi C₁₋₆alquil C₁₋₆carbonilo, haloalcoxicarbonilamino C₁₋₆, alcoxi C₁₋₆alquilaminocarbonilo C₁₋₆, alquiltiocarbonilo C₁₋₆, cicloalqueniloxi C₃₋₈alquilo C₁₋₆, alcoxi C₁₋₆alcoxicarbonilo C₁₋₆, haloalcoxi C₁₋₆haloalcoxi C₁₋₆, alcoxi C₁₋₆haloalcoxi C₁₋₆, halocicloalcoxi C₃₋₈alquilo C₁₋₆, dialquilaminocarbonilamino C₁₋₆, alcoxi C₁₋₆alquenilo C₂₋₆, alquiltiocarboniloxi C₁₋₆, haloalcoxi C₁₋₆alcoxi C₁₋₆, haloalquilsulfoniloxi C₁₋₆, alcoxi C₁₋₆haloalquilo C₁₋₆, dihaloalquilamino C₁₋₆, dialcoxi C₁₋₆alquilo C₁₋₆, alquilaminocarbonilamino C₁₋₆, haloalcoxi C₁₋₆haloalquilo C₁₋₆, alquilaminocarbonilo C₁₋₆alquilamino C₁₋₆, trialquilsililo C₁₋₆alquiniloxi C₂₋₆, trialquilsililoxi C₁₋₆, trialquilsililo C₁₋₆alquinilo C₂₋₆, cianoalcoxi C₁₋₆alquilo C₁₋₆, dialquiltio C₁₋₆alquilo C₁₋₆, alcoxisulfonilo C₁₋₆, halocicloalcoxicarbonilo C₃₋₈, alquil C₁₋₆alquil C₃₋₈carbonilo, halociclo C₃₋₈alquilcarbonilo C₁₋₆, alqueniloxicarbonilo C₂₋₆, alquiniloxicarbonilo C₂₋₆, cianoalcoxicarbonilo C₁₋₆, alquiltio C₁₋₆alcoxicarbonilo C₁₋₆, alquinilcarboniloxi C₂₋₆, haloalquinilcarboniloxi C₂₋₆, cianocarboniloxi, cianoalquil C₁₋₆carboniloxi, cicloalquilsulfoniloxi C₃₋₈, cicloalquil C₃₋₈alquilsulfoniloxi C₁₋₆, halocicloalquilsulfoniloxi C₃₋₈, alquenilsulfoniloxi C₂₋₆, alquinilsulfoniloxi C₂₋₆, cianoalquilsulfoniloxi C₁₋₆, haloalquenilsulfoniloxi C₂₋₆, haloalquinilsulfoniloxi C₂₋₆, alquinilcicloalquiloxi C₂₋₆, cianoalqueniloxi C₂₋₆, cianoalquiniloxi C₂₋₆, alcoxicarboniloxi C₁₋₆, alqueniloxicarboniloxi C₂₋₆, alquiniloxicarboniloxi C₂₋₆, alcoxialquilcarboniloxi C₁₋₆, sulfiliminas, sulfoximinas, SF₅ o Z²Q, R¹⁶ y R¹⁷ se seleccionan independientemente entre alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, cicloalquilo C₃₋₆, halocicloalquilo C₃₋₆, cicloalquil C₁₋₆alquilo C₁₋₆, alquilo C₁₋₆cicloalquilo C₃₋₆, haloalquilo C₁₋₆, alcoxi C₁₋₆ y haloalcoxi C₁₋₆; R⁵ y R⁷ o R⁵ y R¹² tomados junto con los átomos que unen R⁵ y R⁷ o R¹² para formar un anillo saturado, insaturado o parcialmente insaturado de 4 a 7 miembros, cada miembro del anillo seleccionado de C, N, O, S(O)ₐ, C=O, C=S, S=NR⁶ y S(O)=NR⁶, y dicho anillo opcionalmente sustituido en miembros del anillo distintos de los átomos que unen R⁵ y R⁷ o R¹² con R⁸, en donde, R⁸ se selecciona de halógeno, alquilo C₁₋₆, haloalquilo C₁₋₆, cicloalquilo C₃₋₈ y cicloalquilo C₃₋₈; R² y R⁶ se seleccionan independientemente de hidrógeno, halógeno, ciano, hidroxi, aldehído, ácido carboxílico, alquilo C₁₋₆, alquenilo C₂₋₆, alquinilo C₂₋₆, haloalquilo C₁₋₆, haloalquenilo C₂₋₆, haloalquinilo C₂₋₆, cicloalquilo C₃₋₆, halocicloalquilo C₃₋₆, alquilo C₁₋₆cicloalquilo C₃₋₆, cicloalquilo C₃₋₆alquilo C₁₋₆, halocicloalquil C₃₋₆alquilo C₁₋₆, cicloalquenilo C₃₋₆, halocicloalquenilo C₃₋₆, alcoxi C₁₋₆alquilo C₁₋₆, alquiltio C₁₋₆alquilo C₁₋₆, alquilsulfinilo C₁₋₆alquilo C₁₋₆, alquilsulfonilo C₁₋₆alquilo C₁₋₆, alquilamino C₁₋₆alquilo C₁₋₆, dialquilamino C₁₋₆alquilo C₁₋₆, haloalquilamino C₁₋₆alquilo C₁₋₆, alquilcarbonilo C₁₋₆, haloalquilcarbonilo C₁₋₆, cicloalquilcarbonilo C₃₋₆, alcoxicarbonilo C₁₋₆, cicloalcoxicarbonilo C₃₋₆, cicloalquil C₃₋₆alcoxicarbonilo C₁₋₆, alquilaminocarbonilo C₁₋₆, dialquilaminocarbonilo C₁₋₆, alcoxi C₁₋₆, haloalcoxi C₁₋₆, cicloalcoxi C₃₋₆, halocicloalcoxi C₃₋₆, alqueniloxi C₂₋₆, haloalqueniloxi C₂₋₆, alquiniloxi C₂₋₆, haloalquiniloxi C₂₋₆, alcoxi C₁₋₆alcoxi C₁₋₆, alquilcarboniloxi