AR089889A1 - Compuestos fungicidas de pirimidina - Google Patents

Compuestos fungicidas de pirimidina

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Publication number
AR089889A1
AR089889A1 ARP130100334A ARP130100334A AR089889A1 AR 089889 A1 AR089889 A1 AR 089889A1 AR P130100334 A ARP130100334 A AR P130100334A AR P130100334 A ARP130100334 A AR P130100334A AR 089889 A1 AR089889 A1 AR 089889A1
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Argentina
Prior art keywords
alkyl
alkoxy
haloalkoxy
haloalkyl
hydrogen
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ARP130100334A
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English (en)
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Basf Se
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/044—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C07D491/048—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being five-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
    • C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Abstract

Su uso y los métodos para combatir los hongos fitopatogénicos. Además, las semillas tratadas al menos con un compuesto de este tipo. Más aún, procedimientos para preparar los compuestos de fórmula (1). Reivindicación 1: Compuestos de fórmula (1) en donde: Rᵃ² es hidrógeno, halógeno, CN, NO₂, OH, SH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alquiltio C₁₋₄, haloalquiltio C₁₋₄, alquilsulfinilo C₁₋₄, haloalquilsulfinilo C₁₋₄, alquilsulfonilo C₁₋₄, haloalquilsulfonilo C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, alcoxi C₁₋₄-alcoxi C₁₋₄, alquenilo C₂₋₄-, alquinilo C₂₋₄, haloalquenilo C₂₋₄-, haloalquinilo C₂₋₄-, cicloalquilo C₃₋₈, cicloalquiloxi C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₄, NRARB, C(=O)R, C(=NOR)R o -C(=NH)-O-R; RA, RB independientemente uno de otro son hidrógeno, alquilo C₁₋₄, alquenilo C₂₋₄, alquinilo C₂₋₄, fenilo, bencilo, cicloalquilo C₃₋₈, cicloalquenilo C₃₋₈ o -C(=O)-R; R es hidrógeno, OH, NH₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquilamino C₁₋₄- o di(alquil C₁₋₄-)amino; R es hidrógeno, alquilo C₁₋₄-, haloalquilo C₁₋₄, alquenilo C₂₋₄-, alquinilo C₂₋₄- o alcoxi C₁₋₄-alquilo C₁₋₄; R es hidrógeno o alquilo C₁₋₄; Rᵃ⁵, Rᵃ⁶ junto con dos átomos de carbono del miembro del anillo al cual están unidos, forman un carbociclo o heterociclo fusionado de 5 miembros saturado, parcialmente insaturado o aromático, en donde los átomos del miembro del anillo del heterociclo fusionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N y O y en donde el carbociclo o heterociclo fusionado es no sustituido o transporta 1, 2, 3 ó 4 radicales idénticos o diferentes seleccionados del grupo que consiste de halógeno, CN, alquilo C₁₋₄-, alcoxi C₁₋₄-, haloalquilo C₁₋₄ y haloalcoxi C₁₋₄; R es hidrógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo, C₂₋₄, haloalquinilo C₂₋₄, CN, CH₂CN, NRARB o CH₂-O-C(=O)R; en donde RA, RB independientemente uno de otro son hidrógeno, alquilo C₁₋₄, alquenilo C₂₋₄, alquinilo C₂₋₄, fenilo, bencilo, cicloalquilo C₃₋₈, cicloalquenilo C₃₋₈ o -(C=O)-R; R es hidrógeno, NH₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alquenilo C₂₋₄-, alquinilo C₂₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquilamino C₁₋₄- o di(alquil C₁₋₄-)amino; R¹, R² independientemente uno de otro son hidrógeno, halógeno, CN, OH, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄--alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, cicloalquilo C₃₋₈-, cicloalquil C₃₋₈-alquilo C₁₋₄, cicloalquiloxi C₃₋₈, NRARB, C(=O)R, C(=NOR)R, -C(=NH)-O-R o bencilo en donde el resto fenilo de bencilo está no sustituido o transporte 1, 2, 3, 4, ó 5 sustituyentes seleccionados del grupo que consiste de CN, halógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, (alcoxi C₁₋₄)carbonilo y di(alquilo C₁₋₄)aminocarbonilo; o dos radicales R¹ y R² que están unidos al mismo átomo de carbono forman junto con dicho átomo de carbono un carbociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7 miembros o un heterociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7 miembros, en donde los átomos del miembro del anillo del heterociclo antes mencionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el ciclo antes mencionado está no sustituido o transporta 1, 2, 3 ó 4 sustituyentes seleccionados de halógeno, CN, OH, SH, alquilo C₁₋₄-, alcoxi C₁₋₄ o alquiltio C₁₋₄; y uno o dos grupos CH₂ de los ciclos antes mencionados pueden ser reemplazados por uno o dos grupos C(=O) o C(=S) respectivamente; X es un grupo divalente seleccionado de -CR³R⁴-, -C(=O)-, -C(=S)-, -C(=NRD)-, y -C(=NORD)-,en donde RD es hidrógeno o alquilo C₁₋₄-; R³ y R⁴ independientemente uno de otro son hidrógeno, hidrógeno, CN, hidroxialquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, alcoxi C₁₋₄-alquilo C₁₋₄, haloalcoxi C₁₋₄-alquilo C₁₋₄, alquenilo C₂₋₄, haloalquenilo C₂₋₄, alquinilo C₂₋₄, haloalquinilo C₂₋₄, cicloalquilo C₃₋₈-, cicloalcoxi C₃₋₈, cicloalquil C₃₋₈-alquilo C₁₋₄, NRARB, C(=O)R, C(=NOR)R, -C(=NH)-O-R o bencilo, en donde el resto fenilo de bencilo está no sustituido o transporta 1, 2, 3, 4, ó 5 sustituyentes seleccionados del grupo que consiste en CN, halógeno, alquilo C₁₋₄, haloalquilo C₁₋₄, alcoxi C₁₋₄, haloalcoxi C₁₋₄, (alcoxi C₁₋₄-)carbonilo y di(alquil C₁₋₄)aminocarbonilo, o dos radicales R³ y R⁴ que están unidos al mismo átomos de carbono forman juntos con dicho átomo de carbono un carbociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros o un heterociclo saturado o parcialmente insaturado de 3, 4, 5, 6 ó 7-miembros, en donde los átomos del miembro del anillo del heterociclo antes mencionado incluyen además de los átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N, O y S, y en donde el ciclo antes mencionado está no sustituido o transporta 1, 2, 3 ó 4 sustituyentes seleccionados de halógeno, CN, OH, SH, alquilo C₁₋₄-, alcoxi C₁₋₄ o alquiltio C₁₋₄; y uno o dos grupos CH₂ de los ciclos antes mencionados pueden ser reemplazados por uno o dos grupos C(=O) o C(=S) respectivamente; n indica el número de sustituyentes Rᵇ en el anillo fenilo y n es 0, 1, 2, 3 ó 4; Rᵇ es halógeno, CN, NO₂, alquilo C₁₋₄-, haloalquilo C₁₋₄-, alcoxi C₁₋₄-, haloalcoxi C₁₋₄-, alquenilo C₂₋₄-, haloalquenilo C₂₋₄-, alquinilo C₂₋₄-, haloalquinilo C₂₋₄-, NRARB, C(=NOR)R o -C(=NH)-O-R, siendo posible para n = 2, 3, ó 4 que Rᵇ sean idénticos o diferentes; Het es un heteroarilo de 5 ó 6 miembros, en donde los átomos del miembro del anillo del heteroarilo incluyen además de átomos de carbono 1, 2, 3, ó 4 heteroátomos seleccionados del grupo de N, O y S y en donde el heteroarilo está no sustituido o transporta 1, 2, 3 ó 4 grupos Rᶜ idénticos o diferentes: Rᶜ es halógeno, CN, NO₂, NH₂, alquilo C₁₋₆-, haloalquilo C₁₋₆-, alcoxi C₁₋₆-, haloalcoxi C₁₋₆-, alquilamino C₁₋₆-, di(alquil C₁₋₆-)amino, alquiltio C₁₋₆-, haloalquiltio C₁₋₆-, alquilsulfinilo C₁₋₆-, haloalquilsulfinilo C₁₋₆-, alquilsulfonilo C₁₋₆-, haloalquilsulfonilo C₁₋₆-, alcoxi C₁₋₆-alquilo-C₁₋₄-, haloalcoxi C₁₋₆-alquilo-C₁₋₄-, alquenilo C₂₋₆-, alquinilo C₂₋₆-, C(=O)R, C(=NOR)R, cicloalquilo C₃₋₈-, cicloalquil C₃₋₈-alquilo C₁₋₄, fenilo, fenoxi, fenoxi-alquilo C₁₋₄ o un heteroarilo de 5 ó 6 miembros, en donde los átomos del miembro del anillo del heteroarilo incluyen además de átomos de carbono 1, 2, 3 ó 4 heteroátomos seleccionados del grupo de N,
ARP130100334A 2012-02-03 2013-02-01 Compuestos fungicidas de pirimidina AR089889A1 (es)

