AR090789A1 - Intermediarios y procesos para la preparacion de compuestos - Google Patents
Intermediarios y procesos para la preparacion de compuestosInfo
- Publication number
- AR090789A1 AR090789A1 ARP130101330A AR090789A1 AR 090789 A1 AR090789 A1 AR 090789A1 AR P130101330 A ARP130101330 A AR P130101330A AR 090789 A1 AR090789 A1 AR 090789A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- intermediaries
- compounds
- processes
- pyrrolo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Reivindicación 1: 5-bromo-4-cloro-3-nitro-1H-pirrolo[2,3-b]piridina de la fórmula (1) y sus estereoisómeros, tautómeros y sales farmacéuticamente aceptables. Reivindicación 2: Un proceso para la preparación de 5-bromo-4-cloro-3-nitro-1H-pirrolo[2,3-b]piridina de la fórmula (1) que comprende la etapa de sometimiento de la 4-cloro-3-nitro-1H-pirrolo[2,3-b]piridina de la fórmula (2) a una bromación, a fin de obtener 5-bromo-4-cloro-3-nitro-1H-pirrolo[2,3-b]piridina de la fórmula (1).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261637170P | 2012-04-23 | 2012-04-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR090789A1 true AR090789A1 (es) | 2014-12-10 |
Family
ID=48289659
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP130101330 AR090789A1 (es) | 2012-04-23 | 2013-04-22 | Intermediarios y procesos para la preparacion de compuestos |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US9221813B2 (es) |
| EP (1) | EP2855473B1 (es) |
| JP (2) | JP6370772B2 (es) |
| KR (1) | KR102096679B1 (es) |
| CN (1) | CN104395311B (es) |
| AR (1) | AR090789A1 (es) |
| AU (1) | AU2013252514B2 (es) |
| BR (1) | BR112014026367A2 (es) |
| CA (1) | CA2871436C (es) |
| IL (1) | IL235234B (es) |
| MX (1) | MX349255B (es) |
| MY (1) | MY168958A (es) |
| NZ (1) | NZ702135A (es) |
| RU (1) | RU2635359C2 (es) |
| SG (1) | SG11201406818VA (es) |
| WO (1) | WO2013163109A1 (es) |
| ZA (1) | ZA201408568B (es) |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5543523A (en) | 1994-11-15 | 1996-08-06 | Regents Of The University Of Minnesota | Method and intermediates for the synthesis of korupensamines |
| GB0400781D0 (en) * | 2004-01-14 | 2004-02-18 | Novartis Ag | Organic compounds |
| US7618964B2 (en) * | 2004-12-23 | 2009-11-17 | Hoffmann-La Roche Inc. | Benzamide derivatives, their manufacture and use as pharmaceutical agents |
| PL1893612T3 (pl) * | 2005-06-22 | 2012-01-31 | Plexxikon Inc | Pochodne pirolo-[2,3-b]pirydyny jako inhibitory kinazy białkowej |
| CN101223168A (zh) * | 2005-07-14 | 2008-07-16 | 安斯泰来制药株式会社 | Janus激酶3的杂环类抑制剂 |
| WO2007072017A2 (en) | 2005-12-22 | 2007-06-28 | The Institute Of Cancer Research | Enzyme inhibitors |
| WO2008144253A1 (en) * | 2007-05-14 | 2008-11-27 | Irm Llc | Protein kinase inhibitors and methods for using thereof |
| CA2711614A1 (en) | 2008-01-08 | 2009-07-16 | Array Biopharma Inc. | Pyrrolopyridines as kinase inhibitors |
| WO2009089359A1 (en) | 2008-01-09 | 2009-07-16 | Array Biopharma Inc. | Pyrazolopyridines as kinase inhibitors |