C₁₋₆, haloalquil C₁₋₆carboniloxi, alquiltio C₁₋₆, haloalquiltio C₁₋₆, cicloalquiltio C₃₋₆, alquilamino C₁₋₆, dialquilamino C₁₋₆, haloalquilamino C₁₋₆, halodialquilamino C₁₋₆, cicloalquilamino C₃₋₆, alquilcarbonilamino C₁₋₆, haloalquilcarbonilamino C₁₋₆, alquilsulfonilamino C₁₋₆ y haloalquilsulfonilamino C₁₋₆, o dos R² se toman juntos como alquileno C₁₋₄ o alquenileno C₂₋₄ o CH=CH-CH=CH- para formar un sistema de anillo bicíclico o fusionado puenteado opcionalmente sustituido con un sustituyente seleccionado de alquilo C₁₋₆, haloalquilo C₁₋₆, alcoxi C₁₋₆, haloalcoxi C₁₋₆, halógeno, hidroxi, amino, ciano y nitro, con la condición de que los compuestos estén excluidos de la definición de la fórmula (1): etanona, 1-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil]-2-[[5-(trifluorometil)-2-piridinil]tio] - (CAS RN- 1023141-80-1); benzamida, 2-[[2-[4-[-4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]-2-oxoetil]tio]-4-etoxi - (CAS RN- 1177816-84-0); etanona, 2-[(2-cloro-4-fluorofenil)tio]-1-[4-[4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil] - (CAS RN- 1177683-42-9); etanona, 2-(ciclohexiloxi)-1-[4-[4-[5-(2,6-difluorofenil)-4,5-dihidro-3-isoxazolil]-2-tiazolil]-1-piperidinil] - (CAS RN- 1173972-38-7); 1-propanona, 2-(4-clorofenoxi)-2-metil-1-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil] - (CAS RN- 1136418-28-4); etanona, 2-[(2-cloro-4-fluorofenil)tio]-1-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil] - (CAS RN- 1023177-70-9); bencenosulfonamida, N-metil-2-[[2-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil]-2-oxoetil]tio] - (CAS RN- 1023156-55-9); bencenosulfonamida, 2-[[2-[4-[4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]-2-oxoetil]tio]-N-metilo - (CAS RN- 1022602-51-2); etanona, 1-[4-[4-(S-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil]-2-(2,3,4,5,6-pentafluorofenoxi) - (CAS RN- 1022567-65-2); etanona, 1-[4-[4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]-2-[(4-metilfenil)sulfonil] - (CAS RN- 1022566-90-0); etanona, 2-(2,4-diclorofenoxi)-1-[4-[4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]- (CAS RN- 1022328-76-2); etanona, 2-(2,4-diclorofenoxi)-1-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil]- (CAS RN- 1022068-84-3); etanona, 1-[4-[-4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]-2-(2,3,4,5,6-pentafluorofenoxi) - (CAS RN- 1022028-25-6); 1-propanona, 1-[4-[4-(5-metil-3-fenil-4-isoxazolil)-2-tiazolil]-1-piperidinil]-3-[(2-metilfenil)tio] - (CAS RN- 1022326-33-5); y 1-propanona, 1-[4-[4-[3-(3,4-diclorofenil)-5-isoxazolil]-2-tiazolil]-1-piperidinil]-3-[(2-metilfenil)tio] - (CAS RN- 1024410-18-1); las sales, isómeros, complejos metálicos, N-óxidos y polimorfos de los mismos.
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TW202236965A (zh) | 2020-12-15 | 2022-10-01 | 印度商皮埃企業有限公司 | 包含哌啶噻唑化合物之新穎農業化學組成物 |
AR125834A1 (es) | 2021-05-15 | 2023-08-16 | Pi Industries Ltd | Composición agroquímica que comprende compuestos de piperidin-tiazol |
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- 2018-08-29 CN CN201880071012.XA patent/CN111655687A/zh active Pending
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CO2020002396A2 (es) | 2020-07-31 |
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US20200281202A1 (en) | 2020-09-10 |
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