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EP12153767 2012-02-03
EP12154887 2012-02-10
EP12174746 2012-07-03

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US (1) US9072301B2 (es)
EP (1) EP2809659A1 (es)
JP (1) JP2015508752A (es)
CN (1) CN104220428A (es)
AR (1) AR089889A1 (es)
AU (1) AU2013214353A1 (es)
BR (1) BR112014018812A8 (es)
CA (1) CA2862346A1 (es)
CL (1) CL2014002014A1 (es)
EA (1) EA201400858A1 (es)
IL (1) IL233800A0 (es)
IN (1) IN2014DN07224A (es)
WO (1) WO2013113715A1 (es)

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JP2015511940A (ja) 2012-02-03 2015-04-23 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 殺菌性ピリミジン化合物
US9462809B2 (en) 2012-03-13 2016-10-11 Basf Se Fungicidal pyrimidine compounds
WO2014063642A1 (zh) * 2012-10-25 2014-05-01 中国中化股份有限公司 取代嘧啶类化合物及其用途
JP2016179944A (ja) * 2013-08-09 2016-10-13 石原産業株式会社 ジフルオロメチレン化合物
CN105722833A (zh) * 2013-09-16 2016-06-29 巴斯夫欧洲公司 杀真菌的嘧啶化合物
EP3080092B1 (en) 2013-12-12 2019-02-06 Basf Se Substituted [1,2,4]triazole and imidazole compounds
WO2015144480A1 (en) 2014-03-26 2015-10-01 Basf Se Substituted [1,2,4]triazole and imidazole compounds as fungicides
JP2017522266A (ja) 2014-05-13 2017-08-10 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 殺菌剤としての置換［１，２，４］トリアゾール及びイミダゾール化合物
AR100743A1 (es) 2014-06-06 2016-10-26 Basf Se Compuestos de [1,2,4]triazol sustituido
CN110964037B (zh) * 2018-09-29 2023-03-28 沈阳中化农药化工研发有限公司 含嘧啶并环类化合物及其制备方法和用途
CN111394258B (zh) * 2020-04-02 2022-03-18 浙江工业大学 匍枝根霉fl-3及其在提取茯苓多糖中的应用

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