| GEP20125574B (en) * | 2008-01-11 | 2012-07-10 | Glenmark Pharmaceuticals Sa | Fused pyrimidine derivatives as trpv3 modulators |
| CL2009001152A1 (es) | 2008-05-13 | 2009-10-16 | Array Biopharma Inc | Compuestos derivados de n-(4-(cicloalquilo nitrogenado-1-il)-1h-pirrolo[2,3-b]piridin-3-il)amida, inhibidores de cinasa; proceso de preparacion; composicion farmaceutica; y su uso para el tratamiento de una enfermedad proliferativa. |
| BRPI0909957A2 (pt) * | 2008-06-11 | 2016-04-19 | Genentech Inc | "composto, composição farmacêutica, método de inibir o crescimento anormal de células ou de tratar um distúrbio hiperproliferativo em um mamífero, método de tratamento do câncer em um mamífero" |
| GB201201566D0 (en) * | 2012-01-30 | 2012-03-14 | Vernalis R&D Ltd | New chemical compounds |
-
2013
- 2013-04-22 MX MX2014012837A patent/MX349255B/es active IP Right Grant
- 2013-04-22 BR BR112014026367A patent/BR112014026367A2/pt not_active Application Discontinuation
- 2013-04-22 RU RU2014147003A patent/RU2635359C2/ru active
- 2013-04-22 SG SG11201406818VA patent/SG11201406818VA/en unknown
- 2013-04-22 MY MYPI2014002992A patent/MY168958A/en unknown
- 2013-04-22 CA CA2871436A patent/CA2871436C/en active Active
- 2013-04-22 CN CN201380033200.0A patent/CN104395311B/zh active Active
- 2013-04-22 WO PCT/US2013/037646 patent/WO2013163109A1/en active Application Filing
- 2013-04-22 KR KR1020147032707A patent/KR102096679B1/ko active IP Right Grant
- 2013-04-22 NZ NZ702135A patent/NZ702135A/en unknown
- 2013-04-22 AU AU2013252514A patent/AU2013252514B2/en active Active
- 2013-04-22 EP EP13720677.7A patent/EP2855473B1/en active Active
- 2013-04-22 JP JP2015507250A patent/JP6370772B2/ja active Active
- 2013-04-22 AR ARP130101330 patent/AR090789A1/es active IP Right Grant
- 2013-04-22 US US14/396,346 patent/US9221813B2/en active Active
-
2014
- 2014-10-21 IL IL235234A patent/IL235234B/en active IP Right Grant
- 2014-11-21 ZA ZA2014/08568A patent/ZA201408568B/en unknown
-
2017
- 2017-10-25 JP JP2017205900A patent/JP2018058841A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| CN104395311A (zh) | 2015-03-04 |
| US9221813B2 (en) | 2015-12-29 |
| KR102096679B1 (ko) | 2020-04-02 |
| MX349255B (es) | 2017-07-19 |
| RU2635359C2 (ru) | 2017-11-13 |
| JP6370772B2 (ja) | 2018-08-08 |
| EP2855473B1 (en) | 2018-10-03 |
| SG11201406818VA (en) | 2014-11-27 |
| CA2871436C (en) | 2020-07-28 |
| MY168958A (en) | 2019-01-28 |
| RU2014147003A (ru) | 2016-06-10 |
| AU2013252514A1 (en) | 2014-12-11 |
| MX2014012837A (es) | 2015-10-22 |
| AU2013252514B2 (en) | 2017-07-20 |
| BR112014026367A2 (pt) | 2017-06-27 |
| ZA201408568B (en) | 2017-05-31 |
| KR20150005995A (ko) | 2015-01-15 |
| NZ702135A (en) | 2016-09-30 |
| CA2871436A1 (en) | 2013-10-31 |
| US20150105557A1 (en) | 2015-04-16 |
| IL235234B (en) | 2018-01-31 |
| JP2018058841A (ja) | 2018-04-12 |
| EP2855473A1 (en) | 2015-04-08 |
| CN104395311B (zh) | 2017-04-19 |
| WO2013163109A1 (en) | 2013-10-31 |
| JP2015514784A (ja) | 2015-05-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration |