AR063647A1 - Proceso para la sulfinilacion de un derivado de pirazol - Google Patents
Proceso para la sulfinilacion de un derivado de pirazolInfo
- Publication number
- AR063647A1 AR063647A1 ARP070105013A ARP070105013A AR063647A1 AR 063647 A1 AR063647 A1 AR 063647A1 AR P070105013 A ARP070105013 A AR P070105013A AR P070105013 A ARP070105013 A AR P070105013A AR 063647 A1 AR063647 A1 AR 063647A1
- Authority
- AR
- Argentina
- Prior art keywords
- sulfinylation
- cf3s
- hydroxy group
- amine
- acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/44—Oxygen and nitrogen or sulfur and nitrogen atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Agronomy & Crop Science (AREA)
- Wood Science & Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Epidemiology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Un proceso para la sulfinilación de un derivado de pirazol, caracterizado porque 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil]-1H-pirazol-3-carbonitrilo de fórmula (2) reacciona con un agente S de sulfinilación en presencia de al menos un complejo de ácido de amina en donde la(s) amina(s) se selecciona(n) de aminas secundarias cíclicas y el/los ácido(s) se selecciona(n) de derivados de ácido sulfónico, y con la adición de un agente de halogenación, en donde S es [CF3S(O)]2O; o CF3S(O)X, en donde X significa fluoro, cloro, bromo, iodo, un grupo hidroxi, o una sal de metal alcalino o alcalino térreo del grupo hidroxi, o sus mezclas, y compuestos intermediarios.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US86517806P | 2006-11-10 | 2006-11-10 | |
US91363807P | 2007-04-24 | 2007-04-24 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR063647A1 true AR063647A1 (es) | 2009-02-04 |
Family
ID=39167218
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP070105013A AR063647A1 (es) | 2006-11-10 | 2007-11-09 | Proceso para la sulfinilacion de un derivado de pirazol |
Country Status (16)
Country | Link |
---|---|
US (1) | US8629287B2 (es) |
EP (1) | EP2081909B8 (es) |
JP (1) | JP5450078B2 (es) |
KR (1) | KR20090083454A (es) |
CN (1) | CN102746234A (es) |
AR (1) | AR063647A1 (es) |
AU (1) | AU2007316720B2 (es) |
BR (1) | BRPI0718773A2 (es) |
CA (1) | CA2667562A1 (es) |
EA (1) | EA018047B1 (es) |
ES (1) | ES2398595T3 (es) |
IL (1) | IL198260A0 (es) |
MX (1) | MX2009004401A (es) |
NZ (1) | NZ576593A (es) |
WO (1) | WO2008055879A1 (es) |
ZA (1) | ZA200903969B (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1968578A4 (en) | 2005-12-14 | 2011-02-23 | Makhteshim Chem Works Ltd | POLYMORPHIC AND AMORPHOUS FORMS OF 5-AMINO-L- [2,6-DICHLORO-4- (TRIFLUOROMETHYL) PHENYL] -4- [(TRIFLUOROMETHYL) SULFINYL] -IH-PYRAZOLE-3-CARBONITRIL |
CA2667559A1 (en) | 2006-11-10 | 2008-05-15 | Basf Se | Process for the sulfinylation of a pyrazole derivative |
MX2011003455A (es) | 2008-10-02 | 2011-05-23 | Merial Ltd | Metodo para producir y purificar acido trifluorometanosulfinico. |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2716453B1 (fr) * | 1994-02-22 | 1996-03-29 | Rhone Poulenc Agrochimie | Procédé de sulfinylation de composés hétérocycliques. |
DE3568455D1 (en) * | 1984-05-23 | 1989-04-06 | Rhone Poulenc Chimie | Detergent compositions containing copolymers based on polyoxyethylene and polyoxyalkylene used as antisoil redeposition agents, and process for their preparation |
GB8713768D0 (en) * | 1987-06-12 | 1987-07-15 | May & Baker Ltd | Compositions of matter |
