AR107672A1 - Proceso para la fabricación de derivados de 3-piperazin-1-il-propilamina - Google Patents

Proceso para la fabricación de derivados de 3-piperazin-1-il-propilamina

Info

Publication number
AR107672A1
AR107672A1 ARP170100419A ARP170100419A AR107672A1 AR 107672 A1 AR107672 A1 AR 107672A1 AR P170100419 A ARP170100419 A AR P170100419A AR P170100419 A ARP170100419 A AR P170100419A AR 107672 A1 AR107672 A1 AR 107672A1
Authority
AR
Argentina
Prior art keywords
piperazin
manufacture
derivatives
propilamine
raney
Prior art date
Application number
ARP170100419A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of AR107672A1 publication Critical patent/AR107672A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms

Abstract

La presente solicitud se refiere a un proceso para fabricar derivados de 3-piperazin-1-il-propilamina. Reivindicación 1: Un procedimiento para la fabricación de un compuesto de fórmula (1) que comprende la reacción de un compuesto de fórmula (2) en presencia de hidrógeno y un catalizador seleccionado de Raney-níquel y Raney-cobalto; en el que R¹ es alquilo.
ARP170100419A 2016-02-22 2017-02-20 Proceso para la fabricación de derivados de 3-piperazin-1-il-propilamina AR107672A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP16156707 2016-02-22

Publications (1)

Publication Number Publication Date
AR107672A1 true AR107672A1 (es) 2018-05-23

Family

ID=55409779

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170100419A AR107672A1 (es) 2016-02-22 2017-02-20 Proceso para la fabricación de derivados de 3-piperazin-1-il-propilamina

Country Status (12)

Country Link
US (1) US20190092739A1 (es)
EP (1) EP3419965A1 (es)
JP (1) JP2019507152A (es)
KR (1) KR20180116277A (es)
CN (1) CN108699009A (es)
AR (1) AR107672A1 (es)
AU (1) AU2017222159A1 (es)
BR (1) BR112018015092A2 (es)
CA (1) CA3012288A1 (es)
MX (1) MX2018009943A (es)
SG (1) SG11201807010PA (es)
WO (1) WO2017144404A1 (es)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1012751A (fr) * 1949-01-24 1952-07-17 Rhone Poulenc Sa Nouveau dérivé de la pipérazine et de la quinoléïne et son procédé de préparation
GB997036A (en) * 1962-02-23 1965-06-30 Wellcome Found 9-substituted acridines
US5856535A (en) * 1994-08-18 1999-01-05 Magainin Pharmaceuticals, Inc. Aminosterol ester compounds
AU2001263021A1 (en) * 2000-05-10 2001-11-20 Bristol-Myers Squibb Company Alkylamine derivatives of dihydropyridine npy antagonists
GB0416728D0 (en) * 2004-07-27 2004-09-01 7Tm Pharma As Medicinal use of receptor ligands
WO2007146981A2 (en) * 2006-06-15 2007-12-21 Boehringer Ingelheim International Gmbh 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase c-alpha
EP2178864B1 (en) * 2007-08-02 2014-07-23 Cipla Limited Process for the preparation of alfuzosin hydrochloride

Also Published As

Publication number Publication date
MX2018009943A (es) 2018-11-09
CA3012288A1 (en) 2017-08-31
AU2017222159A1 (en) 2018-08-02
SG11201807010PA (en) 2018-09-27
WO2017144404A1 (en) 2017-08-31
EP3419965A1 (en) 2019-01-02
CN108699009A (zh) 2018-10-23
JP2019507152A (ja) 2019-03-14
KR20180116277A (ko) 2018-10-24
US20190092739A1 (en) 2019-03-28
BR112018015092A2 (pt) 2018-12-18

Similar Documents

Publication Publication Date Title
AR098343A1 (es) Proceso para la síntesis de un inhibidor de indolamina 2,3-dioxigenasa
BR112014030365A2 (pt) síntese de composto antiviral
PE20180327A1 (es) Proceso para preparar 4-amino-piridazinas
BR112016028773A2 (pt) processos para preparação de compostos antivirais
ECSP15043280A (es) Nuevos compuestos y composiciones para la inhibición de fasn
UY32096A (es) Derivados de 2-carboxamida - cicloamino - urea especìficos, sus sales farmacèuticamente aceptables, composiciones contenièndolos, pro-farmacos de los mismos, procesos para su produciòn y aplicaciones
AR094948A1 (es) Preparación de haloalcoxiarilhidracinas y los intermediarios a partir de los mismos
CO6410257A2 (es) Herbicidas novedosos
CR20150663A (es) Derivados de diazacarbazol como ligandos de tau para pet
BR112015027432A2 (pt) 3-(4-isobutil-2-metilfenil)propanal como ingrediente de perfume
CO6420341A2 (es) Herbicidas novedosos
AR088983A1 (es) Procedimiento para la preparacion de 5-fluoro-1h-pirazolopiridinas sustituidas
PE20151589A1 (es) Proceso de fabricacion de vortioxetina
BR112016018851A8 (pt) processo para fornecer um composto de fórmula (iv)
BR112018073488A2 (pt) intermediários para a síntese de derivados de ácido biliar, em particular de ácido obeticólico
CL2019000016A1 (es) Procesos novedosos para preparar estimuladores de guanilato ciclasa soluble.
CY1121116T1 (el) Νεα μεθοδος για την συνθεση αγομελατινης
CL2019000017A1 (es) Procesos novedosos para la preparación de estimuladores de guanilato ciclasa soluble.
AR107419A1 (es) Proceso para la preparación de ácidos 4-alcoxi-3-acetoxipicolínicos
AR088358A1 (es) Proceso de obtencion de acidos isoxazolil-metoxi-nicotinicos
BR112015024859A2 (pt) processo e intermediários para a preparação de pregabalina
AR098879A1 (es) Síntesis de ent-progesterona y sus productos intermedios
BR112016011048A8 (pt) processo para preparar um composto, processos para fabricar compostos, compostos e composições farmacêuticas
CR20150387A (es) Proceso para producir compuesto de piridazinona y producción de sus intermediarios
CL2023001049A1 (es) Procedimiento para la fabricación de compuestos orgánicos

Legal Events

Date Code Title Description
FB Suspension of granting procedure