ES2167769T3 (es) * | 1996-08-01 | 2002-05-16 | Rhodia Chimie Sa | Procedimiento para la insercion de un grupo difluorometilo substituido. |
JPH11246555A (ja) * | 1997-10-31 | 1999-09-14 | Sumitomo Chem Co Ltd | フッ素置換ベンゾヘテロ環化合物 |
EP1042281B1 (en) | 1997-12-22 | 2003-03-19 | Minnesota Mining And Manufacturing Company | Process for preparation of fluorinated sulfinates |
DE19853560A1 (de) | 1998-11-20 | 2000-05-25 | Bayer Ag | Verfahren zur Herstellung von 5-Amino-3-(thio)carbamoylpyrazolen |
BR9917518B1 (pt) | 1999-10-22 | 2009-08-11 | processos para a preparação de pesticidas 1-arilpirazóis e seus intermediários. | |
JP2001220386A (ja) * | 1999-11-30 | 2001-08-14 | Takeda Chem Ind Ltd | オキサジアゾリン誘導体の製造方法 |
JP2002020364A (ja) * | 2000-07-06 | 2002-01-23 | Konica Corp | スルフィン酸ナトリウム、スルフィン酸カリウムの製造方法およびそれらを用いた写真用カプラーの製造方法 |
EP1331222A1 (en) * | 2002-01-28 | 2003-07-30 | Virbac S.A. | Environment friendly reagents and process for halogenoalkylsulfinylation of organic compounds |
CN1176078C (zh) * | 2002-03-27 | 2004-11-17 | 江苏省农药研究所 | 带三氟甲基亚磺酰基的吡唑类化合物的亚磺酰化方法 |
CA2667559A1 (en) | 2006-11-10 | 2008-05-15 | Basf Se | Process for the sulfinylation of a pyrazole derivative |
JP5450079B2 (ja) | 2006-11-10 | 2014-03-26 | ビーエーエスエフ ソシエタス・ヨーロピア | ピラゾール誘導体のスルフィニル化の方法 |
FR2924115B1 (fr) | 2007-11-27 | 2010-02-26 | Rhodia Operations | Procede de preparation d'un acide trifluoromethanesulfinique |
MX2011003455A (es) | 2008-10-02 | 2011-05-23 | Merial Ltd | Metodo para producir y purificar acido trifluorometanosulfinico. |
-
2007
- 2007-11-05 EA EA200900627A patent/EA018047B1/ru not_active IP Right Cessation
- 2007-11-05 US US12/514,103 patent/US8629287B2/en not_active Expired - Fee Related
- 2007-11-05 AU AU2007316720A patent/AU2007316720B2/en not_active Ceased
- 2007-11-05 NZ NZ576593A patent/NZ576593A/en not_active IP Right Cessation
- 2007-11-05 CA CA002667562A patent/CA2667562A1/en not_active Abandoned
- 2007-11-05 CN CN2012102457031A patent/CN102746234A/zh active Pending
- 2007-11-05 WO PCT/EP2007/061893 patent/WO2008055879A1/en active Application Filing
- 2007-11-05 MX MX2009004401A patent/MX2009004401A/es active IP Right Grant
- 2007-11-05 JP JP2009535703A patent/JP5450078B2/ja not_active Expired - Fee Related
- 2007-11-05 ES ES07822222T patent/ES2398595T3/es active Active
- 2007-11-05 BR BRPI0718773-4A patent/BRPI0718773A2/pt not_active Application Discontinuation
- 2007-11-05 KR KR1020097011872A patent/KR20090083454A/ko not_active Application Discontinuation
- 2007-11-05 EP EP07822222A patent/EP2081909B8/en active Active
- 2007-11-09 AR ARP070105013A patent/AR063647A1/es not_active Application Discontinuation
-
2009
- 2009-04-21 IL IL198260A patent/IL198260A0/en unknown
- 2009-06-08 ZA ZA2009/03969A patent/ZA200903969B/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2010509272A (ja) | 2010-03-25 |
EP2081909B1 (en) | 2013-01-09 |
IL198260A0 (en) | 2009-12-24 |
EP2081909B8 (en) | 2013-02-20 |
JP5450078B2 (ja) | 2014-03-26 |
AU2007316720A1 (en) | 2008-05-15 |
WO2008055879A1 (en) | 2008-05-15 |
EP2081909A1 (en) | 2009-07-29 |
CN102746234A (zh) | 2012-10-24 |
EA018047B1 (ru) | 2013-05-30 |
AU2007316720B2 (en) | 2013-05-09 |
CA2667562A1 (en) | 2008-05-15 |
NZ576593A (en) | 2011-12-22 |
BRPI0718773A2 (pt) | 2013-12-03 |
US8629287B2 (en) | 2014-01-14 |
MX2009004401A (es) | 2009-05-08 |
KR20090083454A (ko) | 2009-08-03 |
EA200900627A1 (ru) | 2009-10-30 |
US20100093822A1 (en) | 2010-04-15 |
ZA200903969B (en) | 2012-02-29 |
ES2398595T3 (es) | 2013-03-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |